Design, synthesis and biological evaluation of non-peptide PAR1 thrombin receptor antagonists based on small bifunctional templates: arginine and phenylalanine side chain groups are keys for receptor activity

Amino Acids ◽  
2009 ◽  
Vol 38 (4) ◽  
pp. 985-990 ◽  
Author(s):  
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Mahmoud Saifeddine ◽  
Morley D. Hollenberg ◽  
John Matsoukas ◽  
George Agelis
Keyword(s):  
Biological Evaluation ◽  
Receptor Activity ◽  
Side Chain ◽  
Thrombin Receptor ◽  
Receptor Antagonists ◽  
Design Synthesis ◽  
Synthesis And Biological Evaluation

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Vol 22 (11) ◽  
pp. 5472-5480 ◽  
Author(s):  
Jin Cai ◽  
Junqing Chen ◽  
Meng Cao ◽  
Peng Wang ◽  
Chengliang Feng ◽  
...  
Keyword(s):  
Biological Evaluation ◽  
Receptor Antagonists ◽  
Design Synthesis ◽  
Synthesis And Biological Evaluation

Design, synthesis and biological evaluation of cyclic angiotensin II analogues with 3,5 side-Chain bridges

2002 ◽  
Vol 12 (18) ◽  
pp. 2627-2633 ◽  
Author(s):  
Panagiota Roumelioti ◽  
Ludmila Polevaya ◽  
Panagiotis Zoumpoulakis ◽  
Nektarios Giatas ◽  
Ilze Mutule ◽  
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Keyword(s):  
Angiotensin Ii ◽  
Biological Evaluation ◽  
Side Chain ◽  
Design Synthesis ◽  
Angiotensin Ii Analogues ◽  
Synthesis And Biological Evaluation
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