Design, Synthesis, In Vitro, and In Vivo Characterization of Phenylpiperazines and Pyridinylpiperazines as Potent and Selective Antagonists of the Melanocortin-4 Receptor

2007 ◽  
Vol 50 (25) ◽  
pp. 6356-6366 ◽  
Author(s):  
Joe A. Tran ◽  
Wanlong Jiang ◽  
Fabio C. Tucci ◽  
Beth A. Fleck ◽  
Jenny Wen ◽  
...  
Keyword(s):  
Design Synthesis ◽  
Selective Antagonists ◽  
Melanocortin 4 Receptor ◽  
In Vivo Characterization

scholarly journals Design, synthesis, and in vitro and in vivo characterization of 1-{4-[4-(substituted)piperazin-1-yl]butyl}guanidines and their piperidine analogues as histamine H3 receptor antagonists

MedChemComm ◽  
2019 ◽  
Vol 10 (2) ◽  
pp. 234-251 ◽  
Author(s):  
Marek Staszewski ◽  
Anna Stasiak ◽  
Tadeusz Karcz ◽  
Daniel McNaught Flores ◽  
Wiesława Agnieszka Fogel ◽  
...  
Keyword(s):  
Receptor Antagonists ◽  
Design Synthesis ◽  
Histamine H3 Receptor ◽  
H3 Receptor ◽  
In Vivo Characterization ◽  
Histamine H3

The prominent members of 1-{4-[4-(substituted)piperazin-1-yl]butyl}guanidines as histamine H3 receptor antagonists.

scholarly journals Design, Synthesis, In Vitro and In Vivo Characterization of Selective NKCC1 Inhibitors for the Treatment of Core Symptoms in Down Syndrome

2021 ◽  
Author(s):  
Marco Borgogno ◽  
Annalisa Savardi ◽  
Jacopo Manigrasso ◽  
Alessandra Turci ◽  
Corinne Portioli ◽  
...  
Keyword(s):  
Down Syndrome ◽  
Design Synthesis ◽  
Core Symptoms ◽  
In Vivo Characterization

In vitro and in vivo characterization of graphene oxide coated porcine bone granules

Carbon ◽  
2016 ◽  
Vol 103 ◽  
pp. 291-298 ◽  
Author(s):  
Valeria Ettorre ◽  
Patrizia De Marco ◽  
Susi Zara ◽  
Vittoria Perrotti ◽  
Antonio Scarano ◽  
...  
Keyword(s):  
Graphene Oxide ◽  
In Vivo Characterization

P.3.d.011 In vitro and in vivo characterization of glycine transporter type-1 by two inhibitors, Org-24461 and NFPS

2006 ◽  
Vol 16 ◽  
pp. S435 ◽  
Author(s):  
B. Marko ◽  
G. Szabo ◽  
S. Udvari ◽  
M. Agoston ◽  
E. Szabo ◽  
...  
Keyword(s):  
Glycine Transporter ◽  
In Vivo Characterization

scholarly journals Correction to “Improving Paclitaxel Delivery: In Vitro and In Vivo Characterization of PEGylated Polyphosphoester-Based Nanocarriers”

2015 ◽  
Vol 137 (21) ◽  
pp. 6972-6972 ◽  
Author(s):  
Fuwu Zhang ◽  
Shiyi Zhang ◽  
Stephanie F. Pollack ◽  
Richen Li ◽  
Amelia M. Gonzalez ◽  
...  
Keyword(s):  
In Vivo Characterization

Synthesis, in vitro and in vivo characterization of novel 99mTc-‘4+1’-labeled 5-nitroimidazole derivatives as potential agents for imaging hypoxia

2012 ◽  
Vol 39 (5) ◽  
pp. 679-686 ◽  
Author(s):  
Javier Giglio ◽  
Soledad Fernández ◽  
Hans-Jürgen Pietzsch ◽  
Sylvia Dematteis ◽  
María Moreno ◽  
...  
Keyword(s):  
In Vivo Characterization

scholarly journals In vitro and in vivo characterization of new swine-origin H1N1 influenza viruses

Nature ◽  
2009 ◽  
Vol 460 (7258) ◽  
pp. 1021-1025 ◽  
Author(s):  
Yasushi Itoh ◽  
Kyoko Shinya ◽  
Maki Kiso ◽  
Tokiko Watanabe ◽  
Yoshihiro Sakoda ◽  
...  
Keyword(s):  
H1n1 Influenza ◽  
Influenza Viruses ◽  
In Vivo Characterization

In vivo characterization of estrogen receptor modulators with reduced genomic versus nongenomic activity in vitro

2008 ◽  
Vol 111 (1-2) ◽  
pp. 95-100 ◽  
Author(s):  
Christiane Otto ◽  
Iris Fuchs ◽  
Helga Altmann ◽  
Mario Klewer ◽  
Gilda Schwarz ◽  
...  
Keyword(s):  
Estrogen Receptor ◽  
Estrogen Receptor Modulators ◽  
In Vivo Characterization ◽  
Receptor Modulators
Sign in / Sign up

Export Citation Format

Share Document