Improving the inhibitory activity of arylidenaminoguanidine compounds at the N-methyl-d-aspartate receptor complex from a recursive computational-experimental structure–activity relationship study

Activity Relationship ◽

Receptor Complex ◽

Aspartate Receptor ◽

Structure Activity ◽

Relationship Study ◽

Experimental Structure

Synthesis and Structure-activity Relationship Study of 2,4-dioxothiazolidin-5-ylidene Derivatives for 15-hydroxyprostaglandin Dehydrogenase Inhibitory Activity, Prostaglandin E2 Release, and Wound Healing Effect

Biotechnology and Bioprocess Engineering ◽

10.1007/s12257-021-0071-8 ◽

2021 ◽

Author(s):

EunJeong Yoon ◽

DuBok Choi ◽

InSun Yu ◽

Hoon Cho

Keyword(s):

Wound Healing ◽

Prostaglandin E2 ◽

Inhibitory Activity ◽

Activity Relationship ◽

Healing Effect ◽

Structure Activity ◽

Wound Healing Effect ◽

Synthesis, topoisomerase I and II inhibitory activity, cytotoxicity, and structure–activity relationship study of hydroxylated 2,4-diphenyl-6-aryl pyridines

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2010.03.051 ◽

2010 ◽

Vol 18 (9) ◽

pp. 3066-3077 ◽

Cited By ~ 68

Author(s):

Radha Karki ◽

Pritam Thapa ◽

Mi Jeong Kang ◽

Tae Cheon Jeong ◽

Jung Min Nam ◽

...

Keyword(s):

Inhibitory Activity ◽

Topoisomerase I ◽

Activity Relationship ◽

Structure Activity ◽

Dihydroxylated 2,4,6-triphenyl pyridines: Synthesis, topoisomerase I and II inhibitory activity, cytotoxicity, and structure–activity relationship study

European Journal of Medicinal Chemistry ◽

10.1016/j.ejmech.2012.01.015 ◽

2012 ◽

Vol 49 ◽

pp. 219-228 ◽

Cited By ~ 49

Author(s):

Radha Karki ◽

Pritam Thapa ◽

Han Young Yoo ◽

Tara Man Kadayat ◽

Pil-Hoon Park ◽

...

Keyword(s):

Inhibitory Activity ◽

Topoisomerase I ◽

Activity Relationship ◽

Structure Activity ◽

Positive Modulators of the N-Methyl-d-aspartate Receptor: Structure–Activity Relationship Study of Steroidal 3-Hemiesters

Journal of Medicinal Chemistry ◽

10.1021/acs.jmedchem.8b00255 ◽

2018 ◽

Vol 61 (10) ◽

pp. 4505-4516 ◽

Cited By ~ 7

Author(s):

Barbora Krausova ◽

Barbora Slavikova ◽

Michaela Nekardova ◽

Pavla Hubalkova ◽

Vojtech Vyklicky ◽

...

Keyword(s):

Activity Relationship ◽

Receptor Structure ◽

Aspartate Receptor ◽

Structure Activity ◽

Quantitative structure-activity relationship study of bitter di- and tri-peptides including relationship with angiotensin I-converting enzyme inhibitory activity

Journal of Peptide Science ◽

10.1002/psc.800 ◽

2006 ◽

Vol 13 (1) ◽

pp. 63-69 ◽

Cited By ~ 55

Author(s):

Jianping Wu ◽

Rotimi E. Aluko

Keyword(s):

Inhibitory Activity ◽

Quantitative Structure Activity Relationship ◽

Activity Relationship ◽

Converting Enzyme ◽

Quantitative Structure ◽

Angiotensin I ◽

Angiotensin I Converting Enzyme ◽

Structure Activity ◽

Design, synthesis, topoisomerase I & II inhibitory activity, antiproliferative activity, and structure–activity relationship study of pyrazoline derivatives: An ATP-competitive human topoisomerase IIα catalytic inhibitor

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2016.03.017 ◽

2016 ◽

Vol 24 (8) ◽

pp. 1898-1908 ◽

Cited By ~ 14

Author(s):

Pervez Ahmad ◽

Hyunjung Woo ◽

Kyu-Yeon Jun ◽

Adnan A. Kadi ◽

Hatem A. Abdel-Aziz ◽

...

Keyword(s):

Antiproliferative Activity ◽

Inhibitory Activity ◽

Topoisomerase I ◽

Activity Relationship ◽

Topoisomerase Iiα ◽

Design Synthesis ◽

Structure Activity ◽

Catalytic Inhibitor ◽

ChemInform Abstract: Dihydroxylated 2,4,6-Triphenyl Pyridines: Synthesis, Topoisomerase I and II Inhibitory Activity, Cytotoxicity, and Structure-Activity Relationship Study.

ChemInform ◽

10.1002/chin.201231150 ◽

2012 ◽

Vol 43 (31) ◽

pp. no-no

Author(s):

Eung-Seok Lee ◽

et al. et al.

Keyword(s):

Inhibitory Activity ◽

Topoisomerase I ◽

Activity Relationship ◽

Structure Activity ◽

QUANTITATIVE STRUCTURE ACTIVITY RELATIONSHIP STUDY ON THE INHIBITORY ACTIVITY OF COPPER SCHIFF BASE COMPLEXES AGAINST CANDIDA ALBICAN

The Journal of Engineering and Exact Sciences ◽

10.18540/jcecvl5iss1pp0111-0124 ◽

2019 ◽

Vol 5 (1) ◽

pp. 0111-0124

Author(s):

Umma Muhammad ◽

Adamu Uzairu ◽

Sulaiman Ola Idris

Keyword(s):

Schiff Base ◽

Inhibitory Activity ◽

Quantitative Structure Activity Relationship ◽

Schiff Base Complexes ◽

Activity Relationship ◽

Quantitative Structure ◽

Structure Activity ◽

Synthesis, Topoisomerase I and II Inhibitory Activity, Cytotoxicity, and Structure-activity Relationship Study of Rigid Analogues of 2,4,6-Trisubstituted Pyridine Containing 5,6-Dihydrobenzo[h]quinoline Moiety

Bulletin of the Korean Chemical Society ◽

10.5012/bkcs.2011.32.1.303 ◽

2011 ◽

Vol 32 (1) ◽

pp. 303-306 ◽

Cited By ~ 18

Author(s):

Byeong-Seon Jeong ◽

Ho-Young Choi ◽

Pritam Thapa ◽

Radha Karki ◽

Eun-Young Lee ◽

...

Keyword(s):

Inhibitory Activity ◽

Topoisomerase I ◽

Activity Relationship ◽

Structure Activity ◽

Relationship Study ◽

Quinoline Moiety

ChemInform Abstract: Synthesis, Topoisomerase I and II Inhibitory Activity, Cytotoxicity, and Structure-Activity Relationship Study of Rigid Analogues of 2,4,6-Trisubstituted Pyridine Containing 5,6-Dihydrobenzo[h]quinoline Moiety.

ChemInform ◽

10.1002/chin.201124151 ◽

2011 ◽

Vol 42 (24) ◽

pp. no-no

Author(s):

Eung-Seok Lee ◽

et al. et al.

Keyword(s):

Inhibitory Activity ◽

Topoisomerase I ◽

Activity Relationship ◽

Structure Activity ◽

Relationship Study ◽

Quinoline Moiety