Study on Dual Inhibitors of HIV-1 IN/CCR5 Caffeoyl Derivatives as Neuroprotective Agents

2018 ◽  
Vol 3 (22) ◽  
pp. 6170-6173 ◽  
Author(s):  
Yameng Hao ◽  
Bolin Wu ◽  
Ying Chen ◽  
Xuefeng Sun ◽  
Yixing Sun ◽  
...  
Keyword(s):  
Neuroprotective Agents ◽  
Dual Inhibitors ◽  
Caffeoyl Derivatives ◽  
Hiv 1

Design, synthesis and biological evaluation of caffeoyl benzanilides as dual inhibitors of HIV integrase and CCR5

MedChemComm ◽  
2016 ◽  
Vol 7 (10) ◽  
pp. 2028-2032 ◽  
Author(s):  
Xuefeng Sun ◽  
Ningning Fan ◽  
Weisi Xu ◽  
Yixing Sun ◽  
Xin Xie ◽  
...  
Keyword(s):  
Biological Evaluation ◽  
Hiv Integrase ◽  
Dual Inhibitor ◽  
Design Synthesis ◽  
Dual Inhibitors ◽  
Synthesis And Biological Evaluation ◽  
Hiv 1

Novel series of caffeoyl benzanilides have been synthesized and evaluated as dual inhibitors of HIV-1 CCR5/IN. Compound 9a exhibited the possibility of being a dual inhibitor of HIV-1.

Discovery of dual inhibitors targeting both HIV-1 capsid and human cyclophilin A to inhibit the assembly and uncoating of the viral capsid

2009 ◽  
Vol 17 (8) ◽  
pp. 3177-3188 ◽  
Author(s):  
Jiebo Li ◽  
Zhiwu Tan ◽  
Shixing Tang ◽  
Indira Hewlett ◽  
Ruifang Pang ◽  
...  
Keyword(s):  
Cyclophilin A ◽  
Viral Capsid ◽  
Dual Inhibitors ◽  
Hiv 1

Advances in rationally designed dual inhibitors of HIV-1 reverse transcriptase and integrase

2016 ◽  
Vol 24 (21) ◽  
pp. 5007-5016 ◽  
Author(s):  
Shuang-Xi Gu ◽  
Ping Xue ◽  
Xiu-Lian Ju ◽  
Yuan-Yuan Zhu
Keyword(s):  
Reverse Transcriptase ◽  
Dual Inhibitors ◽  
Hiv 1

scholarly journals Structure–Activity Relationship of Pyrrolyl Diketo Acid Derivatives as Dual Inhibitors of HIV-1 Integrase and Reverse Transcriptase Ribonuclease H Domain

2015 ◽  
Vol 58 (4) ◽  
pp. 1915-1928 ◽  
Author(s):  
Giuliana Cuzzucoli Crucitti ◽  
Mathieu Métifiot ◽  
Luca Pescatori ◽  
Antonella Messore ◽  
Valentina Noemi Madia ◽  
...  
Keyword(s):  
Reverse Transcriptase ◽  
Structure Activity Relationship ◽  
Ribonuclease H ◽  
Activity Relationship ◽  
Structure Activity ◽  
Dual Inhibitors ◽  
Relationship Of ◽  
Hiv 1

Fullerene derivatives as dual inhibitors of HIV-1 reverse transcriptase and protease

2021 ◽  
Vol 31 ◽  
pp. 127675
Author(s):  
Takumi Yasuno ◽  
Tomoyuki Ohe ◽  
Hiroki Kataoka ◽  
Kosho Hashimoto ◽  
Yumiko Ishikawa ◽  
...  
Keyword(s):  
Reverse Transcriptase ◽  
Fullerene Derivatives ◽  
Dual Inhibitors ◽  
Hiv 1

Antiretroviral effect simulation from black tea (Camellia sinensis) via dual inhibitors mechanism in HIV-1 and its social perspective in Indonesia

2021 ◽  
Vol 14 (1) ◽  
pp. 455-460
Author(s):  
Viol Dhea Kharisma ◽  
Sasando Dhohan Kharisma ◽  
Arif Nur Muhammad Ansori ◽  
Hanny Priskila Kurniawan ◽  
Adiana Mutamsari Witaningrum ◽  
...  
Keyword(s):  
Camellia Sinensis ◽  
Black Tea ◽  
Social Perspective ◽  
Dual Inhibitors ◽  
Hiv 1

Design, Synthesis, and Biological Evaluation of 1,3-Diarylpropenones as Dual Inhibitors of HIV-1 Reverse Transcriptase

ChemMedChem ◽  
2014 ◽  
pp. n/a-n/a ◽  
Author(s):  
Rita Meleddu ◽  
Valeria Cannas ◽  
Simona Distinto ◽  
Giorgia Sarais ◽  
Claudia Del Vecchio ◽  
...  
Keyword(s):  
Reverse Transcriptase ◽  
Biological Evaluation ◽  
Design Synthesis ◽  
Dual Inhibitors ◽  
Synthesis And Biological Evaluation ◽  
Hiv 1

4-[1-(4-Fluorobenzyl)-4-hydroxy-1H-indol-3-yl]-2-hydroxy-4-oxobut-2-enoic acid as a prototype to develop dual inhibitors of HIV-1 integration process

2011 ◽  
Vol 92 (1) ◽  
pp. 102-107 ◽  
Author(s):  
Laura De Luca ◽  
Rosaria Gitto ◽  
Frauke Christ ◽  
Stefania Ferro ◽  
Sara De Grazia ◽  
...  
Keyword(s):  
Enoic Acid ◽  
Integration Process ◽  
Dual Inhibitors ◽  
Hiv 1

Identification of HIV-1 Reverse Transcriptase Dual Inhibitors by a Combined Shape-, 2D-Fingerprint- and Pharmacophore-based Virtual Screening Approach

2011 ◽  
Vol 90 (2) ◽  
pp. A31 ◽  
Author(s):  
Simona Distinto ◽  
Francesca Esposito ◽  
Johannes Kirchmair ◽  
Cristina M. Cardia ◽  
Elias Maccioni ◽  
...  
Keyword(s):  
Virtual Screening ◽  
Reverse Transcriptase ◽  
Screening Approach ◽  
Dual Inhibitors ◽  
Hiv 1 ◽  
Virtual Screening Approach
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