scholarly journals Potent and selective bivalent inhibitors of BET bromodomains

2016 ◽  
Vol 12 (12) ◽  
pp. 1097-1104 ◽  
Author(s):  
Michael J Waring ◽  
Huawei Chen ◽  
Alfred A Rabow ◽  
Graeme Walker ◽  
Romel Bobby ◽  
...  
Keyword(s):  
Bivalent Inhibitors

Novel bivalent inhibitors with sub-nanomolar affinities towards human glyoxalase I

2015 ◽  
Vol 25 (21) ◽  
pp. 4724-4727 ◽  
Author(s):  
Yankui Sang ◽  
Qing Shi ◽  
Mingguang Mo ◽  
Caixia Ni ◽  
Zonghe Li ◽  
...  
Keyword(s):  
Glyoxalase I ◽  
Bivalent Inhibitors

scholarly journals Bivalent inhibitors of protein kinases

2014 ◽  
Vol 49 (2) ◽  
pp. 102-115 ◽  
Author(s):  
Carrie M. Gower ◽  
Matthew E. K. Chang ◽  
Dustin J. Maly
Keyword(s):  
Protein Kinases ◽  
Bivalent Inhibitors

Synthesis of bivalent inhibitors of eucaryotic proteasomes

2000 ◽  
Vol 6 (1) ◽  
pp. 36-46 ◽  
Author(s):  
G�nther Loidl ◽  
Hans-J�rgen Musiol ◽  
Michael Groll ◽  
Robert Huber ◽  
Luis Moroder
Keyword(s):  
Bivalent Inhibitors

scholarly journals Conversion of a Single Polypharmacological Agent into Selective Bivalent Inhibitors of Intracellular Kinase Activity

2015 ◽  
Vol 11 (1) ◽  
pp. 121-131 ◽  
Author(s):  
Carrie M. Gower ◽  
Jason R. Thomas ◽  
Edmund Harrington ◽  
Jason Murphy ◽  
Matthew E. K. Chang ◽  
...  
Keyword(s):  
Kinase Activity ◽  
Bivalent Inhibitors

scholarly journals A rapid oxime linker-based library approach to identification of bivalent inhibitors of the Yersinia pestis protein-tyrosine phosphatase, YopH

2010 ◽  
Vol 20 (9) ◽  
pp. 2813-2816 ◽  
Author(s):  
Fa Liu ◽  
Ramin Mollaaghababa Hakami ◽  
Beverly Dyas ◽  
Medhanit Bahta ◽  
George T. Lountos ◽  
...  
Keyword(s):  
Yersinia Pestis ◽  
Protein Tyrosine Phosphatase ◽  
Tyrosine Phosphatase ◽  
Protein Tyrosine ◽  
Bivalent Inhibitors

Progesterone–adenine hybrids as bivalent inhibitors of P-glycoprotein-mediated multidrug efflux: Design, synthesis, characterization and biological evaluation

Steroids ◽  
2012 ◽  
Vol 77 (12) ◽  
pp. 1177-1191 ◽  
Author(s):  
Waël Zeinyeh ◽  
Zahia Mahiout ◽  
Sylvie Radix ◽  
Thierry Lomberget ◽  
Axel Dumoulin ◽  
...  
Keyword(s):  
Biological Evaluation ◽  
Multidrug Efflux ◽  
Design Synthesis ◽  
P Glycoprotein ◽  
Bivalent Inhibitors
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