DU127090: A novel partial dopamine agonist with antipsychotic activity: Pilot study of dopamine D2 receptor occupancy after multiple oral administration of DU127090 to healthy male volunteers, using11C-raclopride by means of positron emission tomography

Pilot Study ◽

Dopamine D2 Receptor ◽

D2 Receptor ◽

Receptor Occupancy ◽

Emission Tomography ◽

Healthy Male ◽

Positron Emission ◽

Antipsychotic Activity ◽

Partial Dopamine Agonist

DU 127090: a highly potent, atypical dopamine receptor ligand — pilot study of dopamine D2 receptor occupancy after multiple oral administration of DU 127090 to healthy male volunteers, using 11C-raclopride by means of positron emission tomography

European Neuropsychopharmacology ◽

10.1016/s0924-977x(00)80320-x ◽

2000 ◽

Vol 10 ◽

pp. 294 ◽

Cited By ~ 5

Author(s):

M.H. De Vries ◽

J. Udo de Haes ◽

S.K. Long ◽

A. Grahnén ◽

L. Nyman ◽

...

Keyword(s):

Pilot Study ◽

Oral Administration ◽

Dopamine D2 Receptor ◽

D2 Receptor ◽

Receptor Occupancy ◽

Emission Tomography ◽

Healthy Male ◽

Receptor Ligand ◽

Determination of dopamine D2 receptor occupancy by lurasidone using positron emission tomography in healthy male subjects

Psychopharmacology ◽

10.1007/s00213-013-3103-z ◽

2013 ◽

Vol 229 (2) ◽

pp. 245-252 ◽

Cited By ~ 17

Author(s):

Dean F. Wong ◽

Hiroto Kuwabara ◽

James Robert Brašić ◽

Thomas Stock ◽

Atul Maini ◽

...

Keyword(s):

Dopamine D2 Receptor ◽

D2 Receptor ◽

Receptor Occupancy ◽

Emission Tomography ◽

Healthy Male ◽

Positron Emission ◽

Male Subjects

No regional difference in dopamine D2 receptor occupancy by the second-generation antipsychotic drug risperidone in humans: a positron emission tomography study

The International Journal of Neuropsychopharmacology ◽

10.1017/s1461145708009577 ◽

2008 ◽

Vol 12 (05) ◽

pp. 667 ◽

Cited By ~ 18

Author(s):

Hiroshi Ito ◽

Ryosuke Arakawa ◽

Hidehiko Takahashi ◽

Harumasa Takano ◽

Masaki Okumura ◽

...

Keyword(s):

Antipsychotic Drug ◽

Regional Difference ◽

Second Generation ◽

Dopamine D2 Receptor ◽

D2 Receptor ◽

Receptor Occupancy ◽

Emission Tomography ◽

Positron Emission ◽

Second Generation Antipsychotic

A Positron Emission Tomography Study of Quetiapine in Schizophrenia: A Preliminary Finding of an Antipsychotic Effect With Only Transiently High Dopamine D2 Receptor Occupancy

Archives of General Psychiatry ◽

10.1001/archpsyc.57.6.553 ◽

2000 ◽

Vol 57 (6) ◽

pp. 553-559 ◽

Cited By ~ 253

Author(s):

S. Kapur

Keyword(s):

Dopamine D2 Receptor ◽

D2 Receptor ◽

Preliminary Finding ◽

Receptor Occupancy ◽

Emission Tomography ◽

Antipsychotic Effect ◽

Dopamine D2 receptor occupancy by perospirone: a positron emission tomography study in patients with schizophrenia and healthy subjects

Psychopharmacology ◽

10.1007/s00213-010-1783-1 ◽

2010 ◽

Vol 209 (4) ◽

pp. 285-290 ◽

Cited By ~ 7

Author(s):

Ryosuke Arakawa ◽

Hiroshi Ito ◽

Akihiro Takano ◽

Masaki Okumura ◽

Hidehiko Takahashi ◽

...

Keyword(s):

Healthy Subjects ◽

Dopamine D2 Receptor ◽

D2 Receptor ◽

Receptor Occupancy ◽

Emission Tomography ◽

Dopamine D2 ◽

Savoxepine: striatal dopamine-D2 receptor occupancy in human volunteers measured using positron emission tomography (PET)

European Journal of Clinical Pharmacology ◽

10.1007/bf00315470 ◽

1993 ◽

Vol 44 (2) ◽

pp. 135-140 ◽

Cited By ~ 7

Author(s):

K. L. Leenders ◽

A. Antonini ◽

R. Thomann ◽

J. T. Locher ◽

L. Ma�tre ◽

...

Keyword(s):

Dopamine D2 Receptor ◽

D2 Receptor ◽

Receptor Occupancy ◽

Striatal Dopamine ◽

Emission Tomography ◽

Dopamine D2 ◽

Positron Emission ◽

Human Volunteers

Estimation of Baseline Dopamine D2 Receptor Occupancy in Striatum and Extrastriatal Regions in Humans with Positron Emission Tomography with [18F] Fallypride

Biological Psychiatry ◽

10.1016/j.biopsych.2007.03.022 ◽

2008 ◽

Vol 63 (2) ◽

pp. 241-244 ◽

Cited By ~ 39

Author(s):

Patrizia Riccardi ◽

Ron Baldwin ◽

Ronald Salomon ◽

Sharlet Anderson ◽

Mohammad S. Ansari ◽

...

Keyword(s):

Dopamine D2 Receptor ◽

D2 Receptor ◽

Receptor Occupancy ◽

Emission Tomography ◽

Dopamine D2 ◽

Predicting the dopamine D2 receptor occupancy of ropinirole in rats using positron emission tomography and pharmacokinetic–pharmacodynamic modeling

Xenobiotica ◽

10.1080/00498254.2018.1428383 ◽

2018 ◽

Vol 49 (2) ◽

pp. 143-151 ◽

Cited By ~ 1

Author(s):

Chenrong Huang ◽

Ziteng Wang ◽

Linsheng Liu ◽

Xiaoxue Liu ◽

Ji Dong ◽

...

Keyword(s):

Dopamine D2 Receptor ◽

D2 Receptor ◽

Receptor Occupancy ◽

Emission Tomography ◽

Pharmacodynamic Modeling ◽

Dopamine D2 ◽

Striatal and extrastriatal dopamine D2 receptor occupancy by the partial agonist antipsychotic drug aripiprazole in the human brain: a positron emission tomography study with [11C]raclopride and [11C]FLB457

Psychopharmacology ◽

10.1007/s00213-011-2633-5 ◽

2012 ◽

Vol 222 (1) ◽

pp. 165-172 ◽

Cited By ~ 10

Author(s):

Keisuke Takahata ◽

Hiroshi Ito ◽

Harumasa Takano ◽

Ryosuke Arakawa ◽

Hironobu Fujiwara ◽

...

Keyword(s):

Human Brain ◽

Antipsychotic Drug ◽

Dopamine D2 Receptor ◽

Partial Agonist ◽

D2 Receptor ◽

Receptor Occupancy ◽

Emission Tomography ◽

Dopamine D2 receptor occupancy of lumateperone (ITI-007): a Positron Emission Tomography Study in patients with schizophrenia

Neuropsychopharmacology ◽

10.1038/s41386-018-0251-1 ◽

2018 ◽

Vol 44 (3) ◽

pp. 598-605 ◽

Cited By ~ 8

Author(s):

Kimberly E. Vanover ◽

Robert E. Davis ◽

Yun Zhou ◽

Weiguo Ye ◽

James R. Brašić ◽

...

Keyword(s):

Dopamine D2 Receptor ◽

D2 Receptor ◽

Receptor Occupancy ◽

Emission Tomography ◽

Dopamine D2 ◽