Synthesis, in Vitro Activity, and Three-Dimensional Quantitative Structure−Activity Relationship of Novel Hydrazine Inhibitors of Human Vascular Adhesion Protein-1

Elisa M. Nurminen; Marjo Pihlavisto; László Lázár; Zsolt Szakonyi; Ulla Pentikäinen; Ferenc Fülöp; Olli T. Pentikäinen

doi:10.1021/jm100337z

Synthesis, in Vitro Activity, and Three-Dimensional Quantitative Structure−Activity Relationship of Novel Hydrazine Inhibitors of Human Vascular Adhesion Protein-1

Journal of Medicinal Chemistry ◽

10.1021/jm100337z ◽

2010 ◽

Vol 53 (17) ◽

pp. 6301-6315 ◽

Cited By ~ 22

Author(s):

Elisa M. Nurminen ◽

Marjo Pihlavisto ◽

László Lázár ◽

Zsolt Szakonyi ◽

Ulla Pentikäinen ◽

...

Keyword(s):

Three Dimensional ◽

Quantitative Structure Activity Relationship ◽

Quantitative Structure ◽

In Vitro Activity ◽

Adhesion Protein ◽

Structure Activity ◽

Vascular Adhesion ◽

Relationship Of ◽

Vascular Adhesion Protein 1

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Cytotoxic Activity and Three-Dimensional Quantitative Structure Activity Relationship of 2-Aryl-1,8-naphthyridin-4-ones

Korean Journal of Physiology and Pharmacology ◽

10.4196/kjpp.2009.13.6.511 ◽

2009 ◽

Vol 13 (6) ◽

pp. 511 ◽

Cited By ~ 2

Author(s):

Yong Jin Kim ◽

Eun Ae Kim ◽

Mi Lyang Chung ◽

Chaeuk Im

Keyword(s):

Cytotoxic Activity ◽

Three Dimensional ◽

Quantitative Structure Activity Relationship ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Quantitative Structure ◽

Structure Activity ◽

Relationship Of

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Three-dimensional quantitative structure activity relationship (3D-QSAR) analysis for in vitro toxicity of chlorophenols to HepG2 cells

Chemosphere ◽

10.1016/j.chemosphere.2005.04.019 ◽

2005 ◽

Vol 60 (6) ◽

pp. 791-795 ◽

Cited By ~ 6

Author(s):

Y. Liu ◽

J.N. Chen ◽

J.S. Zhao ◽

H.X. Yu ◽

X.D. Wang ◽

...

Keyword(s):

Hepg2 Cells ◽

Three Dimensional ◽

3D Qsar ◽

Quantitative Structure Activity Relationship ◽

Activity Relationship ◽

In Vitro Toxicity ◽

Quantitative Structure ◽

Qsar Analysis ◽

Structure Activity

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Study on the Three-dimensional Quantitative Structure-activity Relationship of Pyridazinonyl-substituted 1,3,4-Thiadiazoles

Chinese Journal of Chemistry ◽

10.1002/cjoc.200591120 ◽

2005 ◽

Vol 23 (8) ◽

pp. 1120-1122 ◽

Cited By ~ 4

Author(s):

Zou Xia-Juan ◽

Lai Lu-Hua ◽

Jin Gui-Yu

Keyword(s):

Three Dimensional ◽

Quantitative Structure Activity Relationship ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Quantitative Structure ◽

Structure Activity ◽

Relationship Of

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Three-Dimensional Quantitative Structure-Activity Relationship of ArylalkylamineN-acetyltransferase (AANAT) Inhibitors: A Comparative Molecular Field Analysis

Quantitative Structure-Activity Relationships ◽

10.1002/1521-3838(200112)20:5/6<414::aid-qsar414>3.0.co;2-v ◽

2001 ◽

Vol 20 (5-6) ◽

pp. 414-421 ◽

Cited By ~ 2

Author(s):

Philippe Chavatte ◽

Saïd Yous ◽

Nathalie Beaurain ◽

Christophe Mésangeau ◽

Gilles Ferry ◽

...

Keyword(s):

Three Dimensional ◽

Quantitative Structure Activity Relationship ◽

Structure Activity Relationship ◽

Field Analysis ◽

Molecular Field ◽

Activity Relationship ◽

Comparative Molecular Field Analysis ◽

Quantitative Structure ◽

Structure Activity ◽

Relationship Of

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3D-QSAR(Three-Dimensional Quantitative Structure)-Activity Relationship Of Angiotensin-Converting Enzyme And Thermolysin Inhibitors. II. A Comparison Of CoMFA Models Incorporating Molecular Orbital Fields And Desolvation Free Energies Based On Active-Analog And Complementary-Receptor-Field Alignment Rules

Journal of Medicinal Chemistry ◽

10.1021/jm00068a017 ◽

1993 ◽

Vol 36 (16) ◽

pp. 2390-2403 ◽

Cited By ~ 54

Author(s):

Chris L. Waller ◽

Garland R. Marshall

Keyword(s):

Three Dimensional ◽

3D Qsar ◽

Quantitative Structure Activity Relationship ◽

Converting Enzyme ◽

Quantitative Structure ◽

Free Energies ◽

Receptor Field ◽

Active Analog ◽

Structure Activity ◽

Relationship Of

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Three Dimensional Quantitative Structure-Activity Relationship of 5H-Pyrido[4,3-b]indol-4-carboxamide JAK2 Inhibitors

International Journal of Molecular Sciences ◽

10.3390/ijms140612037 ◽

2013 ◽

Vol 14 (6) ◽

pp. 12037-12053 ◽

Cited By ~ 2

Author(s):

Xiaoyun Wu ◽

Shanhe Wan ◽

Jiajie Zhang

Keyword(s):

Three Dimensional ◽

Quantitative Structure Activity Relationship ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Quantitative Structure ◽

Structure Activity ◽

Relationship Of ◽

Jak2 Inhibitors

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Three-Dimensional Quantitative Structure−Activity Relationship of 1,4-Dihydropyridines As Antitubercular Agents

Journal of Medicinal Chemistry ◽

10.1021/jm020217z ◽

2002 ◽

Vol 45 (22) ◽

pp. 4858-4867 ◽

Cited By ~ 68

Author(s):

Prashant S. Kharkar ◽

Bhavik Desai ◽

Harsukh Gaveria ◽

Bharat Varu ◽

Rajesh Loriya ◽

...

Keyword(s):

Three Dimensional ◽

Quantitative Structure Activity Relationship ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Quantitative Structure ◽

Antitubercular Agents ◽

Structure Activity ◽

Relationship Of

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Three-Dimensional Quantitative Structure—Activity Relationship of Nucleosides Acting at the A3 Adenosine Receptor: Analysis of Binding and Relative Efficacy.

ChemInform ◽

10.1002/chin.200734215 ◽

2007 ◽

Vol 38 (34) ◽

Author(s):

Soo-Kyung Kim ◽

Kenneth A. Jacobson

Keyword(s):

Adenosine Receptor ◽

Three Dimensional ◽

Quantitative Structure Activity Relationship ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Relative Efficacy ◽

Quantitative Structure ◽

Structure Activity ◽

A3 Adenosine Receptor ◽

Relationship Of

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Three-Dimensional Quantitative Structure−Activity Relationship of Melatonin Receptor Ligands: A Comparative Molecular Field Analysis Study

Journal of Medicinal Chemistry ◽

10.1021/jm960680+ ◽

1997 ◽

Vol 40 (5) ◽

pp. 739-748 ◽

Cited By ~ 28

Author(s):

Sames Sicsic ◽

Isabelle Serraz ◽

Jean Andrieux ◽

Béatrice Brémont ◽

Monique Mathé-Allainmat ◽

...

Keyword(s):

Three Dimensional ◽

Quantitative Structure Activity Relationship ◽

Field Analysis ◽

Comparative Molecular Field Analysis ◽

Quantitative Structure ◽

Melatonin Receptor ◽

Receptor Ligands ◽

Analysis Study ◽

Structure Activity ◽

Relationship Of

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Three-dimensional quantitative structure-activity relationship of human immunodeficiency virus (I) protease inhibitors. 2. Predictive power using limited exploration of alternate binding modes

Journal of Medicinal Chemistry ◽

10.1021/jm00040a013 ◽

1994 ◽

Vol 37 (14) ◽

pp. 2206-2215 ◽

Cited By ~ 80

Author(s):

Tudor I. Oprea ◽

Chris L. Waller ◽

Garland R. Marshall

Keyword(s):

Human Immunodeficiency Virus ◽

Protease Inhibitors ◽

Predictive Power ◽

Three Dimensional ◽

Quantitative Structure Activity Relationship ◽

Binding Modes ◽

Quantitative Structure ◽

Structure Activity ◽

Immunodeficiency Virus ◽

Relationship Of

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