ChemInform Abstract: Nα-Alkylated Derivatives of 2-Phenylhistamines: Synthesis and in vitro Activity of Potent Histamine H1-Receptor Agonists.

ChemInform ◽  
2010 ◽  
Vol 30 (2) ◽  
pp. no-no
Author(s):  
K. KRAMER ◽  
S. ELZ ◽  
H. H. PERTZ ◽  
W. SCHUNACK
Keyword(s):  
Vitro Activity ◽  
In Vitro Activity ◽  
H1 Receptor ◽  
Histamine H1 Receptor ◽  
Receptor Agonists ◽  
Derivatives Of

Nα-Imidazolylalkyl and Pyridylalkyl Derivatives of Histaprodifen:  Synthesis and in Vitro Evaluation of Highly Potent Histamine H1-Receptor Agonists

2003 ◽  
Vol 46 (25) ◽  
pp. 5458-5470 ◽  
Author(s):  
Sonja Menghin ◽  
Heinz H. Pertz ◽  
Kai Kramer ◽  
Roland Seifert ◽  
Walter Schunack ◽  
...  
Keyword(s):  
H1 Receptor ◽  
In Vitro Evaluation ◽  
Histamine H1 Receptor ◽  
Receptor Agonists ◽  
Derivatives Of

Antimycobacterial 3-phenyl-4-thioxo-2H-1,3-benzoxazine-2(3H)-ones and 3-phenyl-2H-1,3-benzoxazine-2,4(3H)-dithiones substituted on phenyl and benzoxazine moiety in position 6

2011 ◽  
Vol 65 (3) ◽  
Author(s):  
Eva Petrlíková ◽  
Karel Waisser ◽  
Rafael Doležal ◽  
Pavel Holý ◽  
Jiří Gregor ◽  
...  
Keyword(s):  
Mycobacterium Tuberculosis ◽  
Antimycobacterial Activity ◽  
Vitro Activity ◽  
In Vitro Activity ◽  
Derivatives Of

AbstractA series of forty-five derivatives of 3-phenyl-4-thioxo-2H-1,3-benzoxazine-2(3H)-ones and forty-five derivatives of 3-phenyl-2H-1,3-benzoxazine-2,4(3H)-dithiones was synthesised. The compounds exhibited in-vitro activity against Mycobacterium tuberculosis, M. kansasii (two strains), and M. avium. The most active derivatives were more active than isonicotinhydrazide (INH). The quantitative relationships between the structure and antimycobacterial activity were calculated. The activity against M. tuberculosis increased with the lipophilicity of the substituents.

In vitro activity of novel sulphonic derivatives of distamicyn A

1992 ◽  
pp. 455-458 ◽  
Author(s):  
M. Mariani ◽  
A. Paio ◽  
M. Ciomei ◽  
W. Pastori ◽  
C. Franzetti ◽  
...  
Keyword(s):  
Vitro Activity ◽  
In Vitro Activity ◽  
Derivatives Of

In vitro activity of novel derivatives of 1,3-oxazole-4-carboxylate and 1,3-oxazole-4-carbonitrile against human cytomegalovirus

2019 ◽  
Vol 28 (8) ◽  
pp. 1205-1211 ◽  
Author(s):  
Maryna V. Kachaeva ◽  
Stepan G. Pilyo ◽  
Caroll B. Hartline ◽  
Emma A. Harden ◽  
Mark N. Prichard ◽  
...  
Keyword(s):  
Human Cytomegalovirus ◽  
Vitro Activity ◽  
In Vitro Activity ◽  
Derivatives Of

In Vitro Activity of Novel 5-Carbonyl Derivatives of 3-Phenyl-3-(1H-imidazol-1-ylmethyl)-2-methyl-isoxazolidines

1988 ◽  
Vol 544 (1 Antifungal Dr) ◽  
pp. 396-399 ◽  
Author(s):  
GRACE A. BENNETT ◽  
GEORGE B. MULLEN ◽  
THOMAS R. DeCORY,b ◽  
STANLEY D. ALLEN ◽  
JEFFREY T. MITCHELL ◽  
...  
Keyword(s):  
Vitro Activity ◽  
In Vitro Activity ◽  
Carbonyl Derivatives ◽  
Derivatives Of

scholarly journals 3-Keto-11,12-carbazate Derivatives of 6-0-Methylerythromycin A Synthesis and In Vitro Activity.

1996 ◽  
Vol 49 (5) ◽  
pp. 465-477 ◽  
Author(s):  
GEORGE GRIESGRABER ◽  
YAT SUN OR ◽  
DANIEL T. W. CHU ◽  
ANGELA M. NILIUS ◽  
PAULINE M. JOHNSON ◽  
...  
Keyword(s):  
Vitro Activity ◽  
In Vitro Activity ◽  
Derivatives Of
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