Synthesis, structure and biological properties of Z-17α-(2-iodovinyl)-11β-chloromethyl estradiol-17β (Z-CMIV), a high affinity ligand for the characterization of estrogen receptor-positive tumors

Jacques Quivy; Guy Leclercq; Marcel Deblaton; Pierre Henrot; Nicolas Velings; Bernadette Norberg; Guy Evrard; Marc Zeicher

doi:10.1016/s0960-0760(96)00007-6

Synthesis, structure and biological properties of Z-17α-(2-iodovinyl)-11β-chloromethyl estradiol-17β (Z-CMIV), a high affinity ligand for the characterization of estrogen receptor-positive tumors

The Journal of Steroid Biochemistry and Molecular Biology ◽

10.1016/s0960-0760(96)00007-6 ◽

1996 ◽

Vol 59 (1) ◽

pp. 103-117 ◽

Cited By ~ 11

Author(s):

Jacques Quivy ◽

Guy Leclercq ◽

Marcel Deblaton ◽

Pierre Henrot ◽

Nicolas Velings ◽

...

Keyword(s):

Estrogen Receptor ◽

Biological Properties ◽

High Affinity ◽

Affinity Ligand ◽

Estrogen Receptor Positive ◽

Estradiol 17Β ◽

High Affinity Ligand

Download Full-text

Preparation of a photoreactive analog of parathyroid hormone [Nle8,Lys(N-ϵ-4-azido-2-nitrophenyl)13, Nle18,Tyr34]bovine parathyroid hormone-(1–34)NH2, a selective, high-affinity ligand for characterization of parathyroid hormone receptors

Analytical Biochemistry ◽

10.1016/0003-2697(89)90126-7 ◽

1989 ◽

Vol 179 (2) ◽

pp. 268-273 ◽

Cited By ~ 12

Author(s):

Chohei Shigeno ◽

Yuji Hiraki ◽

Henry T. Keutmann ◽

Andrew M. Stern ◽

John T. Potts ◽

...

Keyword(s):

Parathyroid Hormone ◽

Hormone Receptors ◽

High Affinity ◽

Affinity Ligand ◽

High Affinity Ligand ◽

Bovine Parathyroid Hormone

Download Full-text

Characterization of β-adrenergic receptor subtypes in androgen-induced mouse kidney hypertrophy using a new high-affinity ligand, [125I]iodocyanopindolol

Biochimica et Biophysica Acta (BBA) - General Subjects ◽

10.1016/0304-4165(83)90337-9 ◽

1983 ◽

Vol 756 (3) ◽

pp. 286-296 ◽

Cited By ~ 12

Author(s):

S.L. Petrovic ◽

G. Engel ◽

R.P. Haugland ◽

R.M. Dowben

Keyword(s):

Adrenergic Receptor ◽

Mouse Kidney ◽

Receptor Subtypes ◽

High Affinity ◽

Affinity Ligand ◽

Kidney Hypertrophy ◽

High Affinity Ligand

Download Full-text

Structural characterization of a peptoid-inspired conformationally constrained oligomer (PICCO) bound to streptavidin

Chemical Communications ◽

10.1039/d0cc02588g ◽

2020 ◽

Vol 56 (72) ◽

pp. 10560-10563

Author(s):

Patrick McEnaney ◽

Madeline Balzarini ◽

Hajeung Park ◽

Thomas Kodadek

Keyword(s):

Structural Characterization ◽

Conformationally Constrained ◽

High Affinity ◽

Affinity Ligand ◽

High Affinity Ligand

A screen of a DNA-encoded library of PICCOs was screened against streptavidin (SA) resulting in the isolation of a high affinity ligand.

Download Full-text

Two high-affinity ligand binding states of uterine estrogen receptor distinguished by modulation of hydrophobic environment

Biochemistry ◽

10.1021/bi00377a010 ◽

1987 ◽

Vol 26 (3) ◽

pp. 722-727 ◽

Cited By ~ 8

Author(s):

T. William Hutchens ◽

Chee Ming Li ◽

Nezaam M. Zamah ◽

Paige K. Besch

Keyword(s):

Estrogen Receptor ◽

Ligand Binding ◽

High Affinity ◽

Affinity Ligand ◽

High Affinity Ligand

Download Full-text

In vitro characterization of 6-[18F]fluoro-A-85380, a high-affinity ligand for α4β2* nicotinic acetylcholine receptors

Synapse ◽

10.1002/syn.20096 ◽

2004 ◽

Vol 55 (2) ◽

pp. 89-97 ◽

Cited By ~ 15

Author(s):

Daniela Gündisch ◽

Andrei O. Koren ◽

Andrew G. Horti ◽

Olga A. Pavlova ◽

Alane S. Kimes ◽

...

Keyword(s):

Nicotinic Acetylcholine Receptors ◽

Acetylcholine Receptors ◽

Nicotinic Acetylcholine ◽

High Affinity ◽

Affinity Ligand ◽

In Vitro Characterization ◽

High Affinity Ligand

Download Full-text

Characterization of β-adrenergic receptors in rat brain and pituitary using a new high-affinity ligand, [125I]iodocyanopindolol

Brain Research ◽

10.1016/0006-8993(83)90628-5 ◽

1983 ◽

Vol 261 (2) ◽

pp. 249-259 ◽

Cited By ~ 47

Author(s):

S.L. Petrovic ◽

J.K. McDonald ◽

G.D. Snyder ◽

S.M. McCann

Keyword(s):

Rat Brain ◽

Adrenergic Receptors ◽

High Affinity ◽

Affinity Ligand ◽

Β Adrenergic Receptors ◽

High Affinity Ligand

Download Full-text

The molecular structure of 16α-iodo-17β-estradiol, a high affinity ligand for the estrogen receptor

Journal of Steroid Biochemistry ◽

10.1016/0022-4731(86)90002-6 ◽

1986 ◽

Vol 25 (5) ◽

pp. 615-618 ◽

Cited By ~ 9

Author(s):

Richard B. Hochberg ◽

Jan E. Zielinski ◽

William L. Duax ◽

Phyllis Strong

Keyword(s):

Molecular Structure ◽

Estrogen Receptor ◽

High Affinity ◽

Affinity Ligand ◽

17Β Estradiol ◽

High Affinity Ligand

Download Full-text

Faculty Opinions recommendation of Vascular development in the retina and inner ear: control by Norrin and Frizzled-4, a high-affinity ligand-receptor pair.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.1018184.207692 ◽

2004 ◽

Author(s):

Marek Mlodzik

Keyword(s):

Inner Ear ◽

Vascular Development ◽

High Affinity ◽

Affinity Ligand ◽

High Affinity Ligand

Download Full-text

Faculty Opinions recommendation of Cyclic GMP-AMP containing mixed phosphodiester linkages is an endogenous high-affinity ligand for STING.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.718020257.793478725 ◽

2013 ◽

Author(s):

Shigekazu Nagata

Keyword(s):

Cyclic Gmp ◽

High Affinity ◽

Affinity Ligand ◽

High Affinity Ligand

Download Full-text

Multiple domains of the N-formyl peptide receptor are required for high-affinity ligand binding. Construction and analysis of chimeric N-formyl peptide receptors.

Journal of Biological Chemistry ◽

10.1016/s0021-9258(17)46825-6 ◽

1993 ◽

Vol 268 (24) ◽

pp. 18167-18175 ◽

Cited By ~ 3

Author(s):

O. Quehenberger ◽

E.R. Prossnitz ◽

S.L. Cavanagh ◽

C.G. Cochrane ◽

R.D. Ye

Keyword(s):

Ligand Binding ◽

Formyl Peptide Receptor ◽

Peptide Receptors ◽

Formyl Peptide Receptors ◽

Peptide Receptor ◽

High Affinity ◽

Affinity Ligand ◽

Formyl Peptide ◽

Multiple Domains ◽

High Affinity Ligand

Download Full-text