Design, synthesis and biological evaluation of novel indole-xanthendione hybrids as selective estrogen receptor modulators

2018 ◽  
Vol 26 (1) ◽  
pp. 266-277 ◽  
Author(s):  
Ramit Singla ◽  
Kunj Bihari Gupta ◽  
Shishir Upadhyay ◽  
Monisha Dhiman ◽  
Vikas Jaitak
Keyword(s):  
Estrogen Receptor ◽  
Selective Estrogen Receptor Modulators ◽  
Biological Evaluation ◽  
Design Synthesis ◽  
Estrogen Receptor Modulators ◽  
Receptor Modulators ◽  
Synthesis And Biological Evaluation

ChemInform Abstract: Design, Synthesis and Bioevaluation of Novel Candidate Selective Estrogen Receptor Modulators.

ChemInform ◽  
2011 ◽  
Vol 43 (4) ◽  
pp. no-no
Author(s):  
Yogesh Yadav ◽  
Erin D. MacLean ◽  
Annyt Bhattacharyya ◽  
Virinder S. Parmar ◽  
Jan Balzarini ◽  
...  
Keyword(s):  
Estrogen Receptor ◽  
Selective Estrogen Receptor Modulators ◽  
Design Synthesis ◽  
Estrogen Receptor Modulators ◽  
Receptor Modulators

Design, synthesis, anti-proliferative evaluation and docking studies of 1H-1,2,3-triazole tethered ospemifene–isatin conjugates as selective estrogen receptor modulators

2018 ◽  
Vol 42 (5) ◽  
pp. 3703-3713 ◽  
Author(s):  
Sumit Kumar ◽  
Liang Gu ◽  
Gabriella Palma ◽  
Mandeep Kaur ◽  
Ashona Singh-Pillay ◽  
...  
Keyword(s):  
Estrogen Receptor ◽  
Cell Lines ◽  
Selective Estrogen Receptor Modulators ◽  
Docking Studies ◽  
Design Synthesis ◽  
Estrogen Receptor Modulators ◽  
Receptor Modulators ◽  
Mcf 7

A library of 1H-1,2,3-triazole-tethered ospemifene–isatin and ospemifene–spiroisatin conjugates have been synthesized and evaluated for their anti-proliferative activities against MCF-7 and MDA-MB-231 cell lines.

scholarly journals Design, synthesis and bioevaluation of novel candidate selective estrogen receptor modulators

2011 ◽  
Vol 46 (9) ◽  
pp. 3858-3866 ◽  
Author(s):  
Yogesh Yadav ◽  
Erin D. MacLean ◽  
Annyt Bhattacharyya ◽  
Virinder S. Parmar ◽  
Jan Balzarini ◽  
...  
Keyword(s):  
Estrogen Receptor ◽  
Selective Estrogen Receptor Modulators ◽  
Design Synthesis ◽  
Estrogen Receptor Modulators ◽  
Receptor Modulators
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