Synthesis of cinnamic acids and related isosteres as potent and selective αvβ3 receptor antagonists

2004 ◽  
Vol 14 (6) ◽  
pp. 1471-1476 ◽  
Author(s):  
Thomas D. Penning ◽  
Mark A. Russell ◽  
Barbara B. Chen ◽  
Helen Y. Chen ◽  
Bipin N. Desai ◽  
...  
Keyword(s):  
Cinnamic Acids ◽  
Receptor Antagonists ◽  
Αvβ3 Receptor

Cinnamic acids and mono-substituted benzoic acids as useful capping groups for the preparation of hNK2 receptor antagonists

2008 ◽  
Vol 18 (16) ◽  
pp. 4705-4707 ◽  
Author(s):  
Marina Porcelloni ◽  
Piero D’Andrea ◽  
Maria Altamura ◽  
Rose-Marie Catalioto ◽  
Sandro Giuliani ◽  
...  
Keyword(s):  
Benzoic Acids ◽  
Cinnamic Acids ◽  
Receptor Antagonists ◽  
Substituted Benzoic Acids

Synthesis of pyrazoles and isoxazoles as potent αvβ3 receptor antagonists

2006 ◽  
Vol 16 (12) ◽  
pp. 3156-3161 ◽  
Author(s):  
Thomas D. Penning ◽  
Albert Khilevich ◽  
Barbara B. Chen ◽  
Mark A. Russell ◽  
Mark L. Boys ◽  
...  
Keyword(s):  
Receptor Antagonists ◽  
Αvβ3 Receptor

Highly potent and selective αVβ3-receptor antagonists: solid-phase synthesis and SAR of 1-substituted 4-amino-1H-pyrimidin-2-ones

2003 ◽  
Vol 13 (2) ◽  
pp. 165-169 ◽  
Author(s):  
Christian Zechel ◽  
Gisela Backfisch ◽  
Jürgen Delzer ◽  
Hervé Geneste ◽  
Claudia Graef ◽  
...  
Keyword(s):  
Solid Phase Synthesis ◽  
Solid Phase ◽  
Receptor Antagonists ◽  
Phase Synthesis ◽  
Αvβ3 Receptor

Synthesis of Pyrazoles and Isoxazoles as Potent αvβ3 Receptor Antagonists.

ChemInform ◽  
2006 ◽  
Vol 37 (37) ◽  
Author(s):  
Thomas D. Penning ◽  
et al. et al.
Keyword(s):  
Receptor Antagonists ◽  
Αvβ3 Receptor

Synthesis of highly potent and selective hetaryl ureas as integrin αVβ3-Receptor antagonists

2002 ◽  
Vol 12 (10) ◽  
pp. 1379-1382 ◽  
Author(s):  
Udo E.W. Lange ◽  
Gisela Backfisch ◽  
Jürgen Delzer ◽  
Hervé Geneste ◽  
Claudia Graef ◽  
...  
Keyword(s):  
Integrin Αvβ3 ◽  
Receptor Antagonists ◽  
Αvβ3 Receptor

Convergent, parallel synthesis of a series of β-substituted 1,2,4-oxadiazole butanoic acids as potent and selective αvβ3 receptor antagonists

2006 ◽  
Vol 16 (4) ◽  
pp. 839-844 ◽  
Author(s):  
Mark L. Boys ◽  
Lori A. Schretzman ◽  
Nizal S. Chandrakumar ◽  
Michael B. Tollefson ◽  
Scott B. Mohler ◽  
...  
Keyword(s):  
Parallel Synthesis ◽  
Receptor Antagonists ◽  
Αvβ3 Receptor

Design, Synthesis, and Evaluation of Radiolabeled Integrin αvβ3 Receptor Antagonists for Tumor Imaging and Radiotherapy

2003 ◽  
Vol 18 (4) ◽  
pp. 627-641 ◽  
Author(s):  
Thomas D. Harris ◽  
Shirley Kalogeropoulos ◽  
Tiffany Nguyen ◽  
Shuang Liu ◽  
Judit Bartis ◽  
...  
Keyword(s):  
Tumor Imaging ◽  
Integrin Αvβ3 ◽  
Receptor Antagonists ◽  
Design Synthesis ◽  
Αvβ3 Receptor
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