Faculty Opinions recommendation of Design and synthesis of peripherally restricted transient receptor potential vanilloid 1 (TRPV1) antagonists.

Receptor Potential ◽

Design And Synthesis ◽

Design and Synthesis of Peripherally Restricted Transient Receptor Potential Vanilloid 1 (TRPV1) Antagonists

Journal of Medicinal Chemistry ◽

10.1021/jm7014638 ◽

2008 ◽

Vol 51 (9) ◽

pp. 2744-2757 ◽

Cited By ~ 42

Author(s):

Nuria Tamayo ◽

Hongyu Liao ◽

Markian M. Stec ◽

Xianghong Wang ◽

Partha Chakrabarti ◽

...

Keyword(s):

Receptor Potential ◽

Design And Synthesis ◽

Design and Synthesis of Indole-Based Peptoids as Potent Noncompetitive Antagonists of Transient Receptor Potential Vanilloid 1

Journal of Medicinal Chemistry ◽

10.1021/jm070612v ◽

2007 ◽

Vol 50 (24) ◽

pp. 6133-6143 ◽

Cited By ~ 13

Author(s):

Martina Quintanar-Audelo ◽

Asia Fernández-Carvajal ◽

Wim Van Den Nest ◽

Cristina Carreño ◽

Antonio Ferrer-Montiel ◽

...

Keyword(s):

Receptor Potential ◽

Design And Synthesis ◽

Discovery of potent transient receptor potential vanilloid 1 antagonists: Design and synthesis of phenoxyacetamide derivatives

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/j.bmcl.2013.04.016 ◽

2013 ◽

Vol 23 (11) ◽

pp. 3154-3156 ◽

Cited By ~ 2

Author(s):

Eiki Takahashi ◽

Noriyuki Hirano ◽

Takashi Nagahara ◽

Satoru Yoshikawa ◽

Shinobu Momen ◽

...

Keyword(s):

Receptor Potential ◽

Design And Synthesis ◽

Design and synthesis of conformationally restricted capsaicin analogues based in the 1, 3, 4-thiadiazole heterocycle reveal a novel family of transient receptor potential vanilloid 1 (TRPV1) antagonists

European Journal of Medicinal Chemistry ◽

10.1016/j.ejmech.2013.05.001 ◽

2013 ◽

Vol 66 ◽

pp. 193-203 ◽

Cited By ~ 7

Author(s):

Carolyne Lespay Rebolledo ◽

Pamela Sotelo-Hitschfeld ◽

Sebastián Brauchi ◽

Miguel Zárraga Olavarría

Keyword(s):

Receptor Potential ◽

Conformationally Restricted ◽

Design And Synthesis ◽

Transient Receptor ◽

Capsaicin Analogues

The design and synthesis of transient receptor potential vanilloid 3 inhibitors with novel skeleton

Bioorganic Chemistry ◽

10.1016/j.bioorg.2021.105115 ◽

2021 ◽

pp. 105115

Author(s):

Mengqi Lv ◽

Han Wu ◽

Yaxuan Qu ◽

Siyi Wu ◽

Junxia Wang ◽

...

Keyword(s):

Receptor Potential ◽

Design And Synthesis ◽

Design and Synthesis of New Transient Receptor Potential Vanilloid Type-1 (TRPV1) Channel Modulators: Identification, Molecular Modeling Analysis, and Pharmacological Characterization of the N-(4-Hydroxy-3-methoxybenzyl)-4-(thiophen-2-yl)butanamide, a Small Molecule Endowed with Agonist TRPV1 Activity and Protective Effects against Oxidative Stress

ACS Chemical Neuroscience ◽

10.1021/acschemneuro.5b00333 ◽

2016 ◽

Vol 7 (6) ◽

pp. 737-748 ◽

Cited By ~ 12

Author(s):

Francesca Aiello ◽

Mariateresa Badolato ◽

Federica Pessina ◽

Claudia Sticozzi ◽

Vanessa Maestrini ◽

...

Keyword(s):

Receptor Potential ◽

Protective Effects ◽

Pharmacological Characterization ◽

Design And Synthesis ◽

Modeling Analysis ◽

Faculty Opinions recommendation of Transient receptor potential vanilloid 1 is required for intrinsic osmoreception in organum vasculosum lamina terminalis neurons and for normal thirst responses to systemic hyperosmolality.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.1047186.497222 ◽

2006 ◽

Author(s):

Alastair Ferguson

Keyword(s):

Receptor Potential ◽

Lamina Terminalis ◽

Organum Vasculosum Lamina Terminalis ◽

Organum Vasculosum ◽

Faculty Opinions recommendation of Transient receptor potential vanilloid 1 is required for intrinsic osmoreception in organum vasculosum lamina terminalis neurons and for normal thirst responses to systemic hyperosmolality.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.1047186.497108 ◽

2006 ◽

Author(s):

Bernd Nilius

Keyword(s):

Receptor Potential ◽

Lamina Terminalis ◽

Organum Vasculosum Lamina Terminalis ◽

Organum Vasculosum ◽

Faculty Opinions recommendation of Somatostatin modulates the transient receptor potential vanilloid 1 (TRPV1) ion channel.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.1052995.504951 ◽

2006 ◽

Author(s):

Marcos Milla

Keyword(s):

Ion Channel ◽

Receptor Potential ◽

Faculty Opinions recommendation of A specific subset of transient receptor potential vanilloid-type channel subunits in Caenorhabditis elegans endocrine cells function as mixed heteromers to promote neurotransmitter release.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.1063770.516694 ◽

2007 ◽

Author(s):

Oliver Hobert

Keyword(s):

Caenorhabditis Elegans ◽

Neurotransmitter Release ◽

Endocrine Cells ◽

Receptor Potential ◽

Specific Subset ◽