Radiosynthesis of the α4β2 nicotinic acetylcholine receptor ligand: 5-((1-[11C]-methyl-2-(S)-pyrrolidinyl)methoxy)-2-chloro-3-((E)-2-(2-fluoropyridin-4-yl)vinyl)pyridine

Receptor Ligand ◽

Nicotinic Acetylcholine ◽

Vinyl Pyridine

Measurement of the α4β2* nicotinic acetylcholine receptor ligand 2-[18F]Fluoro-A-85380 and its metabolites in human blood during PET investigation: a methodological study

Nuclear Medicine and Biology ◽

10.1016/j.nucmedbio.2006.12.008 ◽

2007 ◽

Vol 34 (3) ◽

pp. 331-342 ◽

Cited By ~ 17

Author(s):

Dietlind Sorger ◽

Georg A. Becker ◽

Marianne Patt ◽

Andreas Schildan ◽

Udo Grossmann ◽

...

Keyword(s):

Acetylcholine Receptor ◽

Human Blood ◽

Methodological Study ◽

Receptor Ligand ◽

Influence of acetylcholine levels on the binding of a SPECT nicotinic acetylcholine receptor ligand [123I]5-I-A-85380

Synapse ◽

10.1002/syn.10194 ◽

2003 ◽

Vol 48 (3) ◽

pp. 116-122 ◽

Cited By ~ 15

Author(s):

Masahiro Fujita ◽

Mohammed S. Al-Tikriti ◽

Gilles Tamagnan ◽

Sami S. Zoghbi ◽

Ali Bozkurt ◽

...

Keyword(s):

Acetylcholine Receptor ◽

Receptor Ligand ◽

Functional Characterization of the Novel Neuronal Nicotinic Acetylcholine Receptor Ligand GTS-21 In Vitro and In Vivo

Pharmacology Biochemistry and Behavior ◽

10.1016/s0091-3057(96)00354-1 ◽

1997 ◽

Vol 57 (1-2) ◽

pp. 231-241 ◽

Cited By ~ 136

Author(s):

Clark A Briggs ◽

David J Anderson ◽

Jorge D Brioni ◽

Jerry J Buccafusco ◽

Michael J Buckley ◽

...

Keyword(s):

Acetylcholine Receptor ◽

Functional Characterization ◽

Neuronal Nicotinic Acetylcholine Receptor ◽

The Novel ◽

Receptor Ligand ◽

Expression of the endogenous, nicotinic acetylcholine receptor ligand, SLURP-1, in human colon cancer

Autonomic and Autacoid Pharmacology ◽

10.1111/j.1474-8673.2008.00424.x ◽

2008 ◽

Vol 28 (4) ◽

pp. 109-116 ◽

Cited By ~ 14

Author(s):

A. Pettersson ◽

S. Nordlander ◽

G. Nylund ◽

A. Khorram-Manesh ◽

S. Nordgren ◽

...

Keyword(s):

Colon Cancer ◽

Acetylcholine Receptor ◽

Human Colon ◽

Human Colon Cancer ◽

Receptor Ligand ◽

Distribution volume of the nicotinic acetylcholine receptor ligand 2-[F-18]F-A-85380: Nonsmokers versus smokers

NeuroImage ◽

10.1016/j.neuroimage.2006.04.139 ◽

2006 ◽

Vol 31 ◽

pp. T156 ◽

Cited By ~ 3

Author(s):

Hans Herzog ◽

M. Minnerop ◽

W. Eschner ◽

F. Jessen ◽

C. Schütz ◽

...

Keyword(s):

Acetylcholine Receptor ◽

Distribution Volume ◽

Receptor Ligand ◽

Primary sensory neuronal expression of SLURP-1, an endogenous nicotinic acetylcholine receptor ligand

Neuroscience Research ◽

10.1016/j.neures.2009.04.014 ◽

2009 ◽

Vol 64 (4) ◽

pp. 403-412 ◽

Cited By ~ 37

Author(s):

Yasuhiro Moriwaki ◽

Yosuke Watanabe ◽

Tomoe Shinagawa ◽

Miho Kai ◽

Mai Miyazawa ◽

...

Keyword(s):

Acetylcholine Receptor ◽

Receptor Ligand ◽

Nicotinic Acetylcholine ◽

Neuronal Expression

Exploring the Relationship between Nicotinic Acetylcholine Receptor Ligand Size, Efficiency, Efficacy, and C-Loop Opening

Journal of Chemical Information and Modeling ◽

10.1021/acs.jcim.7b00152 ◽

2017 ◽

Vol 57 (8) ◽

pp. 1947-1956 ◽

Cited By ~ 4

Author(s):

Qianyun Ma ◽

Han-Shen Tae ◽

Guanzhao Wu ◽

Tao Jiang ◽

Rilei Yu

Keyword(s):

Acetylcholine Receptor ◽

Receptor Ligand ◽

Nicotinic Acetylcholine ◽

The Relationship ◽

Size Efficiency

Potentials of Mean Force for Acetylcholine Unbinding from the Alpha7 Nicotinic Acetylcholine Receptor Ligand-Binding Domain

Journal of the American Chemical Society ◽

10.1021/ja057292u ◽

2006 ◽

Vol 128 (9) ◽

pp. 3019-3026 ◽

Cited By ~ 67

Author(s):

Deqiang Zhang ◽

Justin Gullingsrud ◽

J. Andrew McCammon

Keyword(s):

Ligand Binding ◽

Acetylcholine Receptor ◽

Binding Domain ◽

Ligand Binding Domain ◽

Receptor Ligand ◽

Nicotinic Acetylcholine ◽

Alpha7 Nicotinic Acetylcholine Receptor ◽

Potentials Of Mean Force

A-85380 [3-(2(S)-azetidinylmethoxy) pyridine]: In Vitro pharmacological properties of a novel, high affinity α4β2 nicotinic acetylcholine receptor ligand

Neuropharmacology ◽

10.1016/0028-3908(96)84644-2 ◽

1996 ◽

Vol 35 (6) ◽

pp. 725-734 ◽

Cited By ~ 90

Author(s):

James P. Sullivan ◽

Diana Donnelly-Roberts ◽

Clark A. Briggs ◽

David J. Anderson ◽

Murali Gopalakrishnan ◽

...

Keyword(s):

Acetylcholine Receptor ◽

Pharmacological Properties ◽

Receptor Ligand ◽

Nicotinic Acetylcholine ◽

High Affinity

P2-390: Evaluating a novel alpha7 nicotinic acetylcholine receptor ligand [11C]CHIBA1001 for positron emission tomography

Alzheimer s & Dementia ◽

10.1016/j.jalz.2010.05.1442 ◽

2010 ◽

Vol 6 ◽

pp. S431-S431

Author(s):

Masatomo Ishikawa ◽

Kenji Ishii ◽

Jun Toyohara ◽

Muneyuki Sakata ◽

Keiichi Oda ◽

...

Keyword(s):

Positron Emission Tomography ◽

Acetylcholine Receptor ◽

Emission Tomography ◽

Receptor Ligand ◽

Nicotinic Acetylcholine ◽

Alpha7 Nicotinic Acetylcholine Receptor ◽

Positron Emission