X-ray Crystal Structure of the Novel Enhanced-Affinity Glucocorticoid Agonist Fluticasone Furoate in the Glucocorticoid Receptor−Ligand Binding Domain⊥

2008 ◽  
Vol 51 (12) ◽  
pp. 3349-3352 ◽  
Author(s):  
Keith Biggadike ◽  
Randy K. Bledsoe ◽  
Anne M. Hassell ◽  
Barrie E. Kirk ◽  
Iain M. McLay ◽  
...  
Keyword(s):  
Crystal Structure ◽  
Glucocorticoid Receptor ◽  
Ligand Binding ◽  
Binding Domain ◽  
Ligand Binding Domain ◽  
The Novel ◽  
Fluticasone Furoate ◽  
Receptor Ligand ◽  
X Ray

scholarly journals Crystal Structure of the Glucocorticoid Receptor Ligand Binding Domain Reveals a Novel Mode of Receptor Dimerization and Coactivator Recognition

Cell ◽  
2002 ◽  
Vol 110 (1) ◽  
pp. 93-105 ◽  
Author(s):  
Randy K. Bledsoe ◽  
Valerie G. Montana ◽  
Thomas B. Stanley ◽  
Chris J. Delves ◽  
Christopher J. Apolito ◽  
...  
Keyword(s):  
Crystal Structure ◽  
Glucocorticoid Receptor ◽  
Ligand Binding ◽  
Binding Domain ◽  
Ligand Binding Domain ◽  
Receptor Ligand ◽  
Receptor Dimerization

scholarly journals The antagonistic crystal structure of the glucocorticoid receptor, ligand-binding domain

2002 ◽  
Vol 58 (s1) ◽  
pp. c201-c201
Author(s):  
B. Kauppi ◽  
C. Jakob ◽  
M. Farnegardh ◽  
H. Ahola ◽  
M. Alarcon ◽  
...  
Keyword(s):  
Crystal Structure ◽  
Glucocorticoid Receptor ◽  
Ligand Binding ◽  
Binding Domain ◽  
Ligand Binding Domain ◽  
Receptor Ligand

scholarly journals X-ray Structures of Progesterone Receptor Ligand Binding Domain in Its Agonist State Reveal Differing Mechanisms for Mixed Profiles of 11β-Substituted Steroids

2012 ◽  
Vol 287 (24) ◽  
pp. 20333-20343 ◽  
Author(s):  
Scott J. Lusher ◽  
Hans C. A. Raaijmakers ◽  
Diep Vu-Pham ◽  
Bert Kazemier ◽  
Rolien Bosch ◽  
...  
Keyword(s):  
Progesterone Receptor ◽  
Ligand Binding ◽  
Binding Domain ◽  
Ligand Binding Domain ◽  
Receptor Ligand ◽  
X Ray
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