scholarly journals A Practical Guide to Approaching Biased Agonism at G Protein Coupled Receptors

2017 ◽  
Vol 11 ◽  
Author(s):  
Jaimee Gundry ◽  
Rachel Glenn ◽  
Priya Alagesan ◽  
Sudarshan Rajagopal
Keyword(s):  
G Protein ◽  
G Protein Coupled Receptors ◽  
Biased Agonism ◽  
Practical Guide ◽  
G Protein Coupled

Novel Insights into Biased Agonism at G Protein-Coupled Receptors and their Potential for Drug Design

2013 ◽  
Vol 19 (28) ◽  
pp. 5156-5166 ◽  
Author(s):  
Maria Marti-Solano ◽  
Ramon Guixa-Gonzalez ◽  
Ferran Sanz ◽  
Manuel Pastor ◽  
Jana Selent
Keyword(s):  
Drug Design ◽  
G Protein ◽  
G Protein Coupled Receptors ◽  
Biased Agonism ◽  
G Protein Coupled

Biased Agonism at G Protein-Coupled Receptors: The Promise and the Challenges-A Medicinal Chemistry Perspective

2014 ◽  
Vol 34 (6) ◽  
pp. 1286-1330 ◽  
Author(s):  
Jeremy Shonberg ◽  
Laura Lopez ◽  
Peter J. Scammells ◽  
Arthur Christopoulos ◽  
Ben Capuano ◽  
...  
Keyword(s):  
G Protein ◽  
Medicinal Chemistry ◽  
G Protein Coupled Receptors ◽  
Biased Agonism ◽  
G Protein Coupled

scholarly journals A Novel Method for Analyzing Extremely Biased Agonism at G Protein–Coupled Receptors

2015 ◽  
Vol 87 (5) ◽  
pp. 866-877 ◽  
Author(s):  
Edward L. Stahl ◽  
Lei Zhou ◽  
Frederick J. Ehlert ◽  
Laura M. Bohn
Keyword(s):  
G Protein ◽  
G Protein Coupled Receptors ◽  
Biased Agonism ◽  
Novel Method ◽  
G Protein Coupled

Allostery and Biased Agonism at Class B G Protein-Coupled Receptors

2016 ◽  
Vol 117 (1) ◽  
pp. 111-138 ◽  
Author(s):  
Denise Wootten ◽  
Laurence J. Miller ◽  
Cassandra Koole ◽  
Arthur Christopoulos ◽  
Patrick M. Sexton
Keyword(s):  
G Protein ◽  
G Protein Coupled Receptors ◽  
Biased Agonism ◽  
Class B ◽  
G Protein Coupled

Mechanisms of signalling and biased agonism in G protein-coupled receptors

2018 ◽  
Vol 19 (10) ◽  
pp. 638-653 ◽  
Author(s):  
Denise Wootten ◽  
Arthur Christopoulos ◽  
Maria Marti-Solano ◽  
M. Madan Babu ◽  
Patrick M. Sexton
Keyword(s):  
G Protein ◽  
G Protein Coupled Receptors ◽  
Biased Agonism ◽  
G Protein Coupled

scholarly journals Differential GRK Recruitment and the Phosphorylation Barcode as a Mechanism for Biased Agonism at G Protein‐Coupled Receptors

2021 ◽  
Vol 35 (S1) ◽  
Author(s):  
Julia Gardner ◽  
Dylan Eiger ◽  
Christopher Honeycutt ◽  
Noelia Boldizsar ◽  
Issac Choi ◽  
...  
Keyword(s):  
G Protein ◽  
G Protein Coupled Receptors ◽  
Biased Agonism ◽  
G Protein Coupled
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