De-novo design, synthesis and evaluation of novel 6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline derivatives as HIV-1 reverse transcriptase inhibitors

Design Synthesis ◽

Hiv 1

De novo design and in-silico studies of novel 1-phenyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic acid derivatives as HIV-1 reverse transcriptase inhibitors

Medicinal Chemistry Research ◽

10.1007/s00044-014-0945-9 ◽

2014 ◽

Vol 23 (8) ◽

pp. 3662-3670 ◽

Cited By ~ 9

Author(s):

Ashok Penta ◽

Subhash Chander ◽

S. Ganguly ◽

S. Murugesan

Keyword(s):

Carboxylic Acid ◽

Reverse Transcriptase ◽

In Silico ◽

De Novo ◽

De Novo Design ◽

In Silico Studies ◽

Hiv 1

Arylazolylthioacetanilide. Part 11: Design, Synthesis and Biological Evaluation of 1,2,4-triazole Thioacetanilide Derivatives as Novel Non-nucleoside HIV-1 Reverse Transcriptase Inhibitors

Medicinal Chemistry ◽

10.2174/1573406411309070010 ◽

2013 ◽

Vol 9 (7) ◽

pp. 968-973 ◽

Cited By ~ 9

Author(s):

Zhenyu Li ◽

Yuan Cao ◽

Peng Zhan ◽

Christophe Pannecouque ◽

Jan Balzarini ◽

...

Keyword(s):

Reverse Transcriptase ◽

Biological Evaluation ◽

Design Synthesis ◽

Hiv 1

Design, synthesis, and biological evaluation of novel 5-Alkyl-6-Adamantylmethylpyrimidin-4(3H)-ones as HIV-1 non-nucleoside reverse-transcriptase inhibitors

Chemical Biology & Drug Design ◽

10.1111/cbdd.12765 ◽

2016 ◽

Vol 88 (3) ◽

pp. 380-385 ◽

Cited By ~ 2

Author(s):

Wenxin Li ◽

Boshi Huang ◽

Dongwei Kang ◽

Erik De Clercq ◽

Dirk Daelemans ◽

...

Keyword(s):

Reverse Transcriptase ◽

Biological Evaluation ◽

Design Synthesis ◽

Hiv 1

Design, Synthesis, and Biological Evaluation of Novel 2H-Pyran-2-one Derivatives as Potential HIV-1 Reverse Transcriptase Inhibitors

Archiv der Pharmazie ◽

10.1002/ardp.201400235 ◽

2014 ◽

Vol 348 (1) ◽

pp. 23-33 ◽

Cited By ~ 11

Author(s):

Andrea Defant ◽

Ines Mancini ◽

Rossella Tomazzolli ◽

Jan Balzarini

Keyword(s):

Reverse Transcriptase ◽

Biological Evaluation ◽

Design Synthesis ◽

Hiv 1

Design, Synthesis and Biological Evaluations of Novel Oxindoles as HIV-1 Non-Nucleoside Reverse Transcriptase Inhibitors. Part 1.

ChemInform ◽

10.1002/chin.200629096 ◽

2006 ◽

Vol 37 (29) ◽

Author(s):

Tao Jiang ◽

Kelli L. Kuhen ◽

Karen Wolff ◽

Hong Yin ◽

Kimberly Bieza ◽

...

Keyword(s):

Reverse Transcriptase ◽

Design Synthesis ◽

Hiv 1

Newer aminopyrimidinimino isatin analogues as non-nucleoside HIV-1 reverse transcriptase inhibitors for HIV and other opportunistic infections of AIDS: design, synthesis and biological evaluation

Il Farmaco ◽

10.1016/j.farmac.2005.03.005 ◽

2005 ◽

Vol 60 (5) ◽

pp. 377-384 ◽

Cited By ~ 27

Author(s):

D. Sriram ◽

T.R. Bal ◽

P. Yogeeswari

Keyword(s):

Reverse Transcriptase ◽

Opportunistic Infections ◽

Biological Evaluation ◽

Design Synthesis ◽

Hiv 1

Design, Synthesis, and Biological Evaluation of 1-[(2-Benzyloxyl/alkoxyl)methyl]-5-halo-6-aryluracils as Potent HIV-1 Non-nucleoside Reverse Transcriptase Inhibitors with an Improved Drug Resistance Profile

Journal of Medicinal Chemistry ◽

10.1021/jm201506e ◽

2012 ◽

Vol 55 (5) ◽

pp. 2242-2250 ◽

Cited By ~ 26

Author(s):

Xiaowei Wang ◽

Jianfang Zhang ◽

Yang Huang ◽

Ruiping Wang ◽

Liang Zhang ◽

...

Keyword(s):

Drug Resistance ◽

Reverse Transcriptase ◽

Biological Evaluation ◽

Design Synthesis ◽

Resistance Profile ◽

Drug Resistance Profile ◽

Hiv 1

Newer Aminopyrimidinimino Isatin Analogues as Non-Nucleoside HIV-1 Reverse Transcriptase Inhibitors for HIV and Other Opportunistic Infections of AIDS: Design, Synthesis and Biological Evaluation.

ChemInform ◽

10.1002/chin.200539145 ◽

2005 ◽

Vol 36 (39) ◽

Author(s):

D. Sriram ◽

T. R. Bal ◽

P. Yogeeswari

Keyword(s):

Reverse Transcriptase ◽

Opportunistic Infections ◽

Biological Evaluation ◽

Design Synthesis ◽

Hiv 1

Design, synthesis, docking studies and biological screening of 2-thiazolyl substituted -2,3-dihydro-1H-naphtho[1,2-e][1,3]oxazines as potent HIV-1 reverse transcriptase inhibitors

European Journal of Medicinal Chemistry ◽

10.1016/j.ejmech.2018.07.067 ◽

2018 ◽

Vol 157 ◽

pp. 310-319 ◽

Cited By ~ 8

Author(s):

Rakhi Gawali ◽

Jay Trivedi ◽

Sujit Bhansali ◽

Raghunath Bhosale ◽

Dhiman Sarkar ◽

...

Keyword(s):

Reverse Transcriptase ◽

Docking Studies ◽

Biological Screening ◽

Design Synthesis ◽

Hiv 1

Design, synthesis and biological evaluations of novel oxindoles as HIV-1 non-nucleoside reverse transcriptase inhibitors. Part I

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/j.bmcl.2006.01.073 ◽

2006 ◽

Vol 16 (8) ◽

pp. 2105-2108 ◽

Cited By ~ 150

Author(s):

Tao Jiang ◽

Kelli L. Kuhen ◽

Karen Wolff ◽

Hong Yin ◽

Kimberly Bieza ◽

...

Keyword(s):

Reverse Transcriptase ◽

Design Synthesis ◽

Hiv 1