Synthesis and pharmacological evaluation of 6a,7-dihydro-6H,13H-pyrazino[1,2-a;4,5-a′]diindole analogs as melatonin receptor ligands

Tetrahedron ◽  
2007 ◽  
Vol 63 (3) ◽  
pp. 754-760 ◽  
Author(s):  
Mohamed I. Attia ◽  
Justin Julius ◽  
Paula A. Witt-Enderby ◽  
Darius P. Zlotos
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MT1-Selective Melatonin Receptor Ligands: Synthesis, Pharmacological Evaluation, and Molecular Dynamics Investigation ofN-{[(3-O-Substituted)anilino]alkyl}amides

ChemMedChem ◽  
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Vol 7 (11) ◽  
pp. 1954-1964 ◽  
Author(s):  
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Daniele Pala ◽  
Alessio Lodola ◽  
Marco Mor ◽  
Valeria Lucini ◽  
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scholarly journals The pharmacological evaluation of novel and high‐affinity melatonin receptor ligands

2008 ◽  
Vol 22 (S1) ◽  
Author(s):  
Paula Ann Witt‐Enderby ◽  
Justin Julius ◽  
Mohamed I Attia ◽  
Darius P Zlotos
Keyword(s):  
Melatonin Receptor ◽  
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Synthesis of 2(3H)-Benzoxazolone Derivatives as Potential Melatonin Receptor Ligands

Heterocycles ◽  
2003 ◽  
Vol 60 (12) ◽  
pp. 2621 ◽  
Author(s):  
Pascal Carato ◽  
Christophe Mésangeau ◽  
Jacques H. Poupaert ◽  
Saïd Yous
Keyword(s):  
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Receptor Ligands

Melatonin Receptor Ligands:  Synthesis of New Melatonin Derivatives and Comprehensive Comparative Molecular Field Analysis (CoMFA) Study

1998 ◽  
Vol 41 (20) ◽  
pp. 3831-3844 ◽  
Author(s):  
Marco Mor ◽  
Silvia Rivara ◽  
Claudia Silva ◽  
Fabrizio Bordi ◽  
Pier Vincenzo Plazzi ◽  
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Keyword(s):  
Field Analysis ◽  
Molecular Field ◽  
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Melatonin Receptor ◽  
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Molecular Field Analysis ◽  
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Nature ◽  
2020 ◽  
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pp. 609-614 ◽  
Author(s):  
Reed M. Stein ◽  
Hye Jin Kang ◽  
John D. McCorvy ◽  
Grant C. Glatfelter ◽  
Anthony J. Jones ◽  
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Benzodiazepine Receptor Ligands. 4. Synthesis and Pharmacological Evaluation of 3-Heteroaryl-8-chloropyrazolo[5,1-c][1,2,4]benzotriazine 5-Oxides

1999 ◽  
Vol 42 (12) ◽  
pp. 2218-2226 ◽  
Author(s):  
Annarella Costanzo ◽  
Gabriella Guerrini ◽  
Giovanna Ciciani ◽  
Fabrizio Bruni ◽  
Silvia Selleri ◽  
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Keyword(s):  
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Receptor Ligands ◽  
Benzodiazepine Receptor Ligands ◽  
Pharmacological Evaluation
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