Azaxanthene Based Selective Glucocorticoid Receptor Modulators: Design, Synthesis, and Pharmacological Evaluation of (S)-4-(5-(1-((1,3,4-Thiadiazol-2-yl)amino)-2-methyl-1-oxopropan-2-yl)-5H-chromeno[2,3-b]pyridin-2-yl)-2-fluoro-N,N-dimethylbenzamide (BMS-776532) and Its Methylene Homologue (BMS-791826)

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Hua Gong ◽  
Arthur M. Doweyko ◽  
Mark Cunningham ◽  
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Glucocorticoid Receptor ◽  
Design Synthesis ◽  
Pharmacological Evaluation ◽  
Receptor Modulators

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Serena Monticelli ◽  
Thomas Seidel ◽  
Denise Luger ◽  
Isabella Salzer ◽  
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Aminobutyric Acid ◽  
Design Synthesis ◽  
Pharmacological Evaluation ◽  
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Receptor Modulators

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Glucocorticoid Receptor ◽  
Next Generation ◽  
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Design, synthesis and pharmacological evaluation of tricyclic derivatives as selective RXFP4 agonists

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Guangyao Lin ◽  
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Design Synthesis ◽  
Pharmacological Evaluation

Design, Synthesis, and Pharmacological Evaluation of Glutamate Carboxypeptidase II (GCPII) Inhibitors Based on Thioalkylbenzoic Acid Scaffolds

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Pharmacological Evaluation ◽  
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ChemMedChem ◽  
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Author(s):  
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