Drug–Drug Interaction Potential of Darolutamide: In Vitro and Clinical Studies

Christian Zurth; Mikko Koskinen; Robert Fricke; Olaf Prien; Timo Korjamo; Kristina Graudenz; Karsten Denner; Michaela Bairlein; Clemens-Jeremias von Bühler; Gary Wilkinson; Hille Gieschen

doi:10.1007/s13318-019-00577-5

Drug–Drug Interaction Potential of Darolutamide: In Vitro and Clinical Studies

European Journal of Drug Metabolism and Pharmacokinetics ◽

10.1007/s13318-019-00577-5 ◽

2019 ◽

Vol 44 (6) ◽

pp. 747-759 ◽

Cited By ~ 13

Author(s):

Christian Zurth ◽

Mikko Koskinen ◽

Robert Fricke ◽

Olaf Prien ◽

Timo Korjamo ◽

...

Keyword(s):

Drug Interaction ◽

Interaction Potential ◽

Clinical Studies ◽

Drug Drug Interaction

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In Vitro and Clinical Evaluations of the Drug-Drug Interaction Potential of a Metabotropic Glutamate 2/3 Receptor Agonist Prodrug with Intestinal Peptide Transporter 1

Drug Metabolism and Disposition ◽

10.1124/dmd.116.071118 ◽

2016 ◽

Vol 45 (2) ◽

pp. 137-144 ◽

Cited By ~ 4

Author(s):

Y. Anne Pak ◽

Amanda J. Long ◽

William F. Annes ◽

Jennifer W. Witcher ◽

Mary Pat Knadler ◽

...

Keyword(s):

Drug Interaction ◽

Interaction Potential ◽

Receptor Agonist ◽

Peptide Transporter ◽

Metabotropic Glutamate ◽

Clinical Evaluations ◽

Drug Drug Interaction ◽

Peptide Transporter 1

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ERRATA: Evaluation of Drug-drug Interaction Potential of Beraprost Sodium Mediated by P450 In Vitro

YAKUGAKU ZASSHI ◽

10.1248/yakushi.130.277 ◽

2010 ◽

Vol 130 (2) ◽

pp. 277-277

Author(s):

Tominaga FUKAZAWA ◽

Kanako YAJIMA ◽

Yohei MIYAMOTO

Keyword(s):

Drug Interaction ◽

Interaction Potential ◽

Beraprost Sodium ◽

Drug Drug Interaction

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In vitro–in vivo correlation of the drug–drug interaction potential of antiretroviral HIV treatment regimens on CYP1A1 substrate riociguat

Expert Opinion on Drug Metabolism & Toxicology ◽

10.1080/17425255.2019.1681968 ◽

2019 ◽

Vol 15 (11) ◽

pp. 975-984 ◽

Cited By ~ 2

Author(s):

Natalia A. Jungmann ◽

Dieter Lang ◽

Soundos Saleh ◽

Dorina Van Der Mey ◽

Michael Gerisch

Keyword(s):

Drug Interaction ◽

Interaction Potential ◽

Hiv Treatment ◽

Treatment Regimens ◽

Drug Drug Interaction

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In vitro and physiologically‐based pharmacokinetic based assessment of drug–drug interaction potential of canagliflozin

British Journal of Clinical Pharmacology ◽

10.1111/bcp.13186 ◽

2016 ◽

Vol 83 (5) ◽

pp. 1082-1096 ◽

Cited By ~ 6

Author(s):

Rao N. V. S. Mamidi ◽

Shannon Dallas ◽

Carlo Sensenhauser ◽

Heng Keang Lim ◽

Ellen Scheers ◽

...

Keyword(s):

Drug Interaction ◽

Interaction Potential ◽

Physiologically Based Pharmacokinetic ◽

Physiologically Based ◽

Drug Drug Interaction

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INVESTIGATION OF DRUG-DRUG INTERACTION POTENTIAL OF BORTEZOMIB IN VIVO IN FEMALE SPRAGUE-DAWLEY RATS AND IN VITRO IN HUMAN LIVER MICROSOMES

Drug Metabolism and Disposition ◽

10.1124/dmd.105.008060 ◽

2006 ◽

Vol 34 (4) ◽

pp. 702-708 ◽

Cited By ~ 23

Author(s):

Chuang Lu ◽

Richard Gallegos ◽

Ping Li ◽

Cindy Q. Xia ◽

Sandeepraj Pusalkar ◽

...

Keyword(s):

Drug Interaction ◽

Interaction Potential ◽

Human Liver ◽

Liver Microsomes ◽

Human Liver Microsomes ◽

Sprague Dawley ◽

Sprague Dawley Rats ◽

Drug Drug Interaction

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Drug–Drug Interaction Potential of Marketed Oncology Drugs: In Vitro Assessment of Time-Dependent Cytochrome P450 Inhibition, Reactive Metabolite Formation and Drug–Drug Interaction Prediction

Pharmaceutical Research ◽

10.1007/s11095-012-0724-6 ◽

2012 ◽

Vol 29 (7) ◽

pp. 1960-1976 ◽

Cited By ~ 61

Author(s):

Jane R. Kenny ◽

Sophie Mukadam ◽

Chenghong Zhang ◽

Suzanne Tay ◽

Carol Collins ◽

...

Keyword(s):

Cytochrome P450 ◽

Drug Interaction ◽

Interaction Potential ◽

Time Dependent ◽

Reactive Metabolite ◽

Metabolite Formation ◽

Interaction Prediction ◽

In Vitro Assessment ◽

Drug Drug Interaction

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Response to in vitro and physiologically-based pharmacokinetic assessment of the drug-drug interaction potential of canagliflozin

British Journal of Clinical Pharmacology ◽

10.1111/bcp.13443 ◽

2017 ◽

Vol 84 (2) ◽

pp. 392-393

Author(s):

John O. Miners ◽

Attarat Pattanawongsa ◽

Andrew Rowland

Keyword(s):

Drug Interaction ◽

Interaction Potential ◽

Physiologically Based Pharmacokinetic ◽

Pharmacokinetic Assessment ◽

Physiologically Based ◽

Drug Drug Interaction

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Evaluation of Drug-drug Interaction Potential of Beraprost Sodium Mediated by P450 In Vitro

YAKUGAKU ZASSHI ◽

10.1248/yakushi.128.1459 ◽

2008 ◽

Vol 128 (10) ◽

pp. 1459-1465 ◽

Cited By ~ 8

Author(s):

Tominaga FUKAZAWA ◽

Kanako YAJIMA ◽

Yohei MIYAMOTO

Keyword(s):

Drug Interaction ◽

Interaction Potential ◽

Beraprost Sodium ◽

Drug Drug Interaction

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Preliminary in vitro approach to evaluate the drug-drug interaction potential of EST73502, a dual µ-opioid receptor partial agonist and σ1 receptor antagonist

Xenobiotica ◽

10.1080/00498254.2021.1877850 ◽

2021 ◽

pp. 1-12

Author(s):

Eva Ayet ◽

Sandra Yeste ◽

Raquel F. Reinoso ◽

María José Pretel ◽

Ariadna Balada ◽

...

Keyword(s):

Drug Interaction ◽

Receptor Antagonist ◽

Opioid Receptor ◽

Interaction Potential ◽

Partial Agonist ◽

Σ1 Receptor ◽

Drug Drug Interaction

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In Vitro Assessment of the Drug-Drug Interaction Potential of Verinurad and its Metabolites as Substrates and Inhibitors of Metabolizing Enzymes and Drug Transporters

Journal of Pharmacology and Experimental Therapeutics ◽

10.1124/jpet.121.000549 ◽

2021 ◽

pp. JPET-AR-2021-000549

Author(s):

V. Sashi Gopaul ◽

Anna Vildhede ◽

Tommy B Andersson ◽

Fredrik Erlandsson ◽

Caroline A. Lee ◽

...

Keyword(s):

Drug Interaction ◽

Interaction Potential ◽

Drug Transporters ◽

Metabolizing Enzymes ◽

In Vitro Assessment ◽

Drug Drug Interaction

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