Design, Synthesis and Biological Evaluation of Novel Acridine and Quinoline Derivatives as Tubulin Polymerization Inhibitors with Anticancer Activities

Design, Synthesis and Biological Evaluation of Benz‐Fused Five‐Membered Heterocyclic Compounds as Tubulin Polymerization Inhibitors with Anticancer Activities

Chemical Biology & Drug Design ◽

10.1111/cbdd.13832 ◽

2021 ◽

Author(s):

Buduma Komuraiah ◽

Yichang Ren ◽

Mingming Xue ◽

Binbin Cheng ◽

Jin Liu ◽

...

Keyword(s):

Heterocyclic Compounds ◽

Biological Evaluation ◽

Tubulin Polymerization ◽

Anticancer Activities ◽

Design Synthesis ◽

Design, Synthesis and Biological Evaluation of 1,4-Disubstituted-3,4-dihydroisoquinoline Compounds as New Tubulin Polymerization Inhibitors

International Journal of Molecular Sciences ◽

10.3390/ijms160510173 ◽

2015 ◽

Vol 16 (12) ◽

pp. 10173-10184 ◽

Cited By ~ 1

Author(s):

Ling Zhang ◽

Yunlong Song ◽

Jingjing Huang ◽

Jia Liu ◽

Wenwen Zhu ◽

...

Keyword(s):

Biological Evaluation ◽

Tubulin Polymerization ◽

Design Synthesis ◽

3,5-Diaryl-1H-pyrazolo[3,4-b]pyridines as potent tubulin polymerization inhibitors: Rational design, synthesis and biological evaluation

European Journal of Medicinal Chemistry ◽

10.1016/j.ejmech.2018.12.053 ◽

2019 ◽

Vol 168 ◽

pp. 426-435 ◽

Cited By ~ 14

Author(s):

Min'an Zhai ◽

Shiyuan Liu ◽

Meiqi Gao ◽

Long Wang ◽

Jun Sun ◽

...

Keyword(s):

Rational Design ◽

Biological Evaluation ◽

Tubulin Polymerization ◽

Design Synthesis ◽

Design, synthesis and biological evaluation of novel vicinal diaryl-substituted 1H-Pyrazole analogues of combretastatin A-4 as highly potent tubulin polymerization inhibitors

European Journal of Medicinal Chemistry ◽

10.1016/j.ejmech.2019.111577 ◽

2019 ◽

Vol 181 ◽

pp. 111577 ◽

Cited By ~ 8

Author(s):

Romeo Romagnoli ◽

Paola Oliva ◽

Maria Kimatrai Salvador ◽

Maria Encarnacion Camacho ◽

Chiara Padroni ◽

...

Keyword(s):

Biological Evaluation ◽

Tubulin Polymerization ◽

Design Synthesis ◽

Design, synthesis and biological evaluation of novel 5,6,7-trimethoxy-N-aryl-2-styrylquinolin-4-amines as potential anticancer agents and tubulin polymerization inhibitors

Bioorganic Chemistry ◽

10.1016/j.bioorg.2020.103711 ◽

2020 ◽

Vol 98 ◽

pp. 103711 ◽

Cited By ~ 1

Author(s):

Salimeh Mirzaei ◽

Farhad Eisvand ◽

Farzin Hadizadeh ◽

Fatemeh Mosaffa ◽

Ali Ghasemi ◽

...

Keyword(s):

Anticancer Agents ◽

Biological Evaluation ◽

Tubulin Polymerization ◽

Design Synthesis ◽

Design, synthesis and biological evaluation of resveratrol-cinnamoyl derivates as tubulin polymerization inhibitors targeting the colchicine binding site

Bioorganic Chemistry ◽

10.1016/j.bioorg.2019.103319 ◽

2019 ◽

Vol 93 ◽

pp. 103319 ◽

Cited By ~ 3

Author(s):

Yong Yin ◽

Bao-Ping Lian ◽

Yuan-Zheng Xia ◽

Yu-Ying Shao ◽

Ling-Yi Kong

Keyword(s):

Binding Site ◽

Biological Evaluation ◽

Tubulin Polymerization ◽

Design Synthesis ◽

Colchicine Binding Site ◽

Design, synthesis and biological evaluation of novel indole-based oxalamide and aminoacetamide derivatives as tubulin polymerization inhibitors

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/j.bmcl.2019.126816 ◽

2020 ◽

Vol 30 (2) ◽

pp. 126816 ◽

Cited By ~ 1

Author(s):

Peng-Cheng Diao ◽

Xie-Er Jian ◽

Peng Chen ◽

Chuan Huang ◽

Jie Yin ◽

...

Keyword(s):

Biological Evaluation ◽

Tubulin Polymerization ◽

Design Synthesis ◽

Design, synthesis and biological evaluation of 2-phenylquinoline-4-carboxamide derivatives as a new class of tubulin polymerization inhibitors

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2017.09.004 ◽

2017 ◽

Vol 25 (21) ◽

pp. 5939-5951 ◽

Cited By ~ 6

Author(s):

Li Zhu ◽

Kaixiu Luo ◽

Ke Li ◽

Yi Jin ◽

Jun Lin

Keyword(s):

Biological Evaluation ◽

Tubulin Polymerization ◽

Design Synthesis ◽

New Class ◽

Design, synthesis and biological evaluation of (E)-3-(3,4-dihydroxyphenyl)acrylylpiperazine derivatives as a new class of tubulin polymerization inhibitors

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2014.05.029 ◽

2014 ◽

Vol 22 (15) ◽

pp. 4285-4292 ◽

Cited By ~ 9

Author(s):

Yong Yin ◽

Fang Qiao ◽

Lu-Yi Jiang ◽

She-Feng Wang ◽

Shao Sha ◽

...

Keyword(s):

Biological Evaluation ◽

Tubulin Polymerization ◽

Design Synthesis ◽

New Class ◽

Design, synthesis, and biological evaluation of 2,3‐diphenyl‐cycloalkyl pyrazole derivatives as potential tubulin polymerization inhibitors

Chemical Biology & Drug Design ◽

10.1111/cbdd.13565 ◽

2019 ◽

Vol 94 (5) ◽

pp. 1894-1904

Author(s):

Lin‐Ying Xia ◽

Rong Yang ◽

Ya‐Liang Zhang ◽

Yi‐Chun Chu ◽

Ya‐Lin Qi ◽

...

Keyword(s):

Biological Evaluation ◽

Tubulin Polymerization ◽

Pyrazole Derivatives ◽

Design Synthesis ◽