Synthesis and Biological Evaluation of 7,8,9,10-Tetrahydroimidazo[1,2-c]pyrido[3,4-e]pyrimdin-5(6H)-ones as Functionally Selective Ligands of the Benzodiazepine Receptor Site on the GABAAReceptor

2002 ◽  
Vol 45 (23) ◽  
pp. 5043-5051 ◽  
Author(s):  
Pamela A. Albaugh ◽  
Lu Marshall ◽  
James Gregory ◽  
Geoff White ◽  
Alan Hutchison ◽  
...  
Keyword(s):  
Receptor Site ◽  
Benzodiazepine Receptor ◽  
Biological Evaluation ◽  
Selective Ligands ◽  
Synthesis And Biological Evaluation

Synthesis and biological evaluation of novel cyclopropyl derivatives as subtype-selective ligands for estrogen receptor

2018 ◽  
Vol 70 (7) ◽  
pp. 910-918 ◽  
Author(s):  
Zunyuan Wang ◽  
Yewei Yang ◽  
Xiaoliang Zheng ◽  
Tao Zhang ◽  
Wenhai Huang ◽  
...  
Keyword(s):  
Estrogen Receptor ◽  
Biological Evaluation ◽  
Selective Ligands ◽  
Subtype Selective ◽  
Synthesis And Biological Evaluation

Novel N-Substituted Indol-3-ylglyoxylamides Probing the LDiand L1/L2Lipophilic Regions of the Benzodiazepine Receptor Site in Search for Subtype-Selective Ligands†

2007 ◽  
Vol 50 (7) ◽  
pp. 1627-1634 ◽  
Author(s):  
Giampaolo Primofiore ◽  
Sabrina Taliani ◽  
Federico Da Settimo ◽  
Anna Maria Marini ◽  
Concettina La Motta ◽  
...  
Keyword(s):  
Receptor Site ◽  
Benzodiazepine Receptor ◽  
Selective Ligands ◽  
Subtype Selective

New Fluorescent 2-Phenylindolglyoxylamide Derivatives as Probes Targeting the Peripheral-Type Benzodiazepine Receptor:  Design, Synthesis, and Biological Evaluation

2007 ◽  
Vol 50 (2) ◽  
pp. 404-407 ◽  
Author(s):  
Sabrina Taliani ◽  
Francesca Simorini ◽  
Valentina Sergianni ◽  
Concettina La Motta ◽  
Federico Da Settimo ◽  
...  
Keyword(s):  
Benzodiazepine Receptor ◽  
Biological Evaluation ◽  
Design Synthesis ◽  
Receptor Design ◽  
Peripheral Type ◽  
Synthesis And Biological Evaluation

A3 adenosine receptors: Synthesis and biological evaluation of new potent and selective ligands

2005 ◽  
Author(s):  
Rosaria Volpini ◽  
Catia Lambertucci ◽  
Sara Taffi ◽  
Sauro Vittori ◽  
Karl-Norbert Klotz ◽  
...  
Keyword(s):  
Adenosine Receptors ◽  
Biological Evaluation ◽  
Selective Ligands ◽  
Synthesis And Biological Evaluation
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