Synthesis and biological evaluation of structurally diverse α-conformationally restricted chalcones and related analogues

Casey J. Maguire; Graham J. Carlson; Jacob W. Ford; Tracy E. Strecker; Ernest Hamel; Mary Lynn Trawick; Kevin G. Pinney

doi:10.1039/c9md00127a

Synthesis and biological evaluation of structurally diverse α-conformationally restricted chalcones and related analogues

MedChemComm ◽

10.1039/c9md00127a ◽

2019 ◽

Vol 10 (8) ◽

pp. 1445-1456 ◽

Cited By ~ 3

Author(s):

Casey J. Maguire ◽

Graham J. Carlson ◽

Jacob W. Ford ◽

Tracy E. Strecker ◽

Ernest Hamel ◽

...

Keyword(s):

Biological Evaluation ◽

Cytotoxic Agents ◽

Conformationally Restricted ◽

Structural Analogues ◽

Synthesis And Biological Evaluation

Cyclic chalcones and structural analogues evaluated as cytotoxic agents.

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Synthesis and biological evaluation of new 3-(6-hydroxyindol-2-yl)-5-(Phenyl) pyridine or pyrazine V-Shaped molecules as kinase inhibitors and cytotoxic agents

European Journal of Medicinal Chemistry ◽

10.1016/j.ejmech.2011.08.048 ◽

2011 ◽

Vol 46 (11) ◽

pp. 5416-5434 ◽

Cited By ~ 34

Author(s):

Pamela Kassis ◽

Joanna Brzeszcz ◽

Valérie Bénéteau ◽

Olivier Lozach ◽

Laurent Meijer ◽

...

Keyword(s):

Kinase Inhibitors ◽

Biological Evaluation ◽

Cytotoxic Agents ◽

Synthesis And Biological Evaluation

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Synthesis and biological evaluation of 2-phenol-4-chlorophenyl-6-aryl pyridines as topoisomerase II inhibitors and cytotoxic agents

Bioorganic Chemistry ◽

10.1016/j.bioorg.2016.04.007 ◽

2016 ◽

Vol 66 ◽

pp. 145-159 ◽

Cited By ~ 3

Author(s):

Pritam Thapa ◽

Tara Man Kadayat ◽

Seojeong Park ◽

Somin Shin ◽

Til Bahadur Thapa Magar ◽

...

Keyword(s):

Topoisomerase Ii ◽

Biological Evaluation ◽

Cytotoxic Agents ◽

Topoisomerase Ii Inhibitors ◽

Synthesis And Biological Evaluation

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Design, synthesis, and biological evaluation of N-(4-substituted)-3-phenylisoxazolo[5,4–d]pyrimidin-4-amine derivatives as apoptosis-inducing cytotoxic agents

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/j.bmcl.2021.128294 ◽

2021 ◽

pp. 128294

Author(s):

Nikhil Baliram Gaikwad ◽

Sapana Bansode ◽

Alekhya mara ◽

Ramana Garise ◽

Nanduri Srinivas ◽

...

Keyword(s):

Biological Evaluation ◽

Cytotoxic Agents ◽

Design Synthesis ◽

Synthesis And Biological Evaluation

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ChemInform Abstract: Synthesis and Biological Evaluation of New 3-(6-Hydroxyindol-2-yl)-5-(phenyl) Pyridine or Pyrazine V-Shaped Molecules as Kinase Inhibitors and Cytotoxic Agents.

ChemInform ◽

10.1002/chin.201211125 ◽

2012 ◽

Vol 43 (11) ◽

pp. no-no

Author(s):

Jean-Yves Merour ◽

et al. et al.

Keyword(s):

Kinase Inhibitors ◽

Biological Evaluation ◽

Cytotoxic Agents ◽

Synthesis And Biological Evaluation

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Design, synthesis and biological evaluation of some novel N-arylpyrazole derivatives bearing the sulfonamide moiety as cytotoxic agents

Research on Chemical Intermediates ◽

10.1007/s11164-016-2620-x ◽

2016 ◽

Vol 43 (1) ◽

pp. 271-281 ◽

Cited By ~ 3

Author(s):

Xiaobo Duan ◽

Yingxing Wang ◽

Weipei Feng ◽

Yaxing Yang ◽

Hongyan Li ◽

...

Keyword(s):

Biological Evaluation ◽

Cytotoxic Agents ◽

Design Synthesis ◽

Synthesis And Biological Evaluation

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One Pot Single Step Synthesis and Biological Evaluation of Some Novel Bis(1,3,4-thiadiazole) Derivatives as Potential Cytotoxic Agents

Molecules ◽

10.3390/molecules21111532 ◽

2016 ◽

Vol 21 (11) ◽

pp. 1532 ◽

Cited By ~ 32

Author(s):

Sobhi Gomha ◽

Nabila Kheder ◽

Abdou Abdelhamid ◽

Yahia Mabkhot

Keyword(s):

Biological Evaluation ◽

Single Step ◽

Cytotoxic Agents ◽

One Pot ◽

Thiadiazole Derivatives ◽

Synthesis And Biological Evaluation

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Green Synthesis and Biological Evaluation of New Di-α-aminophosphonate Derivatives as Cytotoxic Agents

Archiv der Pharmazie ◽

10.1002/ardp.201300249 ◽

2013 ◽

Vol 346 (12) ◽

pp. 851-859 ◽

Cited By ~ 4

Author(s):

Kunda Uma Maheswara Rao ◽

Sim Namkoong ◽

Hwan-Chul Yu ◽

Junsoo Park ◽

Chan-Moon Chung ◽

...

Keyword(s):

Green Synthesis ◽

Biological Evaluation ◽

Cytotoxic Agents ◽

Synthesis And Biological Evaluation

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Synthesis and Biological Evaluation of 6-[(1R)-1-Hydroxyethyl]-2,4a(R),6(S),8a(R)-tetrahydropyrano-[3,2-b]-pyran-2-one and Structural Analogues of the Putative Structure of Diplopyrone

The Journal of Organic Chemistry ◽

10.1021/acs.joc.8b02490 ◽

2018 ◽

Vol 84 (2) ◽

pp. 666-678 ◽

Cited By ~ 7

Author(s):

Nicholas C. Lazzara ◽

Robert J. Rosano ◽

Purav P. Vagadia ◽

Matthew T. Giovine ◽

Mark W. Bezpalko ◽

...

Keyword(s):

Biological Evaluation ◽

Structural Analogues ◽

Synthesis And Biological Evaluation

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Parallel Synthesis and Biological Evaluation of 5,6,7,8-Tetrahydrobenzothieno[2,3-d]pyrimidin-4(3H)-one Cytotoxic Agents Selective for p21-Deficient Cells.

ChemInform ◽

10.1002/chin.200605230 ◽

2006 ◽

Vol 37 (5) ◽

Author(s):

Lee D. Jennings ◽

Scott L. Kincaid ◽

Yanong D. Wang ◽

Girija Krishnamurthy ◽

Carl F. Beyer ◽

...

Keyword(s):

Biological Evaluation ◽

Parallel Synthesis ◽

Cytotoxic Agents ◽

Synthesis And Biological Evaluation

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Synthesis and biological evaluation of T-OA analogues as the cytotoxic agents

Research on Chemical Intermediates ◽

10.1007/s11164-014-1737-z ◽

2014 ◽

Vol 41 (9) ◽

pp. 6257-6269 ◽

Cited By ~ 7

Author(s):

Kuo Xu ◽

Xin Xu ◽

Fuhao Chu ◽

Mina Wang ◽

Penglong Wang ◽

...

Keyword(s):

Biological Evaluation ◽

Cytotoxic Agents ◽

Synthesis And Biological Evaluation

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