scholarly journals Structure activity relationship of 2-arylalkynyl-adenine derivatives as human A3 adenosine receptor antagonists

MedChemComm ◽  
2018 ◽  
Vol 9 (11) ◽  
pp. 1920-1932 ◽  
Author(s):  
Jinha Yu ◽  
Philip Mannes ◽  
Young-Hwan Jung ◽  
Antonella Ciancetta ◽  
Amelia Bitant ◽  
...  
Keyword(s):  
Adenosine Receptor ◽  
Structure Activity Relationship ◽  
Activity Relationship ◽  
Receptor Antagonists ◽  
Agonist Affinity ◽  
Structure Activity ◽  
Selective Antagonists ◽  
A3 Adenosine Receptor ◽  
Relationship Of ◽  
Adenine Derivatives

Adenines that incorporate known agonist affinity-enhancing substituents are A3AR-selective antagonists.

Structure–activity relationship studies of a new series of imidazo[2,1-f]purinones as potent and selective A3 adenosine receptor antagonists

2008 ◽  
Vol 16 (24) ◽  
pp. 10281-10294 ◽  
Author(s):  
Pier Giovanni Baraldi ◽  
Delia Preti ◽  
Mojgan Aghazadeh Tabrizi ◽  
Romeo Romagnoli ◽  
Giulia Saponaro ◽  
...  
Keyword(s):  
Adenosine Receptor ◽  
Structure Activity Relationship ◽  
Activity Relationship ◽  
Receptor Antagonists ◽  
Structure Activity ◽  
A3 Adenosine Receptor

ChemInform Abstract: Initial Structure-Activity Relationship of a Novel Class of Nonpeptidyl GnRH Receptor Antagonists: 2-Arylindoles.

ChemInform ◽  
2010 ◽  
Vol 32 (23) ◽  
pp. no-no
Author(s):  
Lin Chu ◽  
Jennifer E. Hutchins ◽  
Ann E. Weber ◽  
Jane-Ling Lo ◽  
Yi-Tien Yang ◽  
...  
Keyword(s):  
Structure Activity Relationship ◽  
Gnrh Receptor ◽  
Activity Relationship ◽  
Initial Structure ◽  
Receptor Antagonists ◽  
Structure Activity ◽  
Relationship Of
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