The 1.1 Å Crystal Structure of Human TGF-β Type II Receptor Ligand Binding Domain

Structure ◽

10.1016/s0969-2126(02)00780-3 ◽

2002 ◽

Vol 10 (7) ◽

pp. 913-919 ◽

Author(s):

Christian C Boesen ◽

Sergei Radaev ◽

Shawn A Motyka ◽

Apisit Patamawenu ◽

Peter D Sun

Keyword(s):

Crystal Structure ◽

Ligand Binding ◽

Binding Domain ◽

Ligand Binding Domain ◽

Type Ii ◽

Receptor Ligand

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Identification of novel α7 nicotinic receptor ligands by in silico screening against the crystal structure of a chimeric α7 receptor ligand binding domain

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2012.06.054 ◽

2012 ◽

Vol 20 (19) ◽

pp. 5992-6002 ◽

Author(s):

Atilla Akdemir ◽

Ewald Edink ◽

Andrew J. Thompson ◽

Sarah C.R. Lummis ◽

Albert J. Kooistra ◽

...

Keyword(s):

Crystal Structure ◽

Ligand Binding ◽

In Silico ◽

Nicotinic Receptor ◽

Binding Domain ◽

Ligand Binding Domain ◽

Receptor Ligands ◽

In Silico Screening ◽

Receptor Ligand

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Solution Structure of the Chick TGFβ Type II Receptor Ligand-binding Domain

Journal of Molecular Biology ◽

10.1016/s0022-2836(03)00023-8 ◽

2003 ◽

Vol 326 (4) ◽

pp. 989-997 ◽

Author(s):

Michael S. Marlow ◽

Christopher B. Brown ◽

Joey V. Barnett ◽

Andrzej M. Krezel

Keyword(s):

Ligand Binding ◽

Solution Structure ◽

Binding Domain ◽

Ligand Binding Domain ◽

Type Ii ◽

Receptor Ligand

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Synthesis and Crystal Structure of a Phosphorylated Estrogen Receptor Ligand Binding Domain

ChemBioChem ◽

10.1002/cbic.201000532 ◽

2010 ◽

Vol 11 (16) ◽

pp. 2251-2254 ◽

Author(s):

Sabine Möcklinghoff ◽

Rolf Rose ◽

Maëlle Carraz ◽

Arie Visser ◽

Christian Ottmann ◽

...

Keyword(s):

Crystal Structure ◽

Estrogen Receptor ◽

Ligand Binding ◽

Binding Domain ◽

Ligand Binding Domain ◽

Receptor Ligand ◽

Synthesis And Crystal Structure ◽

Estrogen Receptor Ligand

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Crystal Structure of the Glucocorticoid Receptor Ligand Binding Domain Reveals a Novel Mode of Receptor Dimerization and Coactivator Recognition

Cell ◽

10.1016/s0092-8674(02)00817-6 ◽

2002 ◽

Vol 110 (1) ◽

pp. 93-105 ◽

Author(s):

Randy K. Bledsoe ◽

Valerie G. Montana ◽

Thomas B. Stanley ◽

Chris J. Delves ◽

Christopher J. Apolito ◽

...

Keyword(s):

Crystal Structure ◽

Glucocorticoid Receptor ◽

Ligand Binding ◽

Binding Domain ◽

Ligand Binding Domain ◽

Receptor Ligand ◽

Receptor Dimerization

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X-ray Crystal Structure of the Novel Enhanced-Affinity Glucocorticoid Agonist Fluticasone Furoate in the Glucocorticoid Receptor−Ligand Binding Domain⊥

Journal of Medicinal Chemistry ◽

10.1021/jm800279t ◽

2008 ◽

Vol 51 (12) ◽

pp. 3349-3352 ◽

Author(s):

Keith Biggadike ◽

Randy K. Bledsoe ◽

Anne M. Hassell ◽

Barrie E. Kirk ◽

Iain M. McLay ◽

...

Keyword(s):

Crystal Structure ◽

Glucocorticoid Receptor ◽

Ligand Binding ◽

Binding Domain ◽

Ligand Binding Domain ◽

The Novel ◽

Fluticasone Furoate ◽

Receptor Ligand ◽

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Faculty Opinions recommendation of Crystal structure of the glucocorticoid receptor ligand binding domain reveals a novel mode of receptor dimerization and coactivator recognition.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.1008747.193353 ◽

2003 ◽

Author(s):

Fraydoon Rastinejad

Keyword(s):

Crystal Structure ◽

Glucocorticoid Receptor ◽

Ligand Binding ◽

Binding Domain ◽

Ligand Binding Domain ◽

Receptor Ligand ◽

Receptor Dimerization

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Vitamin D Analogues with a p-Hydroxyphenyl Group at the C25 Position: Crystal Structure of Vitamin D Receptor Ligand-Binding Domain Complexed with the Ligand Explains the Mechanism Underlying Full Antagonistic Action

Journal of Medicinal Chemistry ◽

10.1021/acs.jmedchem.7b00819 ◽

2017 ◽

Vol 60 (20) ◽

pp. 8394-8406 ◽

Author(s):

Akira Kato ◽

Makiko Yamao ◽

Yuta Hashihara ◽

Hiroaki Ishida ◽

Toshimasa Itoh ◽

...

Keyword(s):

Crystal Structure ◽

Vitamin D ◽

Ligand Binding ◽

Vitamin D Receptor ◽

Binding Domain ◽

Ligand Binding Domain ◽

Antagonistic Action ◽

Receptor Ligand ◽

Vitamin D Analogues

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Crystal structure of the mineralocorticoid receptor ligand‐binding domain in complex with a potent and selective nonsteroidal blocker, esaxerenone (CS‐3150)

FEBS Letters ◽

10.1002/1873-3468.13746 ◽

2020 ◽

Vol 594 (10) ◽

pp. 1615-1623 ◽

Author(s):

Mizuki Takahashi ◽

Osamu Ubukata ◽

Tsuyoshi Homma ◽

Yusuke Asoh ◽

Masatoshi Honzumi ◽

...

Keyword(s):

Crystal Structure ◽

Ligand Binding ◽

Mineralocorticoid Receptor ◽

Binding Domain ◽

Ligand Binding Domain ◽

Receptor Ligand

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Faculty Opinions recommendation of Crystal structure of the glucocorticoid receptor ligand binding domain reveals a novel mode of receptor dimerization and coactivator recognition.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.1008747.110457 ◽

2002 ◽

Author(s):

David Matthews

Keyword(s):

Crystal Structure ◽

Glucocorticoid Receptor ◽

Ligand Binding ◽

Binding Domain ◽

Ligand Binding Domain ◽

Receptor Ligand ◽

Receptor Dimerization

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Faculty Opinions recommendation of X-ray crystal structure of the novel enhanced-affinity glucocorticoid agonist fluticasone furoate in the glucocorticoid receptor-ligand binding domain.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.1111151.572750 ◽

2008 ◽

Author(s):

Robert Fecik

Keyword(s):

Crystal Structure ◽

Glucocorticoid Receptor ◽

Ligand Binding ◽

Binding Domain ◽

Ligand Binding Domain ◽

The Novel ◽

Fluticasone Furoate ◽

Receptor Ligand ◽

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