ChemInform Abstract: Synthesis and Biological Evaluation of Novel Thio-Substituted Chromanes (VIII) as High-Affinity Partial Agonists for the Estrogen Receptor.

Lise B. Christiansen; et al. et al.

doi:10.1002/chin.200212171

ChemInform Abstract: Synthesis and Biological Evaluation of Novel Thio-Substituted Chromanes (VIII) as High-Affinity Partial Agonists for the Estrogen Receptor.

ChemInform ◽

10.1002/chin.200212171 ◽

2010 ◽

Vol 33 (12) ◽

pp. no-no

Author(s):

Lise B. Christiansen ◽

et al. et al.

Keyword(s):

Estrogen Receptor ◽

Biological Evaluation ◽

High Affinity ◽

Partial Agonists ◽

Synthesis And Biological Evaluation

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Synthesis and biological evaluation of novel thio-substituted chromanes as high-affinity partial agonists for the estrogen receptor

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/s0960-894x(01)00679-5 ◽

2002 ◽

Vol 12 (1) ◽

pp. 17-19 ◽

Cited By ~ 5

Author(s):

Lise B Christiansen ◽

Martin Wenckens ◽

Paul S Bury ◽

Birgitte Gissel ◽

Birgit S Hansen ◽

...

Keyword(s):

Estrogen Receptor ◽

Biological Evaluation ◽

High Affinity ◽

Partial Agonists ◽

Synthesis And Biological Evaluation

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Synthesis and biological evaluation of novel m-carborane-containing estrogen receptor partial agonists as SERM candidates

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/j.bmcl.2015.05.083 ◽

2015 ◽

Vol 25 (16) ◽

pp. 3213-3216 ◽

Cited By ~ 8

Author(s):

Kiminori Ohta ◽

Takumi Ogawa ◽

Asako Kaise ◽

Yasuyuki Endo

Keyword(s):

Estrogen Receptor ◽

Biological Evaluation ◽

Partial Agonists ◽

Synthesis And Biological Evaluation

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Design, synthesis, and biological evaluation of novel sulindac derivatives as partial agonists of PPARγ with potential anti-diabetic efficacy

European Journal of Medicinal Chemistry ◽

10.1016/j.ejmech.2021.113542 ◽

2021 ◽

pp. 113542

Author(s):

Fengyu Huang ◽

Zhiping Zeng ◽

Weidong Zhang ◽

Zhiqiang Yan ◽

Jiayun Chen ◽

...

Keyword(s):

Biological Evaluation ◽

Design Synthesis ◽

Partial Agonists ◽

Synthesis And Biological Evaluation

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Synthesis and biological evaluation of 6-aryl-6 H -pyrrolo[3,4- d ]pyridazine derivatives as high-affinity ligands of the α 2 δ subunit of voltage-gated calcium channels

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/j.bmcl.2004.02.070 ◽

2004 ◽

Vol 14 (9) ◽

pp. 2031-2034 ◽

Cited By ~ 14

Author(s):

Tao Hu ◽

Brian A Stearns ◽

Brian T Campbell ◽

Jeannie M Arruda ◽

Chixu Chen ◽

...

Keyword(s):

Calcium Channels ◽

Biological Evaluation ◽

Affinity Ligands ◽

Voltage Gated ◽

High Affinity ◽

Voltage Gated Calcium Channels ◽

Pyridazine Derivatives ◽

Synthesis And Biological Evaluation

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ChemInform Abstract: Novel Selective and Partial Agonists of 5-HT3 Receptors. Part 1. Synthesis and Biological Evaluation of Piperazinopyrrolothienopyrazines.

ChemInform ◽

10.1002/chin.199635160 ◽

2010 ◽

Vol 27 (35) ◽

pp. no-no

Author(s):

S. RAULT ◽

J.-C. LANCELOT ◽

H. PRUNIER ◽

M. ROBBA ◽

P. RENARD ◽

...

Keyword(s):

Biological Evaluation ◽

Partial Agonists ◽

Synthesis And Biological Evaluation

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(+)-p-([18F]fluorobenzyl)spirotrozamicol {(+)-[18F]Spiro-FBT}: synthesis and biological evaluation of a high-affinity ligand for the vesicular acetylcholine transporter (VAChT)

Nuclear Medicine and Biology ◽

10.1016/s0969-8051(98)00090-0 ◽

1999 ◽

Vol 26 (2) ◽

pp. 189-192 ◽

Cited By ~ 10

Author(s):

S.M.N Efange ◽

M.A Nader ◽

R.L.E Ehrenkaufer ◽

A.B Khare ◽

C.R Smith ◽

...

Keyword(s):

Biological Evaluation ◽

Vesicular Acetylcholine Transporter ◽

High Affinity ◽

Affinity Ligand ◽

Synthesis And Biological Evaluation ◽

High Affinity Ligand

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Synthesis and biological evaluation of phenolic 4,5-dihydroisoxazoles and 3-hydroxy ketones as estrogen receptor α and β agonists

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2010.04.007 ◽

2010 ◽

Vol 18 (10) ◽

pp. 3437-3447 ◽

Cited By ~ 23

Author(s):

Pekka K. Poutiainen ◽

Tuomas A. Venäläinen ◽

Mikael Peräkylä ◽

Juha M. Matilainen ◽

Sami Väisänen ◽

...

Keyword(s):

Estrogen Receptor ◽

Estrogen Receptor Α ◽

Biological Evaluation ◽

Hydroxy Ketones ◽

Synthesis And Biological Evaluation

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Synthesis and Biological Evaluation in Vitro of Selective, High Affinity Peptide Antagonists of Human Melanin-Concentrating Hormone Action at Human Melanin-Concentrating Hormone Receptor 1

Biochemistry ◽

10.1021/bi0200514 ◽

2002 ◽

Vol 41 (20) ◽

pp. 6383-6390 ◽

Cited By ~ 35

Author(s):

Maria A. Bednarek ◽

Donna L. Hreniuk ◽

Carina Tan ◽

Oksana C. Palyha ◽

Douglas J. MacNeil ◽

...

Keyword(s):

Hormone Receptor ◽

Biological Evaluation ◽

Hormone Action ◽

High Affinity ◽

Melanin Concentrating Hormone ◽

Affinity Peptide ◽

Synthesis And Biological Evaluation

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Synthesis and biological evaluation of novel cyclopropyl derivatives as subtype-selective ligands for estrogen receptor

Journal of Pharmacy and Pharmacology ◽

10.1111/jphp.12908 ◽

2018 ◽

Vol 70 (7) ◽

pp. 910-918 ◽

Cited By ~ 2

Author(s):

Zunyuan Wang ◽

Yewei Yang ◽

Xiaoliang Zheng ◽

Tao Zhang ◽

Wenhai Huang ◽

...

Keyword(s):

Estrogen Receptor ◽

Biological Evaluation ◽

Selective Ligands ◽

Subtype Selective ◽

Synthesis And Biological Evaluation

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Synthesis and pharmacological evaluation of novel cis-3,4-Diaryl-hydroxychromanes as high affinity partial agonists for the estrogen receptor

Bioorganic & Medicinal Chemistry ◽

10.1016/s0968-0896(01)00257-7 ◽

2002 ◽

Vol 10 (1) ◽

pp. 125-145 ◽

Cited By ~ 23

Author(s):

Paul S. Bury ◽

Lise B. Christiansen ◽

Poul Jacobsen ◽

Anker S. Jørgensen ◽

Anders Kanstrup ◽

...

Keyword(s):

Estrogen Receptor ◽

High Affinity ◽

Pharmacological Evaluation ◽

Partial Agonists

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