SR 141716A Acts as an Inverse Agonist to Increase Neuronal Voltage-Dependent Ca2+ Currents by Reversal of Tonic CB1 Cannabinoid Receptor Activity

Sr 141716A ◽

Voltage Dependent

The CB1 cannabinoid receptor antagonist SR 141716A affects A9 dopamine neuronal activity in the rat

Neuroreport ◽

10.1097/00001756-199507100-00015 ◽

1995 ◽

Vol 6 (10) ◽

pp. 1421-1425 ◽

Cited By ~ 35

Author(s):

Christiane Gueudet ◽

Vincent Santucci ◽

Murielle Rinaldi-Carmona ◽

Philippe Soubrié ◽

Gérard Le Fur

Keyword(s):

Receptor Antagonist ◽

Neuronal Activity ◽

Cannabinoid Receptor ◽

SR 141716A, a CB1 cannabinoid receptor antagonist, potentiates the locomotor stimulant effects of amphetamine and apomorphine

Behavioural Pharmacology ◽

10.1097/00008877-199907000-00010 ◽

1999 ◽

Vol 10 (4) ◽

pp. 429-432 ◽

Cited By ~ 40

Author(s):

J. M. Masserano ◽

F. Karoum ◽

R. J. Wyatt

Keyword(s):

Receptor Antagonist ◽

Cannabinoid Receptor ◽

Acute administration of the CB1 cannabinoid receptor antagonist SR 141716A induces anxiety-like responses in the rat

Neuroreport ◽

10.1097/00001756-199701200-00023 ◽

1997 ◽

Vol 8 (2) ◽

pp. 491-496 ◽

Cited By ~ 208

Author(s):

Miguel Navarro ◽

Elena Hernández ◽

Raúl M. Muñoz ◽

Ignacio del Arco ◽

María Angeles Villanúa ◽

...

Keyword(s):

Receptor Antagonist ◽

Cannabinoid Receptor ◽

Acute Administration ◽

CB1 Cannabinoid Receptor Activity Is Modulated by the Cannabinoid Receptor Interacting Protein CRIP 1a

Molecular Pharmacology ◽

10.1124/mol.107.039263 ◽

2007 ◽

Vol 72 (6) ◽

pp. 1557-1566 ◽

Cited By ~ 75

Author(s):

Jason L. Niehaus ◽

Yunguang Liu ◽

Kathleen T. Wallis ◽

Michaela Egertová ◽

Sheela G. Bhartur ◽

...

Keyword(s):

Cannabinoid Receptor ◽

Receptor Activity ◽

Interacting Protein ◽

The interactive effects of verapamil and CB1 cannabinoid receptor antagonist/inverse agonist, AM251 on passive avoidance learning and memory in rat

Behavioural Pharmacology ◽

10.1097/fbp.0000000000000638 ◽

2021 ◽

Vol Publish Ahead of Print ◽

Author(s):

Seyed Asaad Karimi ◽

Mariam Noorbakhsh ◽

Hamidreza Komaki ◽

Mohammad Reza Nikoo ◽

Parisa Hasanein ◽

...

Keyword(s):

Passive Avoidance ◽

Receptor Antagonist ◽

Learning And Memory ◽

Avoidance Learning ◽

Cannabinoid Receptor ◽

Inverse Agonist ◽

Passive Avoidance Learning ◽

Interactive Effects ◽

Arousal-enhancing properties of the CB1 cannabinoid receptor antagonist SR 141716A in rats as assessed by electroencephalographic spectral and sleep-waking cycle analysis

Life Sciences ◽

10.1016/0024-3205(95)02319-4 ◽

1996 ◽

Vol 58 (6) ◽

pp. PL103-PL110 ◽

Cited By ~ 107

Author(s):

Vincent Santucci ◽

Jean-jacques Storme ◽

Philippe Soubrié ◽

Gérard Le Fur

Keyword(s):

Receptor Antagonist ◽

Cannabinoid Receptor ◽

Effects of the CB1 cannabinoid receptor inverse agonist AM251 on food intake and body weight in mice lacking μ-opioid receptors

Brain Research ◽

10.1016/j.brainres.2006.06.006 ◽

2006 ◽

Vol 1108 (1) ◽

pp. 176-178 ◽

Cited By ~ 21

Author(s):

Richard Z. Chen ◽

Andrea Frassetto ◽

Tung M. Fong

Keyword(s):

Body Weight ◽

Food Intake ◽

Opioid Receptors ◽

Cannabinoid Receptor ◽

Inverse Agonist ◽

Μ Opioid Receptors ◽

Receptor Inverse Agonist

Inverse agonist properties of N-(piperidin-1-yl)-5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl-1H-pyrazole-3-carboxamide HCl (SR141716A) and 1-(2-chlorophenyl)-4-cyano-5-(4-methoxyphenyl)-1H-pyrazole-3-carboxylic acid phenylamide (CP-272871) for the CB1 cannabinoid receptor

Biochemical Pharmacology ◽

10.1016/s0006-2952(00)00447-0 ◽

2000 ◽

Vol 60 (9) ◽

pp. 1315-1323 ◽

Cited By ~ 70

Author(s):

Justin P. Meschler ◽

Dennis M. Kraichely ◽

Gerald H. Wilken ◽

Allyn C. Howlett

Keyword(s):

Carboxylic Acid ◽

Cannabinoid Receptor ◽

Inverse Agonist ◽

Characterization and distribution of binding sites for [3H]-SR 141716A, a selective brain (CB1) cannabinoid receptor antagonist, in rodent brain

Life Sciences ◽

10.1016/0024-3205(96)00085-9 ◽

1996 ◽

Vol 58 (15) ◽

pp. 1239-1247 ◽

Cited By ~ 89

Author(s):

Murielle Rinaldi-Carmona ◽

Françoise Pialot ◽

Christian Congy ◽

Elsa Redon ◽

Francis Barth ◽

...

Keyword(s):

Receptor Antagonist ◽

Binding Sites ◽

Cannabinoid Receptor ◽

Rodent Brain ◽

Falcarinol (Panaxynol) is a CB1 cannabinoid receptor antagonist and induces pro-allergic effects in skin

Planta Medica ◽

10.1055/s-0029-1234271 ◽

2009 ◽

Vol 75 (09) ◽

Author(s):

J Gertsch ◽

M Leonti ◽

L Casu ◽

F Cottiglia ◽

S Raduner ◽

...

Keyword(s):

Receptor Antagonist ◽

Cannabinoid Receptor ◽