Effects of Imidafenacin (KRP-197/ONO-8025), a New Anti-cholinergic Agent, on Muscarinic Acetylcholine Receptors

Arzneimittelforschung ◽

10.1055/s-0031-1296589 ◽

2011 ◽

Vol 57 (02) ◽

pp. 92-100 ◽

Author(s):

Fumiyoshi Kobayashi ◽

Yuichi Yageta ◽

Mitsuru Segawa ◽

Shigeki Matsuzawa

Keyword(s):

Acetylcholine Receptors ◽

Muscarinic Acetylcholine Receptors ◽

Muscarinic Acetylcholine ◽

Cholinergic Agent

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Molecular Biology of Muscarinic Acetylcholine Receptors

Critical Reviews in Neurobiology ◽

10.1615/critrevneurobiol.v10.i1.40 ◽

1996 ◽

Vol 10 (1) ◽

pp. 69-99 ◽

Author(s):

Jurgen Wess

Keyword(s):

Molecular Biology ◽

Acetylcholine Receptors ◽

Muscarinic Acetylcholine Receptors ◽

Muscarinic Acetylcholine

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Faculty Opinions recommendation of Muscarinic acetylcholine receptors chrm1 and chrm3 are essential for REM sleep.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.733874636.793572509 ◽

2020 ◽

Author(s):

Paul Franken

Keyword(s):

Rem Sleep ◽

Acetylcholine Receptors ◽

Muscarinic Acetylcholine Receptors ◽

Muscarinic Acetylcholine

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Bioisosteric Replacement and Related Analogs in the Design, Synthesis and Evaluation of Ligands for Muscarinic Acetylcholine Receptors

Medicinal Chemistry ◽

10.2174/15734064113096660043 ◽

2014 ◽

Vol 10 (4) ◽

pp. 361-375 ◽

Author(s):

Richie Bhandare ◽

Daniel Canney

Keyword(s):

Acetylcholine Receptors ◽

Muscarinic Acetylcholine Receptors ◽

Design Synthesis ◽

Muscarinic Acetylcholine ◽

Bioisosteric Replacement

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Pharmacological Approaches to Targeting Muscarinic Acetylcholine Receptors

Recent Patents on CNS Drug Discovery ◽

10.2174/1574889809666141120131238 ◽

2014 ◽

Vol 9 (2) ◽

pp. 85-100 ◽

Author(s):

Carlo Matera ◽

Ada Tata

Keyword(s):

Acetylcholine Receptors ◽

Muscarinic Acetylcholine Receptors ◽

Muscarinic Acetylcholine

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In Silico Analysis of Binding Interaction of Mamba Toxins with M4 and M2 Muscarinic Acetylcholine Receptors for Therapeutic Use in Alzheimer’s Disease

CNS & Neurological Disorders - Drug Targets ◽

10.2174/1871527314666150821105816 ◽

2015 ◽

Vol 14 (8) ◽

pp. 1031-1040 ◽

Author(s):

Maleeha Waqar ◽

Mohammad Kamal ◽

Sidra Batool

Keyword(s):

Alzheimer’S Disease ◽

Alzheimer's Disease ◽

In Silico ◽

Acetylcholine Receptors ◽

In Silico Analysis ◽

Therapeutic Use ◽

Muscarinic Acetylcholine Receptors ◽

Binding Interaction ◽

Muscarinic Acetylcholine ◽

Silico Analysis

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Characterization of the subtype selectivity of the allosteric modulator, C7/3-phth, at cloned muscarinic acetylcholine receptors

Life Sciences ◽

10.1016/s0024-3205(99)90478-2 ◽

1999 ◽

Vol 64 (6-7) ◽

pp. 561

Author(s):

E.E. El-Fakahany ◽

A. Christopoulos ◽

J.L. Sorman ◽

F. Mitchelson

Keyword(s):

Acetylcholine Receptors ◽

Muscarinic Acetylcholine Receptors ◽

Allosteric Modulator ◽

Muscarinic Acetylcholine ◽

Subtype Selectivity

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Functional role in ligand binding and receptor activation of an asparagine residue present in the sixth transmembrane domain of all muscarinic acetylcholine receptors.

Journal of Biological Chemistry ◽

10.1016/s0021-9258(17)32248-2 ◽

1994 ◽

Vol 269 (29) ◽

pp. 18870-18876

Author(s):

K. Blüml ◽

E. Mutschler ◽

J. Wess

Keyword(s):

Ligand Binding ◽

Acetylcholine Receptors ◽

Functional Role ◽

Transmembrane Domain ◽

Receptor Activation ◽

Muscarinic Acetylcholine Receptors ◽

Muscarinic Acetylcholine ◽

Asparagine Residue

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Evidence for a tandem two-site model of ligand binding to muscarinic acetylcholine receptors. Vol. 275 (2000) 18836-18844

Journal of Biological Chemistry ◽

10.1016/s0021-9258(20)77092-4 ◽

2004 ◽

Vol 279 (41) ◽

pp. 43361

Author(s):

Jan Jakubík ◽

Esam E. El-Fakahany ◽

Stanislav Tuček

Keyword(s):

Ligand Binding ◽

Acetylcholine Receptors ◽

Muscarinic Acetylcholine Receptors ◽

Muscarinic Acetylcholine ◽

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Pulmonary Microcirculation during Experimental Pulmonary Thromboembolism under Conditions of Activation and Blockade of Muscarinic Acetylcholine Receptors

Bulletin of Experimental Biology and Medicine ◽

10.1007/s10517-021-05194-4 ◽

2021 ◽

Author(s):

V. I. Evlakhov ◽

T. P. Berezina ◽

I. Z. Poyassov ◽

V. I. Ovsyannikov

Keyword(s):

Acetylcholine Receptors ◽

Pulmonary Thromboembolism ◽

Muscarinic Acetylcholine Receptors ◽

Muscarinic Acetylcholine ◽

Pulmonary Microcirculation

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Neuroactive steroids, WIN-compounds and cholesterol share a common binding site on muscarinic acetylcholine receptors

Biochemical Pharmacology ◽

10.1016/j.bcp.2021.114699 ◽

2021 ◽

pp. 114699

Author(s):

Eva Dolejší ◽

Nikolai Chetverikov ◽

Eszter Szánti-Pintér ◽

Dominik Nelic ◽

Alena Randáková ◽

...

Keyword(s):

Binding Site ◽

Acetylcholine Receptors ◽

Muscarinic Acetylcholine Receptors ◽

Neuroactive Steroids ◽

Muscarinic Acetylcholine

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