GABAA Receptor Subtype Selectivity of the Proconvulsant Rodenticide TETS

Biophysical Journal ◽

10.1016/j.bpj.2017.11.1756 ◽

2018 ◽

Vol 114 (3) ◽

pp. 310a-311a

Author(s):

Brandon Pressly ◽

Hai Minh Nguyen ◽

Heike Wulff

Keyword(s):

Gabaa Receptor ◽

Receptor Subtype ◽

Subtype Selectivity

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Dose-Dependent EEG Effects of Zolpidem Provide Evidence for GABAA Receptor Subtype Selectivity in Vivo

Journal of Pharmacology and Experimental Therapeutics ◽

10.1124/jpet.102.044859 ◽

2002 ◽

Vol 304 (3) ◽

pp. 1251-1257 ◽

Author(s):

S. A. G. Visser ◽

F. L. C. Wolters ◽

P. H. van der Graaf ◽

L. A. Peletier ◽

M. Danhof

Keyword(s):

Gabaa Receptor ◽

Receptor Subtype ◽

Subtype Selectivity ◽

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GABAA receptor subtype selectivity of the proconvulsant rodenticide TETS

Archives of Toxicology ◽

10.1007/s00204-017-2089-4 ◽

2017 ◽

Vol 92 (2) ◽

pp. 833-844 ◽

Author(s):

Brandon Pressly ◽

Hai M. Nguyen ◽

Heike Wulff

Keyword(s):

Gabaa Receptor ◽

Receptor Subtype ◽

Subtype Selectivity

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GABAA receptor subtype selectivity underlying selective anxiolytic effect of baicalin

Neuropharmacology ◽

10.1016/j.neuropharm.2008.07.040 ◽

2008 ◽

Vol 55 (7) ◽

pp. 1231-1237 ◽

Author(s):

Feng Wang ◽

Zhiwen Xu ◽

Lihuan Ren ◽

Shui Ying Tsang ◽

Hong Xue

Keyword(s):

Gabaa Receptor ◽

Anxiolytic Effect ◽

Receptor Subtype ◽

Subtype Selectivity

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GABAA receptor subtype selectivity underlying anxiolytic effect of 6-hydroxyflavone

Biochemical Pharmacology ◽

10.1016/j.bcp.2009.12.024 ◽

2010 ◽

Vol 79 (9) ◽

pp. 1337-1344 ◽

Author(s):

Lihuan Ren ◽

Feng Wang ◽

Zhiwen Xu ◽

Wing Man Chan ◽

Cunyou Zhao ◽

...

Keyword(s):

Gabaa Receptor ◽

Anxiolytic Effect ◽

Receptor Subtype ◽

Subtype Selectivity

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THE INFLUENCE OF 6-OXIME-, SEMICARBAZONE-, AND HYDRAZONE GROUPS SUBSTITUTIONS ON THE OPIOD RECEPTOR SUBTYPE-SELECTIVITY OF OXYCODONE DERIVATIVES

Analgesia ◽

10.3727/107156995819563582 ◽

1995 ◽

Vol 1 (4) ◽

pp. 425-428

Author(s):

Zsuzsanna Fürst ◽

Tamás Friedmann ◽

Sandor Hosztafi

Keyword(s):

Receptor Subtype ◽

Subtype Selectivity

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Synthesis and Structure−Activity Relationships of 2-Substitutedd-Tryptophan-Containing Peptidic Endothelin Receptor Antagonists: Importance of the C-2 Substituent of thed-Tryptophan Residue for Endothelin A and B Receptor Subtype Selectivity

Journal of Medicinal Chemistry ◽

10.1021/jm9600914 ◽

1996 ◽

Vol 39 (12) ◽

pp. 2313-2330 ◽

Author(s):

Takehiro Fukami ◽

Takeru Yamakawa ◽

Kenji Niiyama ◽

Hisaki Kojima ◽

Yuuka Amano ◽

...

Keyword(s):

Tryptophan Residue ◽

Receptor Subtype ◽

Endothelin Receptor Antagonists ◽

Endothelin Receptor ◽

Receptor Antagonists ◽

Structure Activity Relationships ◽

Subtype Selectivity ◽

Structure Activity ◽

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Diazepam-induced changes in sleep: Role of the 1 GABAA receptor subtype

Proceedings of the National Academy of Sciences ◽

10.1073/pnas.111055398 ◽

2001 ◽

Vol 98 (11) ◽

pp. 6464-6469 ◽

Author(s):

I. Tobler ◽

C. Kopp ◽

T. Deboer ◽

U. Rudolph

Keyword(s):

Gabaa Receptor ◽

Receptor Subtype ◽

Induced Changes

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Modulation of PPAR receptor subtype selectivity of the ligands: Aliphatic chain vs aromatic ring as a spacer between pharmacophore and the lipophilic moiety

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/j.bmcl.2008.10.062 ◽

2008 ◽

Vol 18 (24) ◽

pp. 6471-6475 ◽

Author(s):

Harikishore Pingali ◽

Mukul Jain ◽

Shailesh Shah ◽

Pravin Patil ◽

Pankaj Makadia ◽

...

Keyword(s):

Aromatic Ring ◽

Receptor Subtype ◽

Aliphatic Chain ◽

Subtype Selectivity

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Thiochrome Enhances Acetylcholine Affinity at Muscarinic M4 Receptors: Receptor Subtype Selectivity via Cooperativity Rather than Affinity

Molecular Pharmacology ◽

10.1124/mol.65.1.257 ◽

2004 ◽

Vol 65 (1) ◽

pp. 257-266 ◽

Author(s):

S. Lazareno ◽

V. Doležal ◽

A. Popham ◽

N. J. M. Birdsall

Keyword(s):

Receptor Subtype ◽

Subtype Selectivity

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Strain differences in the effects of GABAA receptor subtype selective compounds in the mouse light-dark test

European Neuropsychopharmacology ◽

10.1016/s0924-977x(06)80049-0 ◽

2006 ◽

Vol 16 ◽

pp. S40-S41 ◽

Author(s):

L. Mathiasen ◽

N.R. Mirza ◽

R.J. Rodgers

Keyword(s):

Gabaa Receptor ◽

Strain Differences ◽

Receptor Subtype ◽

Subtype Selective

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