In vitro functional characteristics of dopamine D2 receptor partial agonists in second and third messenger-based assays of cloned human dopamine D2Long receptor signalling

2006 ◽  
Vol 21 (6) ◽  
pp. 620-627 ◽  
Author(s):  
Shaun Jordan ◽  
Karen Regardie ◽  
Janelle L. Johnson ◽  
Ruoyan Chen ◽  
Junichi Kambayashi ◽  
...  
Keyword(s):  
Dopamine D2 Receptor ◽  
D2 Receptor ◽  
Functional Characteristics ◽  
Partial Agonists ◽  
Receptor Signalling ◽  
Dopamine D2

ACTH/MSH-like peptides inhibit the binding of dopaminergic ligands to the dopamine D2 receptor in vitro

1991 ◽  
Vol 207 (1) ◽  
pp. 43-50 ◽  
Author(s):  
Wouter J. Florijn ◽  
Thijs De Boer ◽  
Jeroen A.D.M. Tonnaer ◽  
Jan W. Van Nispen ◽  
Dirk H.G. Versteeg
Keyword(s):  
Dopamine D2 Receptor ◽  
D2 Receptor ◽  
Dopamine D2

Prediction of CNS occupancy of dopamine D2 receptor based on systemic exposure and in vitro experiments

2016 ◽  
Vol 31 (6) ◽  
pp. 395-404 ◽  
Author(s):  
Kayoko Kanamitsu ◽  
Ryosuke Arakawa ◽  
Yuichi Sugiyama ◽  
Tetsuya Suhara ◽  
Hiroyuki Kusuhara
Keyword(s):  
Dopamine D2 Receptor ◽  
D2 Receptor ◽  
Systemic Exposure ◽  
In Vitro Experiments ◽  
Dopamine D2

scholarly journals Active-State Model of a Dopamine D2 Receptor - Gαi Complex Stabilized by Aripiprazole-Type Partial Agonists

PLoS ONE ◽  
2014 ◽  
Vol 9 (6) ◽  
pp. e100069 ◽  
Author(s):  
Ralf C. Kling ◽  
Nuska Tschammer ◽  
Harald Lanig ◽  
Timothy Clark ◽  
Peter Gmeiner
Keyword(s):  
Dopamine D2 Receptor ◽  
D2 Receptor ◽  
Active State ◽  
State Model ◽  
Partial Agonists ◽  
Dopamine D2

In vitro and in vivo evaluation of the binding of the dopamine D2 receptor agonist11C-(R,S)-5-hydroxy-2-(di-n-propylamino)tetralin in rodents and nonhuman primate

Synapse ◽  
2000 ◽  
Vol 37 (1) ◽  
pp. 64-70 ◽  
Author(s):  
Jogeshwar Mukherjee ◽  
Tanjore K. Narayanan ◽  
Bradley T. Christian ◽  
Bingzhi Shi ◽  
Kelly A. Dunigan ◽  
...  
Keyword(s):  
Nonhuman Primate ◽  
Dopamine D2 Receptor ◽  
D2 Receptor ◽  
In Vivo Evaluation ◽  
Dopamine D2

Aripiprazole and its human metabolite are partial agonists at the human dopamine D2 receptor, but the rodent metabolite displays antagonist properties

2006 ◽  
Vol 546 (1-3) ◽  
pp. 88-94 ◽  
Author(s):  
Martyn D. Wood ◽  
Claire Scott ◽  
Kirsten Clarke ◽  
Julie Westaway ◽  
Ceri H. Davies ◽  
...  
Keyword(s):  
Dopamine D2 Receptor ◽  
D2 Receptor ◽  
Human Metabolite ◽  
Partial Agonists ◽  
Dopamine D2
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