SYNTHESIS, CRYSTAL STRUCTURE, AND BIOLOGICAL  EVALUATION OF (E)-1-(4-(4-BROMOBENZYL)PIPERAZIN-1-YL)-
3-(4-CHLOROPHENYL)PROP-2-EN-1-ONE

L. -Y. Chen; C. -Z. Yang; Y. Xu; C. -Y. Qi; Y. Zhong; B. Wu

doi:10.1134/s002247662103015x

SYNTHESIS, CRYSTAL STRUCTURE, AND BIOLOGICAL EVALUATION OF (E)-1-(4-(4-BROMOBENZYL)PIPERAZIN-1-YL)- 3-(4-CHLOROPHENYL)PROP-2-EN-1-ONE

Journal of Structural Chemistry ◽

10.1134/s002247662103015x ◽

2021 ◽

Vol 62 (3) ◽

pp. 481-490

Author(s):

L. -Y. Chen ◽

C. -Z. Yang ◽

Y. Xu ◽

C. -Y. Qi ◽

Y. Zhong ◽

...

Keyword(s):

Crystal Structure ◽

Biological Evaluation

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2-methylpyridinium 5-(2,4-dinitrophenyl)-6-oxo-2-thioxo-1,2,3,6-tetrahydropyrimidin-4-olate: synthesis, crystal structure, and biological evaluation

Журнал структурной химии ◽

10.15372/jsc20160519 ◽

2016 ◽

Keyword(s):

Crystal Structure ◽

Biological Evaluation

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Synthesis, crystal structure and biological evaluation of novel 2-phenylthiazole derivatives as multi-targeting agents to treat Alzheimer’s disease

Journal of Chemical Research ◽

10.3184/174751917x15070513875024 ◽

2017 ◽

Keyword(s):

Crystal Structure ◽

Alzheimer’S Disease ◽

Alzheimer's Disease ◽

Biological Evaluation

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Discovery of new phenyl sulfonyl-pyrimidine carboxylate derivatives as the potential multi-target drugs with effective anti-Alzheimer’s action: Design, synthesis, crystal structure and in-vitro biological evaluation

European Journal of Medicinal Chemistry ◽

10.1016/j.ejmech.2021.113224 ◽

2021 ◽

Vol 215 ◽

pp. 113224

Author(s):

Shoaib Manzoor ◽

Santosh Kumar Prajapati ◽

Shreyasi Majumdar ◽

Kausar Raza ◽

Moustafa T. Gabr ◽

...

Keyword(s):

Crystal Structure ◽

Biological Evaluation ◽

Design Synthesis

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Structure-Based Design of Highly Selective β-Secretase Inhibitors: Synthesis, Biological Evaluation, and Protein–Ligand X-ray Crystal Structure

Journal of Medicinal Chemistry ◽

10.1021/jm3008823 ◽

2012 ◽

Vol 55 (21) ◽

pp. 9195-9207 ◽

Cited By ~ 23

Author(s):

Arun K. Ghosh ◽

Kalapala Venkateswara Rao ◽

Navnath D. Yadav ◽

David D. Anderson ◽

Navnath Gavande ◽

...

Keyword(s):

Crystal Structure ◽

Biological Evaluation ◽

X Ray

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Synthesis, crystal structure, biological evaluation, electronic aspects of hydrogen bonds, and QSAR studies of some new N-(substituted phenylurea) diazaphosphore derivatives as anticancer agents

Medicinal Chemistry Research ◽

10.1007/s00044-016-1527-9 ◽

2016 ◽

Vol 25 (4) ◽

pp. 769-789 ◽

Cited By ~ 5

Author(s):

Niloufar Dorosti ◽

Bahram Delfan ◽

Khodayar Gholivand ◽

Ali Asghar Ebrahimi Valmoozi

Keyword(s):

Crystal Structure ◽

Hydrogen Bonds ◽

Anticancer Agents ◽

Biological Evaluation ◽

Qsar Studies

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1,2,4-triazole-3-thione Schiff bases compounds: Crystal structure, hirshfeld surface analysis, DFT studies and biological evaluation

Journal of Molecular Structure ◽

10.1016/j.molstruc.2020.128591 ◽

2020 ◽

Vol 1219 ◽

pp. 128591 ◽

Cited By ~ 2

Author(s):

Shaojie Wu ◽

Le Qi ◽

Yinghui Ren ◽

Haixia Ma

Keyword(s):

Crystal Structure ◽

Surface Analysis ◽

Schiff Bases ◽

Biological Evaluation ◽

Hirshfeld Surface ◽

Hirshfeld Surface Analysis ◽

Dft Studies

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Synthesis, crystal structure, DFT studies and biological evaluation of N-benzamido derivatives of oxahexacycloundecyl amines: A case of enantiomerism leading to molecular disorder

Journal of Molecular Structure ◽

10.1016/j.molstruc.2020.128248 ◽

2020 ◽

Vol 1215 ◽

pp. 128248

Author(s):

Rajan Sharma ◽

Jacques Joubert ◽

Hong Su ◽

Mino R. Caira ◽

Sarel F. Malan

Keyword(s):

Crystal Structure ◽

Biological Evaluation ◽

Dft Studies ◽

Derivatives Of

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Design, synthesis and biological evaluation of novel human monoamine oxidase B inhibitors based on a fragment in an X-ray crystal structure

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/j.bmcl.2019.02.008 ◽

2019 ◽

Vol 29 (8) ◽

pp. 1012-1018 ◽

Cited By ~ 5

Author(s):

Kai Cheng ◽

Shiyu Li ◽

Xiao Lv ◽

Yongbin Tian ◽

Haiyan Kong ◽

...

Keyword(s):

Crystal Structure ◽

Monoamine Oxidase ◽

Biological Evaluation ◽

Monoamine Oxidase B ◽

Design Synthesis ◽

X Ray ◽

Synthesis And Biological Evaluation

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A multifunctional therapeutic approach: Synthesis, biological evaluation, crystal structure and molecular docking of diversified 1H-pyrazolo[3,4-b]pyridine derivatives against Alzheimer's disease

European Journal of Medicinal Chemistry ◽

10.1016/j.ejmech.2019.04.038 ◽

2019 ◽

Vol 175 ◽

pp. 2-19 ◽

Cited By ~ 10

Author(s):

Tarana Umar ◽

Shruti Shalini ◽

Md Kausar Raza ◽

Siddharth Gusain ◽

Jitendra Kumar ◽

...

Keyword(s):

Crystal Structure ◽

Alzheimer’S Disease ◽

Alzheimer's Disease ◽

Molecular Docking ◽

Therapeutic Approach ◽

Biological Evaluation ◽

Pyridine Derivatives

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A novel schiff base ligand and its copper complex: Synthesis, characterization, X-ray crystal structure and biological evaluation

Journal of Molecular Structure ◽

10.1016/j.molstruc.2020.129395 ◽

2021 ◽

Vol 1226 ◽

pp. 129395

Author(s):

Tahere Kondori ◽

Niloufar Akbarzadeh-T ◽

Mahboubeh Fazli ◽

Behrouz Mir ◽

Michal Dušek ◽

...

Keyword(s):

Crystal Structure ◽

Schiff Base ◽

Schiff Base Ligand ◽

Copper Complex ◽

Biological Evaluation ◽

X Ray

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