Pharmacophore Modeling and 3D QSAR Studies of Novel Human Carbonic Anhydrase IX Inhibitors

2013 ◽  
Vol 10 (9) ◽  
pp. 808-816
Author(s):  
Kalyan Sethi ◽  
Saurabh Verma
Keyword(s):  
Carbonic Anhydrase ◽  
3D Qsar ◽  
Pharmacophore Modeling ◽  
Carbonic Anhydrase Ix ◽  
Qsar Studies ◽  
Human Carbonic Anhydrase

Design and Synthesis of Quinazolinone Derivatives as Anti-inflammatory Agents: Pharmacophore Modeling and 3D QSAR Studies

2014 ◽  
Vol 10 (7) ◽  
pp. 711-723 ◽  
Author(s):  
P. Chaitanya ◽  
G. Reddy ◽  
G. Varun ◽  
L.M. Srikanth ◽  
V.V.S.R. Prasad ◽  
...  
Keyword(s):  
3D Qsar ◽  
Pharmacophore Modeling ◽  
Qsar Studies ◽  
Design And Synthesis ◽  
Anti Inflammatory ◽  
Quinazolinone Derivatives

Pharmacophore modeling, virtual screening, and 3D-QSAR studies on a series of non-steroidal aromatase inhibitors

2014 ◽  
Vol 24 (5) ◽  
pp. 1901-1915 ◽  
Author(s):  
Huiding Xie ◽  
Kaixiong Qiu ◽  
Xiaoguang Xie
Keyword(s):  
Virtual Screening ◽  
Aromatase Inhibitors ◽  
3D Qsar ◽  
Pharmacophore Modeling ◽  
Qsar Studies ◽  
Steroidal Aromatase Inhibitors

Design, synthesis and biological evaluation of novel pyridine-thiazolidinone derivatives as anticancer agents: Targeting human carbonic anhydrase IX

2018 ◽  
Vol 144 ◽  
pp. 544-556 ◽  
Author(s):  
Mohammad Fawad Ansari ◽  
Danish Idrees ◽  
Md. Imtaiyaz Hassan ◽  
Kamal Ahmad ◽  
Fernando Avecilla ◽  
...  
Keyword(s):  
Carbonic Anhydrase ◽  
Anticancer Agents ◽  
Biological Evaluation ◽  
Carbonic Anhydrase Ix ◽  
Design Synthesis ◽  
Human Carbonic Anhydrase ◽  
Synthesis And Biological Evaluation

Abstract P038: Identification and functional evaluation of monoclonal antibodies specifically targeting human Carbonic Anhydrase IX

2022 ◽  
Author(s):  
Anne E. G. Lenferink ◽  
Jason Baardsnes ◽  
Traian Sulea ◽  
Cunle Wu ◽  
Maurizio Acchione ◽  
...  
Keyword(s):  
Monoclonal Antibodies ◽  
Carbonic Anhydrase ◽  
Carbonic Anhydrase Ix ◽  
Functional Evaluation ◽  
Human Carbonic Anhydrase

Discovery of new 2, 5-disubstituted 1,3-selenazoles as selective human carbonic anhydrase IX inhibitors with potent anti-tumor activity

2018 ◽  
Vol 157 ◽  
pp. 1214-1222 ◽  
Author(s):  
Andrea Angeli ◽  
Elena Trallori ◽  
Marta Ferraroni ◽  
Lorenzo Di Cesare Mannelli ◽  
Carla Ghelardini ◽  
...  
Keyword(s):  
Carbonic Anhydrase ◽  
Carbonic Anhydrase Ix ◽  
Human Carbonic Anhydrase ◽  
Anti Tumor Activity

scholarly journals Novel thiazolidinone-containing compounds, without the well-known sulphonamide zinc-binding group acting as human carbonic anhydrase IX inhibitors

2018 ◽  
Vol 33 (1) ◽  
pp. 1299-1308 ◽  
Author(s):  
Özlen Güzel-Akdemir ◽  
Andrea Angeli ◽  
Kübra Demir ◽  
Claudiu T. Supuran ◽  
Atilla Akdemir
Keyword(s):  
Carbonic Anhydrase ◽  
Carbonic Anhydrase Ix ◽  
Zinc Binding ◽  
Human Carbonic Anhydrase
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