scholarly journals Structure–activity relationships of novel substituted naphthalene diimides as anticancer agents

2012 ◽  
Vol 57 ◽  
pp. 417-428 ◽  
Author(s):  
Andrea Milelli ◽  
Vincenzo Tumiatti ◽  
Marialuisa Micco ◽  
Michela Rosini ◽  
Guendalina Zuccari ◽  
...  
Keyword(s):  
Anticancer Agents ◽  
Structure Activity Relationships ◽  
Structure Activity ◽  
Naphthalene Diimides

Design, synthesis and biological activities of pyrrole-3-carboxamide derivatives as EZH2 (enhancer of zeste homologue 2) inhibitors and anticancer agents

2020 ◽  
Vol 44 (6) ◽  
pp. 2247-2255
Author(s):  
Qifan Zhou ◽  
Lina Jia ◽  
Fangyu Du ◽  
Xiaoyu Dong ◽  
Wanyu Sun ◽  
...  
Keyword(s):  
Biological Activity ◽  
Anticancer Agents ◽  
Biological Activities ◽  
Activity Assay ◽  
Design Synthesis ◽  
Structure Activity Relationships ◽  
Structure Activity ◽  
Enhancer Of Zeste

A novel series of pyrrole-3-carboxamides targeting EZH2 have been designed and synthesized. The structure–activity relationships were summarized by combining with in vitro biological activity assay and docking results.

5-Cinnamoyl-6-aminouracil derivatives as novel anticancer agents. Synthesis, biological evaluation, and structure-activity relationships

1985 ◽  
Vol 28 (4) ◽  
pp. 497-502 ◽  
Author(s):  
Jean Luc Bernier ◽  
Jean Pierre Henichart ◽  
Vincent Warin ◽  
Chantal Trentesaux ◽  
Jean Claude Jardillier
Keyword(s):  
Anticancer Agents ◽  
Biological Evaluation ◽  
Structure Activity Relationships ◽  
Structure Activity

Largazole Analogues as Histone Deacetylase Inhibitors and Anticancer Agents: An Overview of Structure-Activity Relationships

ChemMedChem ◽  
2017 ◽  
Vol 12 (23) ◽  
pp. 1917-1926 ◽  
Author(s):  
Giulio Poli ◽  
Romano Di Fabio ◽  
Luca Ferrante ◽  
Vincenzo Summa ◽  
Maurizio Botta
Keyword(s):  
Histone Deacetylase ◽  
Anticancer Agents ◽  
Histone Deacetylase Inhibitors ◽  
Structure Activity Relationships ◽  
Structure Activity

ChemInform Abstract: Anthrapyrazole Anticancer Agents. Synthesis and Structure-Activity Relationships Against Murine Leukemias.

ChemInform ◽  
1987 ◽  
Vol 18 (24) ◽  
Author(s):  
H. D. H. SHOWALTER ◽  
J. L. JOHNSON ◽  
J. M. HOFTIEZER ◽  
W. R. TURNER ◽  
L. M. WERBEL ◽  
...  
Keyword(s):  
Anticancer Agents ◽  
Structure Activity Relationships ◽  
Structure Activity
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