scholarly journals A lipid-anchored neurokinin 1 receptor antagonist prolongs pain relief by a three-pronged mechanism of action targeting the receptor at the plasma membrane and in endosomes

2021 ◽  
Vol 296 ◽  
pp. 100345
Author(s):  
Quynh N. Mai ◽  
Priyank Shenoy ◽  
Tim Quach ◽  
Jeffri S. Retamal ◽  
Arisbel B. Gondin ◽  
...  
Keyword(s):  
Plasma Membrane ◽  
Pain Relief ◽  
Receptor Antagonist ◽  
Mechanism Of Action ◽  
Neurokinin 1 Receptor ◽  
Neurokinin 1

An FDA Approved Neurokinin-1 Receptor Antagonist is Effective in Reducing Intraabdominal Adhesions when Administered Intraperitoneally, But Not Orally

2008 ◽  
Vol 12 (10) ◽  
pp. 1754-1761 ◽  
Author(s):  
Rizal Lim ◽  
Jonathan M. Morrill ◽  
Scott G. Prushik ◽  
Karen L. Reed ◽  
Adam C. Gower ◽  
...  
Keyword(s):  
Receptor Antagonist ◽  
Neurokinin 1 Receptor ◽  
Intraabdominal Adhesions ◽  
Neurokinin 1

Antitumoral action of the neurokinin-1 receptor antagonist L-733 060 on human melanoma cell lines

2004 ◽  
Vol 14 (3) ◽  
pp. 183-188 ◽  
Author(s):  
Miguel Mu??oz ◽  
Ana P??rez ◽  
Marisa Rosso ◽  
Carmen Zamarriego ◽  
Rosario Rosso
Keyword(s):  
Receptor Antagonist ◽  
Cell Lines ◽  
Melanoma Cell ◽  
Human Melanoma ◽  
Human Melanoma Cell ◽  
Neurokinin 1 Receptor ◽  
Neurokinin 1 ◽  
Antitumoral Action ◽  
Melanoma Cell Lines

Synthesis of the Neurokinin 1 Receptor Antagonist (+)-L-733,060 by Jacobsen’s Hydrolytic Kinetic Resolution

2020 ◽  
Vol 56 (12) ◽  
pp. 2159-2164
Author(s):  
D. N. Bhangare ◽  
V. B. Mahale ◽  
R. G. Shinde ◽  
M. D. Nikalje ◽  
S. D. Duthade ◽  
...  
Keyword(s):  
Receptor Antagonist ◽  
Kinetic Resolution ◽  
Neurokinin 1 Receptor ◽  
Hydrolytic Kinetic Resolution ◽  
Neurokinin 1

Effect of maropitant, a neurokinin 1 receptor antagonist, on anesthetic requirements during noxious visceral stimulation of the ovary in dogs

2011 ◽  
Vol 72 (12) ◽  
pp. 1576-1579 ◽  
Author(s):  
Pedro Boscan ◽  
Eric Monnet ◽  
Khursheed Mama ◽  
David C. Twedt ◽  
Jonathan Congdon ◽  
...  
Keyword(s):  
Receptor Antagonist ◽  
Neurokinin 1 Receptor ◽  
Neurokinin 1 ◽  
Stimulation Of
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