Effects of ZK 93 426, a β-carboline benzodiazepine receptor antagonist on night sleep pattern in healthy male volunteers

Psychopharmacology ◽

10.1007/bf02245185 ◽

1995 ◽

Vol 117 (2) ◽

pp. 178-185 ◽

Author(s):

T. Duka ◽

D. Goerke ◽

K. Fichte

Keyword(s):

Receptor Antagonist ◽

Benzodiazepine Receptor ◽

Sleep Pattern ◽

Healthy Male ◽

Night Sleep ◽

Healthy Male Volunteers ◽

Male Volunteers ◽

Zk 93 426 ◽

Benzodiazepine Receptor Antagonist

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1244 The pharmacokinetic effect of the specific ETA receptor antagonist zibotentan (ZD4054) on CYP3A4 activity using midazolam as a probe in healthy male volunteers

European Journal of Cancer Supplements ◽

10.1016/s1359-6349(09)70456-2 ◽

2009 ◽

Vol 7 (2) ◽

pp. 133-134

Author(s):

J. Kemp ◽

H.K. Tomkinson ◽

D. Mazur ◽

T. Wollseifen ◽

T. Morris ◽

...

Keyword(s):

Receptor Antagonist ◽

Cyp3a4 Activity ◽

Healthy Male ◽

Healthy Male Volunteers ◽

Male Volunteers ◽

Eta Receptor ◽

Eta Receptor Antagonist

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In vitrometabolism of the specific endothelin-A receptor antagonist ZD4054 and clinical drug interactions between ZD4054 and rifampicin or itraconazole in healthy male volunteers

Xenobiotica ◽

10.1080/00498250902810944 ◽

2009 ◽

Vol 39 (6) ◽

pp. 444-456 ◽

Author(s):

H. C. Swaisland ◽

S. D. Oliver ◽

T. Morris ◽

H. K. Jones ◽

A. Bakhtyari ◽

...

Keyword(s):

Drug Interactions ◽

Receptor Antagonist ◽

Healthy Male ◽

Healthy Male Volunteers ◽

Male Volunteers ◽

Endothelin A Receptor ◽

Endothelin A ◽

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Effect on hypothalamic self-stimulation of the novel?-carbolines ZK 93 426 (a benzodiazepine receptor antagonist) and ZK 91296 (a putative partial agonist)

Journal of Neural Transmission ◽

10.1007/bf01260903 ◽

1986 ◽

Vol 66 (2) ◽

pp. 75-84 ◽

Author(s):

L. J. Herberg ◽

A. M. J. Montgomery ◽

Sandra E. File ◽

Sharon Pellow ◽

D. N. Stephens

Keyword(s):

Receptor Antagonist ◽

Partial Agonist ◽

Benzodiazepine Receptor ◽

The Novel ◽

Zk 93 426 ◽

Benzodiazepine Receptor Antagonist ◽

Self Stimulation ◽

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Human studies on the benzodiazepine receptor antagonist ?-carboline ZK 93 426: antagonism of lormetazepam's psychotropic effects

Psychopharmacology ◽

10.1007/bf00172956 ◽

1988 ◽

Vol 95 (4) ◽

Author(s):

T. Duka ◽

D. Goerke ◽

R. Dorow ◽

L. H�ller ◽

K. Fichte

Keyword(s):

Receptor Antagonist ◽

Benzodiazepine Receptor ◽

Human Studies ◽

Zk 93 426 ◽

Psychotropic Effects ◽

Benzodiazepine Receptor Antagonist

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A novel prostanoid EP1 receptor antagonist, ONO-8539, reduces acid-induced heartburn symptoms in healthy male volunteers: a randomized clinical trial

Journal of Gastroenterology ◽

10.1007/s00535-017-1308-3 ◽

2017 ◽

Vol 52 (10) ◽

pp. 1081-1089 ◽

Author(s):

Takashi Kondo ◽

Hiroo Sei ◽

Takahisa Yamasaki ◽

Toshihiko Tomita ◽

Yoshio Ohda ◽

...

Keyword(s):

Clinical Trial ◽

Receptor Antagonist ◽

Randomized Clinical Trial ◽

Healthy Male ◽

Healthy Male Volunteers ◽

Male Volunteers ◽

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Excretion, Metabolism, and Pharmacokinetics of 1-(8-(2-Chlorophenyl)-9-(4-Chlorophenyl)-9H-Purin-6-yl)-4-(Ethylamino)Piperidine-4-Carboxamide, a Selective Cannabinoid Receptor Antagonist, in Healthy Male Volunteers

Drug Metabolism and Disposition ◽

10.1124/dmd.111.043273 ◽

2011 ◽

Vol 40 (3) ◽

pp. 568-578 ◽

Author(s):

Zhuang Miao ◽

Hao Sun ◽

Jennifer Liras ◽

Chandra Prakash

Keyword(s):

Receptor Antagonist ◽

Cannabinoid Receptor ◽

Healthy Male ◽

Healthy Male Volunteers ◽

Male Volunteers

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Evaluation of the ?-carboline ZK 93 426 as a benzodiazepine receptor antagonist

Psychopharmacology ◽

10.1007/bf00464789 ◽

1984 ◽

Vol 83 (3) ◽

pp. 249-256 ◽

Author(s):

Leif H. Jensen ◽

Erling N. Petersen ◽

Claus Braestrup ◽

Tage Honor� ◽

Wolfgang Kehr ◽

...

Keyword(s):

Receptor Antagonist ◽

Benzodiazepine Receptor ◽

Zk 93 426 ◽

Benzodiazepine Receptor Antagonist

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Multiple-Dose Pharmacokinetics, Safety, and Tolerability of Bosentan, an Endothelin Receptor Antagonist, in Healthy Male Volunteers

The Journal of Clinical Pharmacology ◽

10.1177/00912709922008344 ◽

1999 ◽

Vol 39 (7) ◽

pp. 703-714 ◽

Author(s):

Cornelia Weber ◽

Rita Schmitt ◽

Herbert Birnboeck ◽

Gerard Hopfgartner ◽

Herwig Eggers ◽

...

Keyword(s):

Receptor Antagonist ◽

Multiple Dose ◽

Endothelin Receptor Antagonist ◽

Endothelin Receptor ◽

Healthy Male ◽

Healthy Male Volunteers ◽

Male Volunteers ◽

Multiple Dose Pharmacokinetics

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Attenuation by the benzodiazepine receptor antagonist, ZK 93 426, of the deficit in spatial navigation induced by nucleus basalis lesions

Behavioral and Neural Biology ◽

10.1016/0163-1047(92)90411-v ◽

1992 ◽

Vol 58 (2) ◽

pp. 159-163 ◽

Author(s):

Maria Mazurkiewicz ◽

Jouni Sirviö ◽

Paavo Riekkinen

Keyword(s):

Receptor Antagonist ◽

Spatial Navigation ◽

Benzodiazepine Receptor ◽

Nucleus Basalis ◽

Zk 93 426 ◽

Benzodiazepine Receptor Antagonist ◽

Nucleus Basalis Lesions

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Human studies on the benzodiazepine receptor antagonist ?-carboline ZK 93 426: preliminary observations on psychotropic activity

Psychopharmacology ◽

10.1007/bf00207229 ◽

1987 ◽

Vol 93 (4) ◽

Author(s):

T. Duka ◽

D.N. Stephens ◽

W. Krause ◽

R. Dorow

Keyword(s):

Receptor Antagonist ◽

Benzodiazepine Receptor ◽

Human Studies ◽

Psychotropic Activity ◽

Zk 93 426 ◽

Benzodiazepine Receptor Antagonist

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