Synthesis of two potent glucocorticoid receptor agonists labeled with carbon-14 and stable isotopes

2015 ◽  
Vol 58 (11-12) ◽  
pp. 445-452 ◽  
Author(s):  
Bachir Latli ◽  
Jonathan T. Reeves ◽  
Zhulin Tan ◽  
Matt Hrapchak ◽  
Jinhua J. Song ◽  
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Keyword(s):  
Stable Isotopes ◽  
Glucocorticoid Receptor ◽  
Receptor Agonists ◽  
Carbon 14

scholarly journals The triterpene echinocystic acid and its 3-O-glucoside derivative are revealed as potent and selective glucocorticoid receptor agonists

2016 ◽  
Vol 79 ◽  
pp. 277-287 ◽  
Author(s):  
Demetra Georgatza ◽  
Vyron A. Gorgogietas ◽  
Paraskevi Kylindri ◽  
Maria Ch. Charalambous ◽  
Kalliope K. Papadopoulou ◽  
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Keyword(s):  
Glucocorticoid Receptor ◽  
Receptor Agonists ◽  
Echinocystic Acid

Detection of glucocorticoid receptor agonists in effluents from sewage treatment plants in Japan

2015 ◽  
Vol 527-528 ◽  
pp. 328-334 ◽  
Author(s):  
Go Suzuki ◽  
Kentaro Sato ◽  
Tomohiko Isobe ◽  
Hidetaka Takigami ◽  
Abraham Brouwer ◽  
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Keyword(s):  
Glucocorticoid Receptor ◽  
Sewage Treatment ◽  
Sewage Treatment Plants ◽  
Receptor Agonists

Structure Guided Design of 5-Arylindazole Glucocorticoid Receptor Agonists and Antagonists

2010 ◽  
Vol 53 (11) ◽  
pp. 4531-4544 ◽  
Author(s):  
Christopher M. Yates ◽  
Peter J. Brown ◽  
Eugene L. Stewart ◽  
Christopher Patten ◽  
Robert J. H. Austin ◽  
...  
Keyword(s):  
Glucocorticoid Receptor ◽  
Receptor Agonists ◽  
Receptor Agonists And Antagonists

Aryl aminopyrazole benzamides as oral non-steroidal selective glucocorticoid receptor agonists

2009 ◽  
Vol 19 (1) ◽  
pp. 158-162 ◽  
Author(s):  
Heather A. Barnett ◽  
Diane M. Coe ◽  
Tony W.J. Cooper ◽  
Torquil I. Jack ◽  
Haydn T. Jones ◽  
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Keyword(s):  
Glucocorticoid Receptor ◽  
Receptor Agonists

Discovery of acylurea isosteres of 2-acylaminothiadiazole in the azaxanthene series of glucocorticoid receptor agonists

2014 ◽  
Vol 24 (15) ◽  
pp. 3268-3273 ◽  
Author(s):  
Hua Gong ◽  
Michael Yang ◽  
Zili Xiao ◽  
Arthur M. Doweyko ◽  
Mark Cunningham ◽  
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Glucocorticoid Receptor ◽  
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Identification of Highly Efficacious Glucocorticoid Receptor Agonists with a Potential for Reduced Clinical Bone Side Effects

2014 ◽  
Vol 57 (4) ◽  
pp. 1583-1598 ◽  
Author(s):  
Christian Harcken ◽  
Doris Riether ◽  
Daniel Kuzmich ◽  
Pingrong Liu ◽  
Raj Betageri ◽  
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Glucocorticoid Receptor ◽  
Receptor Agonists

Identification of dissociated non-steroidal glucocorticoid receptor agonists

2007 ◽  
Vol 17 (18) ◽  
pp. 5025-5031 ◽  
Author(s):  
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Tom Kirrane ◽  
John Proudfoot ◽  
Younes Bekkali ◽  
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Receptor Agonists

scholarly journals Selective Non-Steroidal Glucocorticoid Receptor Agonists Attenuate Inflammation but Do Not Impair Intestinal Epithelial Cell Restitution In Vitro

PLoS ONE ◽  
2012 ◽  
Vol 7 (1) ◽  
pp. e29756 ◽  
Author(s):  
Kerstin C. Reuter ◽  
Stefan M. Loitsch ◽  
Axel U. Dignass ◽  
Dieter Steinhilber ◽  
Jürgen Stein
Keyword(s):  
Epithelial Cell ◽  
Glucocorticoid Receptor ◽  
Intestinal Epithelial Cell ◽  
Intestinal Epithelial ◽  
Receptor Agonists
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