D.8 - BEHAVIORAL PROFILE OF CARIPRAZINE, A DOPAMINE D3/D2 RECEPTOR PARTIAL AGONIST NOVEL ANTIPSYCHOTIC CANDIDATE, IN RODENT MODELS OF SCHIZOPHRENIA, MANIA, DEPRESSION AND COGNITION

2013 ◽  
Vol 24 ◽  
pp. e39
Author(s):  
István Gyertyán ◽  
Béla Kiss ◽  
Nika Adham
Keyword(s):  
Partial Agonist ◽  
D2 Receptor ◽  
Rodent Models ◽  
Behavioral Profile ◽  
Dopamine D3 ◽  
Novel Antipsychotic

DOPAMINE D3 RECEPTOR OCCUPANCY AND D3 RECEPTOR-MEDIATED ACTIONS OF CARIPRAZINE, A DOPAMINE D3/D2 RECEPTOR PARTIAL AGONIST ANTIPSYCHOTIC CANDIDATE

2014 ◽  
Vol 153 ◽  
pp. S23
Author(s):  
Ashok Rakhit ◽  
Suresh Durgam ◽  
Nika Adham ◽  
István Gyertyán ◽  
Béla Kiss ◽  
...  
Keyword(s):  
Partial Agonist ◽  
D2 Receptor ◽  
Receptor Occupancy ◽  
Dopamine D3 Receptor ◽  
D3 Receptor ◽  
Dopamine D3

Pharmacology of aripiprazole, a novel antipsychotic: dopamine D2 receptor partial agonist

2004 ◽  
Vol 19 (3) ◽  
pp. 190
Author(s):  
Tetsuro Kikuchi ◽  
Stark Arlene ◽  
Frank Yocca ◽  
Yoshihiro Tadori ◽  
Tsuyoshi Hirose ◽  
...  
Keyword(s):  
Dopamine D2 Receptor ◽  
Partial Agonist ◽  
D2 Receptor ◽  
Dopamine D2 ◽  
Novel Antipsychotic

Cariprazine (RGH-188), a D3-preferring dopamine D3/D2 receptor partial agonist antipsychotic candidate demonstrates anti-abuse potential in rats

2012 ◽  
Vol 226 (2) ◽  
pp. 285-293 ◽  
Author(s):  
V. Román ◽  
I. Gyertyán ◽  
K. Sághy ◽  
B. Kiss ◽  
Zs. Szombathelyi
Keyword(s):  
Partial Agonist ◽  
D2 Receptor ◽  
Abuse Potential ◽  
Dopamine D3

Pharmacology of human dopamine D3 receptor expressed in a mammalian cell line: comparison with D2 receptor

1992 ◽  
Vol 225 (4) ◽  
pp. 331-337 ◽  
Author(s):  
Pierre Sokoloff ◽  
Marc Andrieux ◽  
Roger Besançon ◽  
Catherine Pilon ◽  
Marie-Pascale Martres ◽  
...  
Keyword(s):  
Cell Line ◽  
Mammalian Cell ◽  
D2 Receptor ◽  
Dopamine D3 Receptor ◽  
D3 Receptor ◽  
Mammalian Cell Line ◽  
Dopamine D3

Characterization of aripiprazole partial agonist activity at human dopamine D3 receptors

2008 ◽  
Vol 597 (1-3) ◽  
pp. 27-33 ◽  
Author(s):  
Yoshihiro Tadori ◽  
Robert A. Forbes ◽  
Robert D. McQuade ◽  
Tetsuro Kikuchi
Keyword(s):  
Partial Agonist ◽  
Agonist Activity ◽  
Dopamine D3 Receptors ◽  
D3 Receptors ◽  
Partial Agonist Activity ◽  
Dopamine D3
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