Identification of C10 nitrogen-containing aporphines with dopamine D1 versus D5 receptor selectivity

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/j.bmcl.2020.127053 ◽

2020 ◽

Vol 30 (8) ◽

pp. 127053 ◽

Author(s):

Anupam Karki ◽

Reecan Juarez ◽

Hari K. Namballa ◽

Ian Alberts ◽

Wayne W. Harding

Keyword(s):

Receptor Selectivity

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In vivo demonstration of muscarinic receptor selectivity of fesoterodine active metabolite, 5-hydroxymethl tolterodine (5-HMT), in rat tissue

10.26226/morressier.59b63e3fd462b8029238928f ◽

2017 ◽

Author(s):

Yoshihiko Ito

Keyword(s):

Muscarinic Receptor ◽

Active Metabolite ◽

Receptor Selectivity ◽

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Type and location of fluorescent probes incorporated into the potent mu-opioid peptide [Dmt1]DALDA affect potency, receptor selectivity and intrinsic efficacy*

Journal of Peptide Research ◽

10.1111/j.1399-3011.2005.00252.x ◽

2005 ◽

Vol 65 (6) ◽

pp. 556-563 ◽

Author(s):

P.W. Schiller ◽

I. Berezowska ◽

G. Weltrowska ◽

H. Chen ◽

C. Lemieux ◽

...

Keyword(s):

Fluorescent Probes ◽

Opioid Peptide ◽

Receptor Selectivity ◽

Mu Opioid ◽

Intrinsic Efficacy

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Multiple N-Methylation by a Designed Approach Enhances Receptor Selectivity

Journal of Medicinal Chemistry ◽

10.1021/jm701044r ◽

2007 ◽

Vol 50 (24) ◽

pp. 5878-5881 ◽

Author(s):

Jayanta Chatterjee ◽

Oded Ovadia ◽

Grit Zahn ◽

Luciana Marinelli ◽

Amnon Hoffman ◽

...

Keyword(s):

Receptor Selectivity

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A Proteomic Microarray Approach for Exploring Ligand-initiated Nuclear Hormone Receptor Pharmacology, Receptor Selectivity, and Heterodimer Functionality

Molecular & Cellular Proteomics ◽

10.1074/mcp.m400192-mcp200 ◽

2004 ◽

Vol 4 (3) ◽

pp. 267-277 ◽

Author(s):

Sung Hoon Kim ◽

Anobel Tamrazi ◽

Kathryn E. Carlson ◽

John A. Katzenellenbogen

Keyword(s):

Hormone Receptor ◽

Nuclear Hormone Receptor ◽

Receptor Selectivity ◽

Receptor Pharmacology

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Flupentixol and dopamine receptor selectivity

Psychopharmacology ◽

10.1007/bf00432192 ◽

1981 ◽

Vol 75 (2) ◽

pp. 217-217 ◽

Author(s):

John Hyttel

Keyword(s):

Dopamine Receptor ◽

Receptor Selectivity

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Modification of Receptor Selectivity and Functional Activity in Cholecystokinin Peptoid Ligands

Journal of Medicinal Chemistry ◽

10.1021/jm00017a022 ◽

1995 ◽

Vol 38 (17) ◽

pp. 3384-3390 ◽

Author(s):

Milana Dezube ◽

Elizabeth E. Sugg ◽

Larry S. Birkemo ◽

Dallas K. Croom ◽

Robert W. Dougherty ◽

...

Keyword(s):

Functional Activity ◽

Receptor Selectivity

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Receptor selectivity of cholecystokinin effects on mesoaccumbens dopamine neurons

Synapse ◽

10.1002/syn.890080207 ◽

1991 ◽

Vol 8 (2) ◽

pp. 137-143 ◽

Author(s):

Mark D. Kelland ◽

Jing Zhang ◽

Louis A. Chiodo ◽

Arthur S. Freeman

Keyword(s):

Dopamine Neurons ◽

Receptor Selectivity

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Crystal Structures of the GluR5 and GluR6 Ligand Binding Cores: Molecular Mechanisms Underlying Kainate Receptor Selectivity

Neuron ◽

10.1016/j.neuron.2005.01.031 ◽

2005 ◽

Vol 45 (4) ◽

pp. 539-552 ◽

Author(s):

Mark L. Mayer

Keyword(s):

Ligand Binding ◽

Crystal Structures ◽

Molecular Mechanisms ◽

Kainate Receptor ◽

Receptor Selectivity

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Synthesis of 3H-deltorphin analogues with high δ opioid receptor selectivity and high specific radioactivity

Peptides 1992 ◽

10.1007/978-94-011-1470-7_296 ◽

1993 ◽

pp. 653-654

Author(s):

Géza Tóth ◽

Ferenc Ötvös ◽

Katalin Soós ◽

Libor Havlicek ◽

Beáta Búzás ◽

...

Keyword(s):

Opioid Receptor ◽

Specific Radioactivity ◽

Receptor Selectivity ◽

High Specific Radioactivity ◽

Δ Opioid Receptor ◽

Opioid Receptor Selectivity

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Role of positions 9 and 10 in the desensitizing and receptor selectivity properties of endothelin-1

Peptides 1994 ◽

10.1007/978-94-011-1468-4_293 ◽

1995 ◽

pp. 642-643

Author(s):

N. Miasiro ◽

R. de Castiglione ◽

A. C. M. Paiva

Keyword(s):

Receptor Selectivity ◽

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