scholarly journals Discovery of 2,4-thiazolidinedione-tethered coumarins as novel selective inhibitors for carbonic anhydrase IX and XII isoforms

2022 ◽  
Vol 37 (1) ◽  
pp. 531-541
Author(s):  
Wagdy M. Eldehna ◽  
Mohammed S. Taghour ◽  
Tarfah Al-Warhi ◽  
Alessio Nocentini ◽  
Mostafa M. Elbadawi ◽  
...  
Keyword(s):  
Carbonic Anhydrase ◽  
Carbonic Anhydrase Ix ◽  
Selective Inhibitors

Metallacarborane Sulfamides: Unconventional, Specific, and Highly Selective Inhibitors of Carbonic Anhydrase IX

2019 ◽  
Vol 62 (21) ◽  
pp. 9560-9575 ◽  
Author(s):  
Bohumír Grüner ◽  
Jiří Brynda ◽  
Viswanath Das ◽  
Václav Šícha ◽  
Jana Štěpánková ◽  
...  
Keyword(s):  
Carbonic Anhydrase ◽  
Carbonic Anhydrase Ix ◽  
Selective Inhibitors

scholarly journals α,γ-Diketocarboxylic Acids and Their Esters Act as Carbonic Anhydrase IX and XII Selective Inhibitors

2019 ◽  
Vol 10 (4) ◽  
pp. 661-665 ◽  
Author(s):  
Alessio Nocentini ◽  
Alessia Lucidi ◽  
Francesca Perut ◽  
Annamaria Massa ◽  
Daniela Tomaselli ◽  
...  
Keyword(s):  
Carbonic Anhydrase ◽  
Carbonic Anhydrase Ix ◽  
Selective Inhibitors

scholarly journals Cobalt Bis(dicarbollide) Alkylsulfonamides: Potent and Highly Selective Inhibitors of Tumor Specific Carbonic Anhydrase IX

ChemPlusChem ◽  
2020 ◽  
Author(s):  
Bohumír Grüner ◽  
Michael Kugler ◽  
Suzan El Anwar ◽  
Josef Holub ◽  
Jan Nekvinda ◽  
...  
Keyword(s):  
Carbonic Anhydrase ◽  
Carbonic Anhydrase Ix ◽  
Selective Inhibitors

Discovery and Characterization of Novel Selective Inhibitors of Carbonic Anhydrase IX

2014 ◽  
Vol 57 (22) ◽  
pp. 9435-9446 ◽  
Author(s):  
Virginija Dudutienė ◽  
Jurgita Matulienė ◽  
Alexey Smirnov ◽  
David D. Timm ◽  
Asta Zubrienė ◽  
...  
Keyword(s):  
Carbonic Anhydrase ◽  
Carbonic Anhydrase Ix ◽  
Selective Inhibitors

Sulfonamido carboranes as highly selective inhibitors of cancer-specific carbonic anhydrase IX

2020 ◽  
Vol 200 ◽  
pp. 112460 ◽  
Author(s):  
Jana Dvořanová ◽  
Michael Kugler ◽  
Josef Holub ◽  
Václav Šícha ◽  
Viswanath Das ◽  
...  
Keyword(s):  
Carbonic Anhydrase ◽  
Carbonic Anhydrase Ix ◽  
Selective Inhibitors

scholarly journals Novel benzoyl thioureido benzene sulfonamides as highly potent and selective inhibitors of carbonic anhydrase IX: optimization and bioactive studies

MedChemComm ◽  
2018 ◽  
Vol 9 (12) ◽  
pp. 2100-2105 ◽  
Author(s):  
Li Liu ◽  
Wanqi Wang ◽  
Jin Huang ◽  
Zhenjiang Zhao ◽  
Honglin Li ◽  
...  
Keyword(s):  
Carbonic Anhydrase ◽  
Inhibitory Activity ◽  
Carbonic Anhydrase Ix ◽  
Selective Inhibitors ◽  
Ca Ix

Novel benzoyl thioureido benzene sulfonamides as CA IX inhibitors such as 6a displayed inhibitory activity against CA IX with an IC50 value of 0.48 nM and about 1500-fold selectivity over CA II were reported.

Cobalt Bis(dicarbollide) Alkylsulfonamides: Potent and Highly Selective Inhibitors of Tumor Specific Carbonic Anhydrase IX

ChemPlusChem ◽  
2020 ◽  
Author(s):  
Bohumír Grüner ◽  
Michael Kugler ◽  
Suzan El Anwar ◽  
Josef Holub ◽  
Jan Nekvinda ◽  
...  
Keyword(s):  
Carbonic Anhydrase ◽  
Carbonic Anhydrase Ix ◽  
Selective Inhibitors
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