Synthesis of Borylated Hydrazino Acid Derivatives
Abstractα-Boryl-α-hydrazinoacetic acid is a highly functionalized boron-containing building block that can be easily accessed from readily available α-borylacetaldehyde. The hydrazine motif can be converted into a variety of α-borylated azoles and diazines in a straightforward protocol. Furthermore, the carboxy group can be derivatized to afford novel organoboron compounds that should find applications in various cross-coupling transformations.
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2001 ◽
Vol 74
(2)
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pp. 371-376
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2018 ◽
Vol 6
(8)
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pp. 2148-2154
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Keyword(s):