1-(Phenyl)isoquinoline Carboxamides: A Novel Class of Subtype Selective Inhibitors of Thyrotropin-Releasing Hormone (TRH) Receptors.

Selective Inhibitors ◽

Releasing Hormone ◽

Subtype Selective ◽

1-(Phenyl)isoquinoline carboxamides: a novel class of subtype selective inhibitors of thyrotropin-releasing hormone (TRH) receptors

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/j.bmcl.2004.11.017 ◽

2005 ◽

Vol 15 (3) ◽

pp. 733-736 ◽

Cited By ~ 7

Author(s):

Jian-kang Jiang ◽

Craig J. Thomas ◽

Susanne Neumann ◽

Xinping Lu ◽

Kenner C. Rice ◽

...

Keyword(s):

Selective Inhibitors ◽

Releasing Hormone ◽

Subtype Selective ◽

Thyrotropin-releasing hormone (TRH) receptor number determines the size of the TRH-responsive phosphoinositide pool. Demonstration using controlled expression of TRH receptors by adenovirus mediated gene transfer.

Journal of Biological Chemistry ◽

10.1016/s0021-9258(17)37443-4 ◽

1994 ◽

Vol 269 (9) ◽

pp. 6779-6783

Author(s):

M.C. Gershengorn ◽

M. Heinflink ◽

D.R. Nussenzveig ◽

P.M. Hinkle ◽

E. Falck-Pedersen

Keyword(s):

Gene Transfer ◽

Releasing Hormone ◽

Receptor Number ◽

Trh Receptor ◽

Ex vivo binding characteristics of thyrotropin-releasing hormone(TRH) and its analogue, JTP-2942, to TRH receptors in rat brain

The Japanese Journal of Pharmacology ◽

10.1016/s0021-5198(19)40362-4 ◽

1998 ◽

Vol 76 ◽

pp. 61

Author(s):

Akihiko Urayama ◽

Shizuo Yamada ◽

Ryohei Kimura

Keyword(s):

Rat Brain ◽

Ex Vivo ◽

Releasing Hormone ◽

Binding Characteristics ◽

Effect of Chronic Administration of Scopolamine on Thyrotropin-Releasing Hormone (TRH)-mediated Wet-Dog Shakes and TRH Receptors as Measured by Quantitative Autoradiography

Annals of the New York Academy of Sciences ◽

10.1111/j.1749-6632.1989.tb46687.x ◽

1989 ◽

Vol 553 (1 Thyrotropin-R) ◽

pp. 532-534

Author(s):

MATTHEW A. SILLS ◽

ALAN M. MELLOW ◽

TREY SUNDERLAND ◽

CHARANJIT S. AULAKH ◽

PAUL A. NEWHOUSE ◽

...

Keyword(s):

Chronic Administration ◽

Quantitative Autoradiography ◽

Releasing Hormone ◽

Wet Dog Shakes ◽

Binding of Fluorinated Analogues of Thyrotropin-Releasing Hormone to TRH Receptors in the Rat Brain

Annals of the New York Academy of Sciences ◽

10.1111/j.1749-6632.1989.tb46683.x ◽

1989 ◽

Vol 553 (1 Thyrotropin-R) ◽

pp. 524-525 ◽

Cited By ~ 2

Author(s):

STEFAN VONHOF ◽

ILARI PAAKKARI ◽

VIRENDER M. LABROO ◽

LOUIS A. COHEN ◽

GIORA FEUERSTEIN

Keyword(s):

Rat Brain ◽

Releasing Hormone ◽

Autoradiographic localization of thyrotropin-releasing hormone (TRH) receptors in human spinal cord

Neurology ◽

10.1212/wnl.35.3.328 ◽

1985 ◽

Vol 35 (3) ◽

pp. 328-328 ◽

Cited By ~ 40

Author(s):

S. Manaker ◽

A. Winokur ◽

C. H. Rhodes ◽

T. C. Rainbow

Keyword(s):

Spinal Cord ◽

Releasing Hormone ◽

Human Spinal Cord ◽

Distribution of Thyrotropin-Releasing Hormone (TRH) Receptors in the Brain of the Ataxic Mutant Mouse, Rolling Mouse Nagoya.

Biological and Pharmaceutical Bulletin ◽

10.1248/bpb.20.86 ◽

1997 ◽

Vol 20 (1) ◽

pp. 86-87 ◽

Cited By ~ 2

Author(s):

Kiyoshi KINOSHITA ◽

Michio YAMAMURA ◽

Juko SUGIHARA

Keyword(s):

Mutant Mouse ◽

Releasing Hormone ◽

The Brain ◽

Regulator of G Protein Signaling 4 Suppresses Basal and Thyrotropin Releasing-Hormone (TRH)-Stimulated Signaling by Two Mouse TRH Receptors, TRH-R1and TRH-R21

Endocrinology ◽

10.1210/endo.142.3.8019 ◽

2001 ◽

Vol 142 (3) ◽

pp. 1188-1194 ◽

Cited By ~ 6

Author(s):

Sönke Harder ◽

Xinping Lu ◽

Wei Wang ◽

Friedrich Buck ◽

Marvin C. Gershengorn ◽

...

Keyword(s):

G Protein ◽

G Protein Signaling ◽

Protein Signaling ◽

Releasing Hormone ◽

Thyrotropin-releasing hormone (TRH) receptors. Localization by light microscopic autoradiography in rat brain using [3H][3-Me-His2]TRH as the radioligand

Journal of Neuroscience ◽

10.1523/jneurosci.05-02-00551.1985 ◽

1985 ◽

Vol 5 (2) ◽

pp. 551-561 ◽

Cited By ~ 85

Author(s):

PW Mantyh ◽

SP Hunt

Keyword(s):

Rat Brain ◽

Releasing Hormone ◽

Localization of thyrotropin-releasing hormone (TRH) receptors in the septal nucleus of the rat brain

Brain Research ◽

10.1016/0006-8993(84)90081-7 ◽

1984 ◽

Vol 296 (2) ◽

pp. 393-395 ◽

Cited By ~ 19

Author(s):

Steven M. Simasko ◽

Akira Horita

Keyword(s):

Rat Brain ◽

Septal Nucleus ◽

Releasing Hormone ◽