Novel gallium(III) complexes as potential pet imaging agents for probing multidrug resistance (MDR1) P-glycoprotein (PGP) transport activity: Effect of MDR reversal agents

2001 ◽  
Vol 44 (S1) ◽  
pp. S75-S77
Author(s):  
V. Sharma ◽  
J. Dahlheimer ◽  
D. Piwnica-Worms
Keyword(s):  
Multidrug Resistance ◽  
Pet Imaging ◽  
Imaging Agents ◽  
Transport Activity ◽  
Reversal Agents ◽  
Activity Effect ◽  
P Glycoprotein ◽  
Mdr Reversal

Ingol diterpenoids as P-glycoprotein-dependent multidrug resistance (MDR) reversal agents from Euphorbia marginata

2020 ◽  
Vol 95 ◽  
pp. 103546 ◽  
Author(s):  
Yao Zhang ◽  
Run-Zhu Fan ◽  
Jun Sang ◽  
Yi-Jing Tian ◽  
Jia-Qi Chen ◽  
...  
Keyword(s):  
Multidrug Resistance ◽  
Reversal Agents ◽  
P Glycoprotein ◽  
Mdr Reversal

Design and Syntheses of Permethyl Ningalin B Analogues: Potent Multidrug Resistance (MDR) Reversal Agents of Cancer Cells

2010 ◽  
Vol 53 (14) ◽  
pp. 5108-5120 ◽  
Author(s):  
Pu Yong Zhang ◽  
Iris L. K. Wong ◽  
Clare S. W. Yan ◽  
Xiao Yu Zhang ◽  
Tao Jiang ◽  
...  
Keyword(s):  
Multidrug Resistance ◽  
Cancer Cells ◽  
Reversal Agents ◽  
Mdr Reversal

Design, synthesis and biological evaluation of novel triazole-core reversal agents against P-glycoprotein-mediated multidrug resistance

RSC Advances ◽  
2016 ◽  
Vol 6 (31) ◽  
pp. 25819-25828 ◽  
Author(s):  
Bo Zhang ◽  
Tianxiao Zhao ◽  
Jie Zhou ◽  
Qianqian Qiu ◽  
Yuxuan Dai ◽  
...  
Keyword(s):  
Multidrug Resistance ◽  
Click Chemistry ◽  
Biological Evaluation ◽  
Glycoprotein P ◽  
Design Synthesis ◽  
Reversal Agents ◽  
P Glycoprotein ◽  
Synthesis And Biological Evaluation

We designed and synthesized a novel series of P-glycoprotein (P-gp)-mediated multidrug resistance (MDR) inhibitors bearing a triazolphenethyl–tetrahydroisoquinoline scaffold through click chemistry.

Sign in / Sign up

Export Citation Format

Share Document