Design, synthesis and biological evaluation of multivalent glucosides with high affinity as ligands for brain targeting liposomes

European Journal of Medicinal Chemistry ◽

10.1016/j.ejmech.2013.10.007 ◽

2014 ◽

Vol 72 ◽

pp. 110-118 ◽

Author(s):

Boyi Qu ◽

Xiaocen Li ◽

Mei Guan ◽

Xun Li ◽

Li Hai ◽

...

Keyword(s):

Biological Evaluation ◽

Brain Targeting ◽

Design Synthesis ◽

High Affinity ◽

Synthesis And Biological Evaluation

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Design, synthesis and biological evaluation of novel pyrrolo[2,3-d]pyrimidine as tumor-targeting agents with selectivity for tumor uptake by high affinity folate receptors over the reduced folate carrier

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2020.115544 ◽

2020 ◽

Vol 28 (12) ◽

pp. 115544 ◽

Author(s):

Lalit K. Golani ◽

Farhana Islam ◽

Carrie O'Connor ◽

Aamod S. Dekhne ◽

Zhanjun Hou ◽

...

Keyword(s):

Tumor Targeting ◽

Biological Evaluation ◽

Reduced Folate Carrier ◽

Tumor Uptake ◽

Design Synthesis ◽

Folate Receptors ◽

High Affinity ◽

Synthesis And Biological Evaluation

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Design, synthesis and biological evaluation for docetaxel-loaded brain targeting liposome with “lock-in” function

Journal of Drug Targeting ◽

10.3109/1061186x.2013.865032 ◽

2013 ◽

Vol 22 (3) ◽

pp. 251-261 ◽

Author(s):

Xiaocen Li ◽

Boyi Qu ◽

Xiuxiu Jin ◽

Li Hai ◽

Yong Wu

Keyword(s):

Biological Evaluation ◽

Brain Targeting ◽

Design Synthesis ◽

Lock In ◽

Synthesis And Biological Evaluation

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Rational Design, Synthesis and Biological Evaluation of Modular Fluorogenic Substrates with High Affinity and Selectivity for PTP1B

ChemBioChem ◽

10.1002/cbic.201400033 ◽

2014 ◽

Vol 15 (7) ◽

pp. 961-976 ◽

Author(s):

Silvano Sanchini ◽

Francesca Perruccio ◽

Grazia Piizzi

Keyword(s):

Rational Design ◽

Biological Evaluation ◽

Fluorogenic Substrates ◽

Design Synthesis ◽

High Affinity ◽

Synthesis And Biological Evaluation

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Design, synthesis and biological evaluation of brain targeting l-ascorbic acid prodrugs of ibuprofen with “lock-in” function

European Journal of Medicinal Chemistry ◽

10.1016/j.ejmech.2014.05.072 ◽

2014 ◽

Vol 82 ◽

pp. 314-323 ◽

Author(s):

Yi Zhao ◽

Boyi Qu ◽

Xueying Wu ◽

Xiaocen Li ◽

Qingqing Liu ◽

...

Keyword(s):

Ascorbic Acid ◽

Biological Evaluation ◽

Brain Targeting ◽

Design Synthesis ◽

Lock In ◽

Synthesis And Biological Evaluation

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Design, synthesis and biological evaluation of novel estrone phosphonates as high affinity organic anion-transporting polypeptide 2B1 (OATP2B1) inhibitors

Bioorganic Chemistry ◽

10.1016/j.bioorg.2021.104914 ◽

2021 ◽

pp. 104914

Author(s):

Rebeka Jójárt ◽

Réka Laczkó-Rigó ◽

Máté Klement ◽

Gabriella Kőhl ◽

Gábor Kecskeméti ◽

...

Keyword(s):

Organic Anion ◽

Biological Evaluation ◽

Design Synthesis ◽

Organic Anion Transporting Polypeptide ◽

High Affinity ◽

Synthesis And Biological Evaluation

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Design, Synthesis, and Biological Evaluation of Small, High-Affinity Siglec-7 Ligands: Toward Novel Inhibitors of Cancer Immune Evasion

Journal of Medicinal Chemistry ◽

10.1021/acs.jmedchem.6b01111 ◽

2017 ◽

Vol 60 (3) ◽

pp. 941-956 ◽

Author(s):

Horst Prescher ◽

Martin Frank ◽

Stephan Gütgemann ◽

Elena Kuhfeldt ◽

Astrid Schweizer ◽

...

Keyword(s):

Immune Evasion ◽

Biological Evaluation ◽

Design Synthesis ◽

High Affinity ◽

Synthesis And Biological Evaluation

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Neurochemistry of aging. 2. Design, synthesis and biological evaluation of halomethyl analogs of choline with high affinity choline transport inhibitory activity

Journal of Medicinal Chemistry ◽

10.1021/jm00111a016 ◽

1991 ◽

Vol 34 (7) ◽

pp. 2031-2036 ◽

Author(s):

Jehangir S. Mistry ◽

Donald J. Abraham ◽

Alan P. Kozikowski ◽

Israel Hanin

Keyword(s):

Inhibitory Activity ◽

Biological Evaluation ◽

Choline Transport ◽

Design Synthesis ◽

High Affinity ◽

Synthesis And Biological Evaluation

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ChemInform Abstract: Neurochemistry of Aging. Part 2. Design, Synthesis, and Biological Evaluation of Halomethyl Analogues of Choline with High Affinity Choline Transport Inhibitory Activity.

10.1002/chin.199152181 ◽

2010 ◽

Vol 22 (52) ◽

pp. no-no

Author(s):

J. S. MISTRY ◽

D. J. ABRAHAM ◽

A. P. KOZIKOWSKI ◽

I. HANIN

Keyword(s):

Inhibitory Activity ◽

Biological Evaluation ◽

Choline Transport ◽

Design Synthesis ◽

High Affinity ◽

Synthesis And Biological Evaluation

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Design, Synthesis and Biological Evaluation of some Chalcone Derivatives as Potential Pancreatic Lipase Inhibitors

10.3390/ecsoc-17-b024 ◽

2013 ◽

Author(s):

Dao Tran

Keyword(s):

Pancreatic Lipase ◽

Biological Evaluation ◽

Design Synthesis ◽

Chalcone Derivatives ◽

Pancreatic Lipase Inhibitors ◽

Synthesis And Biological Evaluation

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Faculty Opinions recommendation of Structure-Based Design, Synthesis, and Biological Evaluation of Highly Selective and Potent G Protein-Coupled Receptor Kinase 2 Inhibitors.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.726271231.793520213 ◽

2016 ◽

Author(s):

Miles Congreve ◽

Mark Pickworth

Keyword(s):

G Protein ◽

Biological Evaluation ◽

Receptor Kinase ◽

G Protein Coupled Receptor ◽

Design Synthesis ◽

G Protein Coupled ◽

Synthesis And Biological Evaluation

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