Synthesis, NMR conformational analysis and pharmacological evaluation of 7,7a,13,14-tetrahydro-6H-cyclobuta[b]pyrimido[1,2-a:3,4-a′]diindole analogues as melatonin receptor ligands

2007 ◽  
Vol 5 (13) ◽  
pp. 2129-2137 ◽  
Author(s):  
Mohamed I. Attia ◽  
Deniz Güclü ◽  
Barbara Hertlein ◽  
Justin Julius ◽  
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MT1-Selective Melatonin Receptor Ligands: Synthesis, Pharmacological Evaluation, and Molecular Dynamics Investigation ofN-{[(3-O-Substituted)anilino]alkyl}amides

ChemMedChem ◽  
2012 ◽  
Vol 7 (11) ◽  
pp. 1954-1964 ◽  
Author(s):  
Silvia Rivara ◽  
Daniele Pala ◽  
Alessio Lodola ◽  
Marco Mor ◽  
Valeria Lucini ◽  
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scholarly journals The pharmacological evaluation of novel and high‐affinity melatonin receptor ligands

2008 ◽  
Vol 22 (S1) ◽  
Author(s):  
Paula Ann Witt‐Enderby ◽  
Justin Julius ◽  
Mohamed I Attia ◽  
Darius P Zlotos
Keyword(s):  
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Synthesis and pharmacological evaluation of 6a,7-dihydro-6H,13H-pyrazino[1,2-a;4,5-a′]diindole analogs as melatonin receptor ligands

Tetrahedron ◽  
2007 ◽  
Vol 63 (3) ◽  
pp. 754-760 ◽  
Author(s):  
Mohamed I. Attia ◽  
Justin Julius ◽  
Paula A. Witt-Enderby ◽  
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Synthesis of 2(3H)-Benzoxazolone Derivatives as Potential Melatonin Receptor Ligands

Heterocycles ◽  
2003 ◽  
Vol 60 (12) ◽  
pp. 2621 ◽  
Author(s):  
Pascal Carato ◽  
Christophe Mésangeau ◽  
Jacques H. Poupaert ◽  
Saïd Yous
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Receptor Ligands

Conformational analysis and molecular modeling of 1-phenyl-, 4-phenyl-, and 1-benzyl-1,2,3,4-tetrahydroisoquinolines as D1 dopamine receptor ligands

1989 ◽  
Vol 32 (9) ◽  
pp. 2050-2058 ◽  
Author(s):  
Paul S. Charifson ◽  
J. Phillip Bowen ◽  
Steven D. Wyrick ◽  
Andrew J. Hoffman ◽  
Michael Cory ◽  
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Highly Potent and Selective MT2 Melatonin Receptor Full Agonists from Conformational Analysis of 1-Benzyl-2-acylaminomethyl-tetrahydroquinolines

2015 ◽  
Vol 58 (18) ◽  
pp. 7512-7525 ◽  
Author(s):  
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Annalida Bedini ◽  
Simone Lucarini ◽  
Michele Mari ◽  
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Melatonin Receptor

Conformational Analysis of Bivalent Estrogen Receptor Ligands: From Intramolecular to Intermolecular Binding

ChemBioChem ◽  
2011 ◽  
Vol 12 (17) ◽  
pp. 2587-2598 ◽  
Author(s):  
Min Shan ◽  
Alexander Bujotzek ◽  
Frank Abendroth ◽  
Anja Wellner ◽  
Ronald Gust ◽  
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Melatonin Receptor Ligands:  Synthesis of New Melatonin Derivatives and Comprehensive Comparative Molecular Field Analysis (CoMFA) Study

1998 ◽  
Vol 41 (20) ◽  
pp. 3831-3844 ◽  
Author(s):  
Marco Mor ◽  
Silvia Rivara ◽  
Claudia Silva ◽  
Fabrizio Bordi ◽  
Pier Vincenzo Plazzi ◽  
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Keyword(s):  
Field Analysis ◽  
Molecular Field ◽  
Comparative Molecular Field Analysis ◽  
Melatonin Receptor ◽  
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scholarly journals Virtual discovery of melatonin receptor ligands to modulate circadian rhythms

Nature ◽  
2020 ◽  
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pp. 609-614 ◽  
Author(s):  
Reed M. Stein ◽  
Hye Jin Kang ◽  
John D. McCorvy ◽  
Grant C. Glatfelter ◽  
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Benzodiazepine Receptor Ligands. 4. Synthesis and Pharmacological Evaluation of 3-Heteroaryl-8-chloropyrazolo[5,1-c][1,2,4]benzotriazine 5-Oxides

1999 ◽  
Vol 42 (12) ◽  
pp. 2218-2226 ◽  
Author(s):  
Annarella Costanzo ◽  
Gabriella Guerrini ◽  
Giovanna Ciciani ◽  
Fabrizio Bruni ◽  
Silvia Selleri ◽  
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