Sonogashira cross-coupling reaction with 4-[18F]fluoroiodobenzene for rapid 18F-labelling of peptides

2015 ◽  
Vol 51 (18) ◽  
pp. 3838-3841 ◽  
Author(s):  
Jenilee D. Way ◽  
Cody Bergman ◽  
Frank Wuest

The study describes the Sonogashira cross-coupling reaction with 4-[18F]fluoroiodobenzene ([18F]FIB) as novel and efficient method for rapid labelling of peptides with the short-lived positron emitter fluorine-18.

2015 ◽  
Vol 13 (15) ◽  
pp. 4367-4373 ◽  
Author(s):  
Harish K. Potukuchi ◽  
Anatol P. Spork ◽  
Timothy J. Donohoe

The enolate cross coupling reaction is a highly efficient method for the de novo synthesis of aromatic rings.


Synthesis ◽  
2021 ◽  
Author(s):  
Yanghui Zhang ◽  
Bin Wan

AbstractAn efficient protocol for the palladium-catalyzed cross-coupling reaction of 2-iodobiphenyls with biphenylene has been developed through C–H activation. The reaction provides a simple and efficient method for the synthesis of unsymmetrically substituted tetra­phenylenes.


2021 ◽  
Author(s):  
Guiwen Hu ◽  
Ping Li ◽  
Zhiqiang Zhou ◽  
Fan Yang ◽  
Shijie Xu ◽  
...  

An efficient NBS-assisted palladium-catalyzed bromination/cross-coupling synthesis of 3-thiocyanindoles from 2-alkynyl arylazides with KSCN has been described.


Sign in / Sign up

Export Citation Format

Share Document