Benzodiazepine receptor ligands — Part II. Synthesis and biological evaluation of pyrazolo[5,1-c][1,2,4]benzotriazine 4-oxide

European Journal of Medicinal Chemistry ◽

10.1016/s0223-5234(98)80013-5 ◽

1998 ◽

Vol 33 (3) ◽

pp. 237-244 ◽

Author(s):

Annarella Costanzo ◽

Gabriella Guerrini ◽

Fabrizio Bruni ◽

Giovanna Ciciani ◽

Silvia Selleri ◽

...

Keyword(s):

Benzodiazepine Receptor ◽

Biological Evaluation ◽

Receptor Ligands ◽

Benzodiazepine Receptor Ligands ◽

Synthesis And Biological Evaluation

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ChemInform Abstract: Benzodiazepine Receptor Ligands. Part 2. Synthesis and Biological Evaluation of Pyrazolo[5,1-c][1,2,4]benzotriazine 4-Oxide.

10.1002/chin.199830184 ◽

2010 ◽

Vol 29 (30) ◽

pp. no-no

Author(s):

A. COSTANZO ◽

G. GUERRINI ◽

F. BRUNI ◽

G. CICIANI ◽

S. SELLERI ◽

...

Keyword(s):

Benzodiazepine Receptor ◽

Biological Evaluation ◽

Receptor Ligands ◽

Benzodiazepine Receptor Ligands ◽

Synthesis And Biological Evaluation

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High Affinity Central Benzodiazepine Receptor Ligands: Synthesis and Biological Evaluation of a Series of Phenyltriazolobenzotriazindione Derivatives

Journal of Medicinal Chemistry ◽

10.1021/jm0408722 ◽

2005 ◽

Vol 48 (8) ◽

pp. 2936-2943 ◽

Author(s):

Giampaolo Primofiore ◽

Federico Da Settimo ◽

Sabrina Taliani ◽

Silvia Salerno ◽

Ettore Novellino ◽

...

Keyword(s):

Benzodiazepine Receptor ◽

Biological Evaluation ◽

Receptor Ligands ◽

Benzodiazepine Receptor Ligands ◽

High Affinity ◽

Central Benzodiazepine Receptor ◽

Synthesis And Biological Evaluation

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Insight into 2-phenylpyrazolo[1,5-a]pyrimidin-3-yl acetamides as peripheral benzodiazepine receptor ligands: Synthesis, biological evaluation and 3D-QSAR investigation

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2005.05.015 ◽

2005 ◽

Vol 13 (16) ◽

pp. 4821-4834 ◽

Author(s):

Silvia Selleri ◽

Paola Gratteri ◽

Camilla Costagli ◽

Claudia Bonaccini ◽

Annarella Costanzo ◽

...

Keyword(s):

Benzodiazepine Receptor ◽

3D Qsar ◽

Biological Evaluation ◽

Peripheral Benzodiazepine Receptor ◽

Receptor Ligands ◽

Benzodiazepine Receptor Ligands ◽

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Peripheral benzodiazepine receptor ligands induce apoptosis and cell cycle arrest in human hepatocellular carcinoma cells and enhance chemosensitivity to paclitaxel, docetaxel, doxorubicin and the Bcl–2 inhibitor HA14–1

Zeitschrift für Gastroenterologie ◽

10.1055/s-2004-831695 ◽

2004 ◽

Vol 42 (08) ◽

Author(s):

A Sutter ◽

K Maaser ◽

P Grabowski ◽

M Höpfner ◽

A Krahn ◽

...

Keyword(s):

Hepatocellular Carcinoma ◽

Cell Cycle Arrest ◽

Benzodiazepine Receptor ◽

Carcinoma Cells ◽

Peripheral Benzodiazepine Receptor ◽

Receptor Ligands ◽

Benzodiazepine Receptor Ligands ◽

Cycle Arrest ◽

Human Hepatocellular Carcinoma Cells

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Benzodiazepine Receptor Ligands, Memory and Information Processing

10.1007/978-3-642-73288-1 ◽

1988 ◽

Keyword(s):

Information Processing ◽

Benzodiazepine Receptor ◽

Receptor Ligands ◽

Benzodiazepine Receptor Ligands

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Benzodiazepine receptor ligands and sexual behavior in the male rat: The role of GABAergic mechanisms

Pharmacology Biochemistry and Behavior ◽

10.1016/0091-3057(91)90242-t ◽

1991 ◽

Vol 38 (4) ◽

pp. 781-788 ◽

Author(s):

Anders Ågmo ◽

Hilda Fernández

Keyword(s):

Sexual Behavior ◽

Benzodiazepine Receptor ◽

Male Rat ◽

Receptor Ligands ◽

Benzodiazepine Receptor Ligands

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Design, synthesis and biological evaluation of piperazine analogues as CB1 cannabinoid receptor ligands

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2008.01.023 ◽

2008 ◽

Vol 16 (7) ◽

pp. 4035-4051 ◽

Author(s):

Kwang-Seop Song ◽

Sung-Han Lee ◽

Hyun Ji Chun ◽

Jong Yup Kim ◽

Myung Eun Jung ◽

...

Keyword(s):

Cannabinoid Receptor ◽

Biological Evaluation ◽

Receptor Ligands ◽

Design Synthesis ◽

Cb1 Cannabinoid Receptor ◽

Synthesis And Biological Evaluation

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Specific high-affinity binding of peripheral benzodiazepine receptor ligands to brain tumors in rat and man

Cancer ◽

10.1002/1097-0142(19900101)65:1<93::aid-cncr2820650120>3.0.co;2-1 ◽

1990 ◽

Vol 65 (1) ◽

pp. 93-97 ◽

Author(s):

Keith L. Black ◽

Kiyonobu Ikezaki ◽

Emily Santori ◽

Donald P. Becker ◽

Harry V. Vinters

Keyword(s):

Brain Tumors ◽

Benzodiazepine Receptor ◽

Affinity Binding ◽

Peripheral Benzodiazepine Receptor ◽

Receptor Ligands ◽

High Affinity Binding ◽

Benzodiazepine Receptor Ligands ◽

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Selective changes in the in vivo effects of benzodiazepine receptor ligands after chemical kindling with FG 7142

Neuropharmacology ◽

10.1016/0028-3908(87)90040-2 ◽

1987 ◽

Vol 26 (1) ◽

pp. 25-31 ◽

Author(s):

H.J. Little ◽

D.J. Nutt ◽

S.C. Taylor

Keyword(s):

Benzodiazepine Receptor ◽

Fg 7142 ◽

Receptor Ligands ◽

Benzodiazepine Receptor Ligands ◽

Chemical Kindling ◽

In Vivo Effects

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Design, synthesis and biological evaluation of bitopic arylpiperazine-hexahydro-pyrazinoquinolines as preferential dopamine D3 receptor ligands

Bioorganic Chemistry ◽

10.1016/j.bioorg.2017.12.026 ◽

2018 ◽

Vol 77 ◽

pp. 125-135

Author(s):

Benhua Zhou ◽

Min Ji ◽

Jin Cai

Keyword(s):

Biological Evaluation ◽

Dopamine D3 Receptor ◽

D3 Receptor ◽

Receptor Ligands ◽

Design Synthesis ◽

Dopamine D3 ◽

Synthesis And Biological Evaluation

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