Cloning, Expression, and Pharmacological Characterization of a Novel Human Histamine Receptor

2001 ◽  
Vol 59 (3) ◽  
pp. 434-441 ◽  
Author(s):  
Yuan Zhu ◽  
David Michalovich ◽  
Hsiao-Ling Wu ◽  
K. B. Tan ◽  
George M. Dytko ◽  
...  
Keyword(s):  
Histamine Receptor ◽  
Pharmacological Characterization ◽  
Human Histamine

scholarly journals Design and pharmacological characterization of VUF14480, a covalent partial agonist that interacts with cysteine 983.36of the human histamine H4receptor

2013 ◽  
Vol 170 (1) ◽  
pp. 89-100 ◽  
Author(s):  
S Nijmeijer ◽  
H Engelhardt ◽  
S Schultes ◽  
A C van de Stolpe ◽  
V Lusink ◽  
...  
Keyword(s):  
Partial Agonist ◽  
Pharmacological Characterization ◽  
Human Histamine

Cloning and Pharmacological Characterization of a Fourth Histamine Receptor (H4) Expressed in Bone Marrow

2001 ◽  
Vol 59 (3) ◽  
pp. 420-426 ◽  
Author(s):  
Changlu Liu ◽  
Xiao-Jun Ma ◽  
Xiaoxia Jiang ◽  
Sandy J. Wilson ◽  
Claudia L. Hofstra ◽  
...  
Keyword(s):  
Bone Marrow ◽  
Histamine Receptor ◽  
Pharmacological Characterization

Pharmacological characterization of the histamine uptake system in HL-60 human promyelocytic leukemia cells

1986 ◽  
Vol 6 (4) ◽  
pp. 403-407 ◽  
Author(s):  
Christian Gespach ◽  
Noel Marrec ◽  
Jean-Pierre Abita
Keyword(s):  
Peripheral Blood ◽  
Histamine Receptor ◽  
Promyelocytic Leukemia ◽  
Leukemia Cells ◽  
Uptake System ◽  
Active Process ◽  
Pharmacological Characterization ◽  
H2 Receptor ◽  
Histamine Uptake

Serotonin and histamine H1, H2 receptor agonists or antagonists inhibited [3H]histamine uptake by HL-60 cells, according to the following order of potency: impromidine >4-MH>histamine>AET>PEA and: cimetidine, histamine>diphenhydramine, serotonin. It is concluded that histamine uptake by HL-60 cells was specifically controlled by the H2 type histamine receptor and that this active process might be involved in pathophysiological regulations in leukemic and normal granulocytic precursors and in the control of histamine levels in peripheral blood and tissues in man.

Molecular Cloning and Characterization of a New Human Histamine Receptor, HH4R

2000 ◽  
Vol 279 (2) ◽  
pp. 615-620 ◽  
Author(s):  
Takao Nakamura ◽  
Hiraku Itadani ◽  
Yusuke Hidaka ◽  
Masataka Ohta ◽  
Kenichi Tanaka
Keyword(s):  
Molecular Cloning ◽  
Histamine Receptor ◽  
Human Histamine
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