Heterocyclic Synthesis: A Convenient Route to Some 2-Mercapto 1,3,4-Oxadiazole and Green Chemistry Microwave-Induced One-Pot Synthesis of 2-Aryl 1,3,4-Oxadiazole in Quinazolone and Their Antibacterial and Antifungal Activity.

ChemInform ◽  
2005 ◽  
Vol 36 (49) ◽  
Author(s):  
A. R. Desai ◽  
K. R. Desai
Keyword(s):  
Antifungal Activity ◽  
Green Chemistry ◽  
Heterocyclic Synthesis ◽  
Antibacterial And Antifungal Activity ◽  
One Pot ◽  
One Pot Synthesis ◽  
Convenient Route ◽  
Antibacterial And Antifungal

Copper-catalyzed Convenient Synthesis and SAR Studies of Substituted-1,2,3-triazole as Antimicrobial Agents

2018 ◽  
Vol 16 (1) ◽  
pp. 3-10
Author(s):  
Aniket P. Sarkate ◽  
Kshipra S. Karnik ◽  
Pravin S. Wakte ◽  
Ajinkya P. Sarkate ◽  
Ashwini V. Izankar ◽  
...  
Keyword(s):  
Antimicrobial Activity ◽  
Antifungal Activity ◽  
Antimicrobial Agents ◽  
Cycloaddition Reaction ◽  
Dipolar Cycloaddition ◽  
One Pot ◽  
Triazole Derivatives ◽  
Sar Studies ◽  
Convenient Synthesis ◽  
Antibacterial And Antifungal

Background:A novel copper-catalyzed synthesis of substituted-1,2,3-triazole derivatives has been developed and performed by Huisgen 1,3-dipolar cycloaddition reaction of azides with alkynes. The reaction is one-pot multicomponent.Objective:We state the advancement and execution of a methodology allowing for the synthesis of some new substituted 1,2,3-triazole analogues with antimicrobial activity.Methods:A series of triazole derivatives was synthesized by Huisgen 1,3-dipolar cycloaddition reaction of azides with alkynes. The structures of the synthesized compounds were elucidated and confirmed by 1H NMR, IR, MS and elemental analysis. All the synthesized compounds were tested for their antimicrobial activity against a series of strains of Bacillus subtilis, Staphylococcus aureus and Escherichia coli for antibacterial activity and against the strains of Candida albicans, Aspergillus flavus and Aspergillus nigar for antifungal activity, respectively.Results and Conclusion:From the antimicrobial data, it was observed that all the newly synthesized compounds showed good to moderate level of antibacterial and antifungal activity.

Synthesis of Coumarin Derivatives with Cytotoxic, Antibacterial and Antifungal Activity

2004 ◽  
Vol 19 (4) ◽  
pp. 373-379 ◽  
Author(s):  
Khalid Mohammed Khan ◽  
Zafar S. Saify ◽  
Muhammad Zarrar Khan ◽  
Zia-Ullah ◽  
M. Iqbal Choudhary ◽  
...  
Keyword(s):  
Antifungal Activity ◽  
Coumarin Derivatives ◽  
Antibacterial And Antifungal Activity ◽  
Antibacterial And Antifungal
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