scholarly journals Pyrazolyl-pyrimidones inhibit the function of human solute carrier protein SLC11A2 (hDMT1) by metal chelation

2020 ◽  
Vol 11 (9) ◽  
pp. 1023-1031
Author(s):  
Marion Poirier ◽  
Jonai Pujol-Giménez ◽  
Cristina Manatschal ◽  
Sven Bühlmann ◽  
Ahmed Embaby ◽  
...  

Activity optimization of a pyrazolyl-pyrimidone against the iron transporter SLC11A2 (hDMT1) and mechanistic studies revealed that this class of inhibitors act by metal chelation.

2013 ◽  
Vol 105 (8) ◽  
pp. 1822-1828 ◽  
Author(s):  
Oluwarotimi Okunade ◽  
Joseph Santos-Sacchi

2016 ◽  
Vol 41 (3) ◽  
pp. 671-677 ◽  
Author(s):  
Nisha Singh ◽  
Mallikarjuna Rao Gedda ◽  
Neeraj Tiwari ◽  
Suya P. Singh ◽  
Surabhi Bajpai ◽  
...  

1994 ◽  
Vol 1189 (1) ◽  
pp. 52-60 ◽  
Author(s):  
Judith K Woodford ◽  
Ivan Hapala ◽  
John R Jefferson ◽  
James J Knittel ◽  
Juraj Kavecansky ◽  
...  

2018 ◽  
Vol 1689 ◽  
pp. 30-44 ◽  
Author(s):  
Kojiro Suda ◽  
Ibuki Ueoka ◽  
Yumiko Azuma ◽  
Yuuka Muraoka ◽  
Hideki Yoshida ◽  
...  

2007 ◽  
Vol 35 (7) ◽  
pp. 1239-1245 ◽  
Author(s):  
Yasuna Kobayashi ◽  
Ayumi Tsuchiya ◽  
Tomofumi Hayashi ◽  
Noriko Kohyama ◽  
Masayuki Ohbayashi ◽  
...  

Theranostics ◽  
2021 ◽  
Vol 11 (20) ◽  
pp. 9752-9771
Author(s):  
Arun Pandian Chandrasekaran ◽  
Kamini Kaushal ◽  
Chang-Hwan Park ◽  
Kye-Seong Kim ◽  
Suresh Ramakrishna

2008 ◽  
Vol 75 (10) ◽  
pp. 1495-1504 ◽  
Author(s):  
Kazuyuki Hiratsuka ◽  
Shan-Ai Yin ◽  
Takayuki Ohtomo ◽  
Mariko Fujita ◽  
Kazutoshi Ohtsuki ◽  
...  

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