Design, Synthesis, and Biological Evaluation of Nonsteroidal Cycloalkane[d]isoxazole-Containing Androgen Receptor Modulators

2012 ◽  
Vol 55 (14) ◽  
pp. 6316-6327 ◽  
Author(s):  
Pekka K. Poutiainen ◽  
Tuomas Oravilahti ◽  
Mikael Peräkylä ◽  
Jorma J. Palvimo ◽  
Janne A. Ihalainen ◽  
...  
Keyword(s):  
Androgen Receptor ◽  
Biological Evaluation ◽  
Design Synthesis ◽  
Receptor Modulators ◽  
Synthesis And Biological Evaluation

Design, Synthesis, and Biological Evaluation of 16-Substituted 4-Azasteroids as Tissue-Selective Androgen Receptor Modulators (SARMs)

2009 ◽  
Vol 52 (15) ◽  
pp. 4578-4581 ◽  
Author(s):  
Helen J. Mitchell ◽  
William P. Dankulich ◽  
George D. Hartman ◽  
Thomayant Prueksaritanont ◽  
Azriel Schmidt ◽  
...  
Keyword(s):  
Androgen Receptor ◽  
Biological Evaluation ◽  
Design Synthesis ◽  
Selective Androgen Receptor Modulators ◽  
Receptor Modulators ◽  
Synthesis And Biological Evaluation

Synthesis and Biological Evaluation of Second-Generation Tropanol-Based Androgen Receptor Modulators

2015 ◽  
Vol 58 (3) ◽  
pp. 1569-1574 ◽  
Author(s):  
Henrik Sundén ◽  
Mareike C. Holland ◽  
Pekka K. Poutiainen ◽  
Tiina Jääskeläinen ◽  
Juha T. Pulkkinen ◽  
...  
Keyword(s):  
Androgen Receptor ◽  
Second Generation ◽  
Biological Evaluation ◽  
Receptor Modulators ◽  
Synthesis And Biological Evaluation

Design, synthesis, and biological evaluation of 2-(5-methyl-1H-pyrazol-1-yl) acetamide derivatives as androgen receptor antagonists

2019 ◽  
Vol 28 (3) ◽  
pp. 380-386
Author(s):  
Junze Dong ◽  
Jingya Zhang ◽  
Zilu Li ◽  
Solomon Asnake ◽  
Daoguang Zhang ◽  
...  
Keyword(s):  
Androgen Receptor ◽  
Biological Evaluation ◽  
Receptor Antagonists ◽  
Design Synthesis ◽  
Synthesis And Biological Evaluation ◽  
Androgen Receptor Antagonists

Design, synthesis, and biological evaluation of 3-aryl-3-hydroxy-1-phenylpyrrolidine derivatives as novel androgen receptor antagonists

2013 ◽  
Vol 21 (1) ◽  
pp. 70-83 ◽  
Author(s):  
Satoshi Yamamoto ◽  
Hiromi Kobayashi ◽  
Tomohiro Kaku ◽  
Katsuji Aikawa ◽  
Takahito Hara ◽  
...  
Keyword(s):  
Androgen Receptor ◽  
Biological Evaluation ◽  
Receptor Antagonists ◽  
Design Synthesis ◽  
Synthesis And Biological Evaluation ◽  
Androgen Receptor Antagonists

Design, synthesis, and biological evaluation of 4-arylmethyl-1-phenylpyrazole and 4-aryloxy-1-phenylpyrazole derivatives as novel androgen receptor antagonists

2012 ◽  
Vol 20 (7) ◽  
pp. 2338-2352 ◽  
Author(s):  
Satoshi Yamamoto ◽  
Naoki Tomita ◽  
Yuri Suzuki ◽  
Tomohiko Suzaki ◽  
Tomohiro Kaku ◽  
...  
Keyword(s):  
Androgen Receptor ◽  
Biological Evaluation ◽  
Receptor Antagonists ◽  
Design Synthesis ◽  
Synthesis And Biological Evaluation ◽  
Androgen Receptor Antagonists

Design, synthesis and biological evaluation of novel 5-oxo-2-thioxoimidazolidine derivatives as potent androgen receptor antagonists

2015 ◽  
Vol 99 ◽  
pp. 51-66 ◽  
Author(s):  
Alexandre V. Ivachtchenko ◽  
Yan A. Ivanenkov ◽  
Oleg D. Mitkin ◽  
Anton A. Vorobiev ◽  
Irina V. Kuznetsova ◽  
...  
Keyword(s):  
Androgen Receptor ◽  
Biological Evaluation ◽  
Receptor Antagonists ◽  
Design Synthesis ◽  
Synthesis And Biological Evaluation ◽  
Androgen Receptor Antagonists

scholarly journals New Generation of Selective Androgen Receptor Degraders: Our Initial Design, Synthesis, and Biological Evaluation of New Compounds with Enzalutamide-Resistant Prostate Cancer Activity

2018 ◽  
Vol 62 (2) ◽  
pp. 491-511 ◽  
Author(s):  
Dong-Jin Hwang ◽  
Yali He ◽  
Suriyan Ponnusamy ◽  
Michael L. Mohler ◽  
Thirumagal Thiyagarajan ◽  
...  
Keyword(s):  
Prostate Cancer ◽  
Androgen Receptor ◽  
Biological Evaluation ◽  
Design Synthesis ◽  
Initial Design ◽  
New Generation ◽  
New Compounds ◽  
Synthesis And Biological Evaluation ◽  
Cancer Activity

Design, synthesis and biological evaluation of novel indole-xanthendione hybrids as selective estrogen receptor modulators

2018 ◽  
Vol 26 (1) ◽  
pp. 266-277 ◽  
Author(s):  
Ramit Singla ◽  
Kunj Bihari Gupta ◽  
Shishir Upadhyay ◽  
Monisha Dhiman ◽  
Vikas Jaitak
Keyword(s):  
Estrogen Receptor ◽  
Selective Estrogen Receptor Modulators ◽  
Biological Evaluation ◽  
Design Synthesis ◽  
Estrogen Receptor Modulators ◽  
Receptor Modulators ◽  
Synthesis And Biological Evaluation
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