2-Phenylcyclopropylmethylamine Derivatives as Dopamine D2 Receptor Partial Agonists: Design, Synthesis, and Biological Evaluation

2021 ◽  
Author(s):  
Wenzhong Yan ◽  
Luyu Fan ◽  
Jing Yu ◽  
Ruiquan Liu ◽  
Huan Wang ◽  
...  
Keyword(s):  
Dopamine D2 Receptor ◽  
D2 Receptor ◽  
Biological Evaluation ◽  
Design Synthesis ◽  
Partial Agonists ◽  
Dopamine D2 ◽  
Synthesis And Biological Evaluation

Design, synthesis and pharmacological profile of novel dopamine D2 receptor ligands

2003 ◽  
Vol 11 (22) ◽  
pp. 4807-4813 ◽  
Author(s):  
Ricardo Menegatti ◽  
Anna C Cunha ◽  
Vı́tor F Ferreira ◽  
Edna F.R Perreira ◽  
Ahmed El-Nabawi ◽  
...  
Keyword(s):  
Dopamine D2 Receptor ◽  
D2 Receptor ◽  
Receptor Ligands ◽  
Pharmacological Profile ◽  
Design Synthesis ◽  
Dopamine D2

scholarly journals Active-State Model of a Dopamine D2 Receptor - Gαi Complex Stabilized by Aripiprazole-Type Partial Agonists

PLoS ONE ◽  
2014 ◽  
Vol 9 (6) ◽  
pp. e100069 ◽  
Author(s):  
Ralf C. Kling ◽  
Nuska Tschammer ◽  
Harald Lanig ◽  
Timothy Clark ◽  
Peter Gmeiner
Keyword(s):  
Dopamine D2 Receptor ◽  
D2 Receptor ◽  
Active State ◽  
State Model ◽  
Partial Agonists ◽  
Dopamine D2

Preparation and preliminary biological evaluation of [18F]NCQ-115: a new selective reversible dopamine D2 receptor ligand

1993 ◽  
Vol 20 (4) ◽  
pp. 549-555 ◽  
Author(s):  
A. Najafi ◽  
A. Peterson ◽  
M. Buchsbaum ◽  
S. O'Dell ◽  
F. Weihmuller
Keyword(s):  
Dopamine D2 Receptor ◽  
D2 Receptor ◽  
Biological Evaluation ◽  
Receptor Ligand ◽  
Dopamine D2

Aripiprazole and its human metabolite are partial agonists at the human dopamine D2 receptor, but the rodent metabolite displays antagonist properties

2006 ◽  
Vol 546 (1-3) ◽  
pp. 88-94 ◽  
Author(s):  
Martyn D. Wood ◽  
Claire Scott ◽  
Kirsten Clarke ◽  
Julie Westaway ◽  
Ceri H. Davies ◽  
...  
Keyword(s):  
Dopamine D2 Receptor ◽  
D2 Receptor ◽  
Human Metabolite ◽  
Partial Agonists ◽  
Dopamine D2

Serotonergic agonists behave as partial agonists at the dopamine D2 receptor

Neuroreport ◽  
1999 ◽  
Vol 10 (3) ◽  
pp. 493-495 ◽  
Author(s):  
Ago Rinken ◽  
Sergi Ferré ◽  
Anton Terasmaa ◽  
Christer Owman ◽  
Kjell Fuxe
Keyword(s):  
Dopamine D2 Receptor ◽  
D2 Receptor ◽  
Partial Agonists ◽  
Dopamine D2
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